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(3aS,6aS)-2-methyl-5-{[5-(methylcarbamoyl)thiophen-3-yl]sulfonyl}-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
3-{3-[4-methyl-5-(morpholin-4-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}propan-1-ol
6-(morpholin-4-yl)-N-{pyrazolo[1,5-a]pyridin-3-ylmethyl}pyridine-3-sulfonamide
N-[(dimethyl-1,2-oxazol-4-yl)methyl]-2-(1H-1,2,4-triazol-3-yl)benzamide
4-{[3-(2-aminoethyl)phenyl]methyl}-1-(4-methoxyphenyl)-3-methylpiperazin-2-one
N-(oxolan-2-ylmethyl)-3-(pyridin-2-yl)-N-(thiophen-3-ylmethyl)-1H-pyrazole-5-carboxamide
2-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-4-[4-(thiomorpholine-4-carbonyl)piperidin-1-yl]-2,3-dihydro-1H-isoindole-1,3-dione
3-ethyl-1-(3-methylbutyl)-8-[(2E)-3-phenylprop-2-en-1-yl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-(adamantan-1-yl)-N-{[3-(pyrimidin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}acetamide
5-[1-(benzenesulfonyl)cyclopropyl]-3-benzyl-1H-1,2,4-triazole
[1-(2,3-dihydro-1,4-benzodioxin-6-yl)ethyl][(1,2-dimethyl-1H-imidazol-5-yl)methyl]methylamine
4-chloro-N-[(3R,5S)-5-(ethylcarbamoyl)-1-(1H-imidazol-2-ylmethyl)pyrrolidin-3-yl]-1-methyl-1H-pyrazole-5-carboxamide
5-ethyl-4-[3-(3-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-2-methylpyrimidine
3-(1-{[1-(pyridin-3-yl)-1H-pyrrol-2-yl]methyl}piperidin-3-yl)-1-(pyrrolidin-1-yl)propan-1-one
1-(5-chloro-2-fluorobenzoyl)-4-[(2-methylphenyl)methyl]-1,4-diazepan-5-one
N-{[1-(1-phenylcyclopropanecarbonyl)piperidin-3-yl]methyl}thiophene-2-sulfonamide
7-(oxan-4-yl)-2-[2-(2-oxo-1,2-dihydropyridin-1-yl)acetyl]-2,7-diazaspiro[4.5]decan-6-one
2,4-dimethyl-6-[3-(phenoxymethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]pyrimidine
2-{[4-(6-aminopyridin-3-yl)-1H-pyrrolo[2,3-b]pyridin-6-yl]amino}ethan-1-ol
5-(2-methylphenyl)-2-(pyridin-4-yl)-4-[1-(thiophen-3-ylmethyl)piperidin-3-yl]pyrimidine
4-(1H-1,3-benzodiazol-1-yl)-1-(pyridine-3-carbonyl)piperidine-4-carboxylic acid
dimethyl(2-{3-[3-(3-methylpyridin-2-yl)phenyl]-1H-pyrazol-1-yl}ethyl)amine
N-cyclobutyl-3-[(oxan-3-ylmethyl)sulfamoyl]benzamide
2-methoxy-N-[3-(1-methyl-1H-pyrazol-4-yl)phenyl]acetamide
N-ethyl-1-(2-methoxyphenyl)-N-(pyridin-4-ylmethyl)-1H-pyrazole-4-carboxamide
3-[(1-{imidazo[2,1-b][1,3]thiazole-6-carbonyl}pyrrolidin-3-yl)methyl]benzoic acid
3-{3-[4-(4-fluorophenyl)-1H-pyrazol-5-yl]piperidine-1-carbonyl}-1,6-dimethyl-1,2-dihydropyridin-2-one
8-[(2,6-difluorophenyl)methyl]-2-(3-phenylpropyl)-2,8-diazaspiro[4.5]decan-3-one
3-(3-fluoro-4-phenylbenzoyl)-1-(propane-2-sulfonyl)piperidine
N-[1-(azepan-1-yl)-2-methylpropan-2-yl]pyrimidin-4-amine
4-({7,11-dimethyl-3,7,11-triazaspiro[5.6]dodecan-3-yl}methyl)benzoic acid
2-[1-(cyclopropylmethyl)-4-[2-(dimethylamino)-4-methylpyrimidine-5-carbonyl]piperazin-2-yl]ethan-1-ol
1-(carbamoylmethyl)-N-ethyl-N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperidine-4-carboxamide
2-amino-3-ethyl-N-(2-{5H,6H,7H-[1,3]thiazolo[3,2-a]pyrimidin-3-yl}ethyl)-3H-imidazo[4,5-b]pyridine-6-carboxamide
N-[(3R,4S)-1-acetyl-4-(propan-2-yl)pyrrolidin-3-yl]-2-acetamido-2-methylpropanamide
[(3R,4R)-1-[4-(dimethylamino)-5-methylpyrimidin-2-yl]-4-{[4-(hydroxymethyl)piperidin-1-yl]methyl}pyrrolidin-3-yl]methanol
N-[(7S,8aS)-2-methyl-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-methyl-6-(propan-2-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
methyl 3-benzamido-5-[(2-methylpropyl)amino]-1-(oxolan-2-ylmethyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
2-[(1-{5H,6H,7H,8H-imidazo[1,5-a]pyrazin-7-yl}-1-oxopropan-2-yl)sulfanyl]-6-methyl-3,4-dihydropyrimidin-4-one
(oxolan-2-ylmethyl)({[3-(pyrimidin-2-yloxy)phenyl]methyl})(thiophen-3-ylmethyl)amine
{[5-({4-[1-(dimethylamino)ethyl]piperidin-1-yl}methyl)thiophen-3-yl]methyl}dimethylamine
2-methyl-6-{2-[(4-methyl-1H-imidazol-2-yl)methyl]-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-1-yl}pyridine
N-{[7-methoxy-2-(3-methylphenyl)quinolin-3-yl]methyl}-N-(2-methoxyethyl)-1,3-dimethyl-1H-pyrazole-5-carboxamide
2-methyl-N-[2-(morpholin-4-yl)-2-(pyridin-4-yl)ethyl]-2-(thiophen-2-ylformamido)propanamide
3-[(3R,4S)-1-(5-ethylthiophene-3-carbonyl)-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propan-1-ol
2-(3-fluorophenyl)-N-[(7-{[4-(furan-2-yl)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)methyl]acetamide
2-[(2R)-2-hydroxypropanoyl]-N-(pyridin-3-yl)-1,2,3,4-tetrahydroisoquinoline-7-sulfonamide
2-methyl-3-[3-(methylsulfanyl)phenyl]-6-(4H-1,2,4-triazol-4-yl)pyridine
1-(4-methoxyphenyl)-2,2-dimethyl-4-[1-(1H-pyrazol-1-ylmethyl)cyclopropanecarbonyl]piperazine
2-[(2-methylpiperidin-1-yl)methyl]-N-(thiophen-2-ylmethyl)quinazolin-4-amine