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(3R,4R)-1-[6-amino-2-(methylsulfanyl)pyrimidin-4-yl]-4-ethylpiperidine-3,4-diol
(furan-2-ylmethyl)[(4-methyloxan-4-yl)methyl](pyridin-2-ylmethyl)amine
2-(2-aminoethyl)-N-[2-(2,3-dihydro-1H-indol-1-yl)ethyl]quinazolin-4-amine
ethyl 3-[(3-chlorophenyl)methyl]-1-(1-methyl-3-propyl-1H-pyrazole-5-carbonyl)piperidine-3-carboxylate
4-[1-(1-{[4-(propan-2-yl)phenyl]methyl}piperidin-4-yl)-1H-1,2,3-triazole-4-carbonyl]morpholine
5-[(methylsulfanyl)methyl]-N-[1-(pyrimidin-2-yl)piperidin-3-yl]furan-2-carboxamide
5-cyclobutyl-3-(2-phenylethyl)-1H-1,2,4-triazole
N-[1-(3-phenylpropyl)piperidin-3-yl]pent-4-enamide
1-benzyl-3-methyl-8-(3-phenylbutyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
ethyl 2-[1-(1-methyl-1H-indole-3-carbonyl)piperidin-2-yl]acetate
1-[1-(7-fluoro-3-methyl-1-benzofuran-2-carbonyl)piperidin-3-yl]-3-methylbutan-1-one
N-cyclopropyl-4-{[3-(4-methoxyphenoxy)phenyl]methyl}piperazine-2-carboxamide
ethyl 4-{5H,6H,7H,8H,9H-imidazo[1,5-a][1,4]diazepin-8-ylmethyl}-1H-pyrazole-3-carboxylate
2-[ethyl({[(3R,4R)-4-(hydroxymethyl)-1-(5-methylpyrazine-2-carbonyl)pyrrolidin-3-yl]methyl})amino]ethan-1-ol
1-(3-methoxypropyl)-3-(naphthalen-2-ylmethyl)-8-propyl-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-(dimethylamino)-8-[2-(propylsulfanyl)pyrimidin-5-yl]-4H,5H,6H,7H,8H-[1,3]thiazolo[4,5-c]azepin-6-one
N-[3-(2-oxo-1,2-dihydropyridin-1-yl)propyl]-1H-pyrazole-4-carboxamide
N-[3-(1-methyl-1H-pyrazol-4-yl)propyl]-5-phenylpyrazolo[1,5-a]pyrimidin-7-amine
N-benzyl-3-({1-[(1-ethyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}oxy)benzamide
1-(4-tert-butylbenzoyl)-4-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]piperidine
5-{[({3-[2-(4-cyclohexanecarbonylpiperazin-1-yl)ethoxy]phenyl}methyl)(methyl)amino]methyl}pyrrolidin-2-one
N-(4,6-dimethyl-2-oxo-1,2-dihydropyridin-1-yl)-3-(1,2-oxazinan-2-yl)propanamide
3-(6-methyl-2-oxo-1,2-dihydropyridin-1-yl)-N-{[5-(thiophen-2-yl)-1,2,4-oxadiazol-3-yl]methyl}propanamide
9-{[1-(2-hydroxyethyl)-3-methyl-1H-pyrazol-4-yl]methyl}-1-oxa-9-azaspiro[5.5]undecan-5-ol
1-[2-(ethoxymethyl)-7-methyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl]-3-methoxypiperidine
3-[6-hydroxy-4-(oxan-4-yl)-1,4-diazepan-1-yl]pyrazine-2-carbonitrile
6-{[3-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-2,5-dioxo-1,2,5,6-tetrahydro-1,6-naphthyridine-3-carbonitrile
3-[4-(1,2,3,4-tetrahydronaphthalen-2-yl)piperazine-1-carbonyl]phenol
1-(azepan-1-yl)-3-(4-{[(cyclopropylmethyl)(methyl)amino]methyl}-2-methoxyphenoxy)propan-2-ol
2-[3-(2-fluorophenyl)-1H-pyrazol-1-yl]-N-[3-methyl-1-(pyridin-2-yl)-1H-pyrazol-5-yl]acetamide
3-(pyridin-3-yl)-N-({7-[2-(trifluoromethyl)phenyl]-2,3-dihydro-1-benzofuran-2-yl}methyl)propanamide
1-[5-({[2-(4-fluorophenyl)ethyl]amino}methyl)-2-methoxyphenoxy]-3-(piperidin-1-yl)propan-2-ol
2-[2-(4-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]-N-(oxolan-2-ylmethyl)acetamide
(2E)-N-({3-methyl-7-[4-(pyrrolidin-1-yl)benzoyl]-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-3-(thiophen-2-yl)prop-2-enamide
2-(3-hydroxypropyl)-8-(1H-indole-6-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
[(3R,4R)-1-{[2-methyl-4-(1H-pyrazol-1-yl)phenyl]methyl}-4-(piperidin-1-ylmethyl)pyrrolidin-3-yl]methanol
N-{[4-(methylsulfanyl)phenyl]methyl}-N-(prop-2-en-1-yl)piperidine-4-carboxamide
1-[(2,3-dimethoxyphenyl)methyl]-3-[(ethylamino)methyl]-3-hydroxypiperidin-2-one
1-(4-methoxybenzoyl)-4-[1-(1H-pyrazol-1-ylmethyl)cyclopropanecarbonyl]piperazine
2-[2-(3-benzoylpiperidin-1-yl)-2-oxoethyl]-5-(piperazin-1-yl)-2,3-dihydropyridazin-3-one
1-(3-{2-[(3-fluorophenyl)methyl]morpholin-4-yl}-3-oxopropyl)piperidin-2-one
1-[(2,6-difluorophenyl)methyl]-N-methyl-N-[(4-methylphenyl)methyl]-1H-1,2,3-triazole-4-carboxamide
3-(1-methylpiperidin-3-yl)-N-[(5-methylthiophen-2-yl)methyl]-N-(pyridin-2-ylmethyl)propanamide
1-[(1-ethyl-1H-pyrazol-4-yl)methyl]-N-[4-(1,3-thiazol-4-yl)phenyl]pyrrolidine-2-carboxamide
6-(azepan-1-yl)-N-methyl-N-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-amine
(4aR,8aR)-7-(1-benzofuran-5-ylmethyl)-4a-hydroxy-N,N-dimethyl-decahydro-2,7-naphthyridine-2-carboxamide
2-methoxy-1-[4-(5-methyl-1-propyl-1H-pyrazole-4-carbonyl)-1,4-diazepan-1-yl]ethan-1-one
1'-{[3-(furan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-1-methyl-1,2-dihydrospiro[indole-3,4'-piperidine]-2-one
1-(5-chloro-2-methoxyphenyl)-3-{[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]methyl}urea
N-(3,3-diphenylpropyl)-3-{2-[(3-methoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}propanamide