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(4aR,7aS)-1-(2-methylpropanoyl)-4-{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-[4-(4-fluorophenyl)-1,2,3,6-tetrahydropyridin-1-yl]-3-[(3S,4R)-4-[4-(2-fluorophenyl)piperazin-1-yl]-1-(pyridin-2-ylmethyl)piperidin-3-yl]propan-1-one
N-methyl-2-[2-(propan-2-yl)-1H-imidazol-1-yl]-N-{[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl}propanamide
N-({1-[(3-hydroxyphenyl)methyl]piperidin-3-yl}methyl)pyridazine-3-carboxamide
(2R,6S)-4-[6-(methoxymethyl)pyridine-2-carbonyl]-2,6-dimethylmorpholine
4-hydroxy-N-[(1R,2S)-2-(methoxymethyl)cyclopentyl]-2-(phenoxymethyl)pyrimidine-5-carboxamide
(2H-1,3-benzodioxol-5-ylmethyl)({[3-(pyridin-3-yl)phenyl]methyl})amine
[(3-ethyl-1,2-oxazol-5-yl)methyl](methyl)[(trimethyl-1H-pyrazol-4-yl)methyl]amine
2-[(1-methylpiperidin-3-yl)methyl]-2,3-dihydro-1,2-benzothiazol-3-one
1-[7-(hydroxymethyl)-3,9-diazaspiro[5.5]undecan-3-yl]-2-(3-methyl-4,5-dihydro-1H-pyrazol-1-yl)ethan-1-one
2-[3-methyl-1-(3-methylphenyl)-5-oxo-4,5-dihydro-1H-1,2,4-triazol-4-yl]-N-{2-[(3-methylpyridin-2-yl)amino]ethyl}acetamide
[(2-ethylpyrimidin-5-yl)methyl]({[2-(2-methylphenoxy)pyridin-3-yl]methyl})amine
2-methyl-6-[3-(4-phenoxybenzoyl)piperidine-1-carbonyl]-2,3-dihydropyridazin-3-one
1-{2-[(1S,5R)-3-[(4-fluorophenyl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-oxoethyl}-1,2-dihydropyridin-2-one
N-[1-(3-cyclopropyl-1,2,4-oxadiazol-5-yl)-2-methylpropyl]-1-ethyl-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
2,2-dimethyl-N-({2-[3-(trifluoromethyl)phenoxy]pyridin-3-yl}methyl)cyclopropane-1-carboxamide
(4aR,8aS)-1-[2-(methylsulfanyl)-1,3-thiazole-4-carbonyl]-6-(2-phenylethyl)-decahydro-1,6-naphthyridine
(1-{1-[(3-{[3-(trifluoromethyl)phenyl]methyl}-1,2,4-oxadiazol-5-yl)methyl]piperidin-4-yl}piperidin-3-yl)methanol
1-benzyl-N3-cyclopropyl-N5-[(4-methylphenyl)methyl]-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
3-[(3S,4R)-3,4-dihydroxy-4-methylpiperidin-1-yl]-N-(furan-2-ylmethyl)propanamide
1-methyl-N-[(5-oxopyrrolidin-2-yl)methyl]-N-(propan-2-yl)-1H-indole-3-carboxamide
1-{3-[4-(2-amino-6-methylpyrimidin-4-yl)piperazine-1-carbonyl]piperidin-1-yl}propan-1-one
6-phenyl-3-(4-phenyl-1,2,3,6-tetrahydropyridine-1-carbonyl)-1,2-dihydropyridin-2-one
4-({[5-(5-acetylthiophen-2-yl)-7-chloro-2,3-dihydro-1-benzofuran-2-yl]methyl}carbamoyl)pyridin-1-ium-1-olate
3-(2-hydroxyphenyl)-N-(2-oxo-1,2,3,4-tetrahydroquinolin-4-yl)-1H-pyrazole-5-carboxamide
2-{[(7-methoxynaphthalen-2-yl)oxy]methyl}-N-[(5-methylpyrazin-2-yl)methyl]-1,3-oxazole-4-carboxamide
N-benzyl-1-[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl]-N-methylpiperidin-3-amine
2-cyclopentyl-9-{[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-2,9-diazaspiro[5.5]undecan-3-one
5-fluoro-N4,N4-dimethyl-N2-[1-(pyridin-3-yl)pentyl]pyrimidine-2,4-diamine
{[7-chloro-2-(thiophen-3-yl)quinolin-3-yl]methyl}(methyl)(pyrimidin-4-ylmethyl)amine
4-(2-methoxyphenyl)-N-methyl-N-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]benzamide
3-{2-oxo-2-[(1S,5R)-3-(pyridine-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethyl}-1,3-oxazolidin-2-one
N-({2-[benzyl(methyl)amino]pyridin-3-yl}methyl)-5-hydroxy-4-oxo-4H-pyran-2-carboxamide
5-(2-{4-[(2-fluorophenyl)methyl]piperidin-1-yl}-2-oxoethyl)-1,3-dimethylimidazolidine-2,4-dione
7-(pyridin-3-yl)-4-[6-(trifluoromethyl)pyridin-2-yl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N-cyclooctyl-4-[4-(1-hydroxyethyl)piperidin-1-yl]-4-oxobutanamide
1-{2-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl}-N-[(2-methoxyphenyl)methyl]piperidine-3-carboxamide
N-{[2-(ethylsulfanyl)pyrimidin-5-yl]methyl}-N-methylthian-4-amine
2-{[(3S,4S)-3-carboxy-4-cyclopropylpyrrolidin-1-yl]methyl}-1,3-oxazole-4-carboxylic acid
3-{[(2-hydroxyethyl)(propyl)amino]methyl}-7-methyl-1,2-dihydroquinolin-2-one
2-methyl-N-[2-(7-{[3-(trifluoromethyl)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)ethyl]propanamide
(1R,5S,8S)-3-(trimethylpyrimidin-4-yl)-3-azabicyclo[3.2.1]octan-8-ol
6-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl}-7-methylpyrazolo[1,5-a]pyrimidine
N-(4-{[3-(4-phenylpiperazin-1-yl)piperidin-1-yl]methyl}phenyl)acetamide
methyl 3-(1,3-dimethyl-1H-pyrazole-5-amido)-5-{[(2E)-3-(3-fluorophenyl)prop-2-enamido]methyl}benzoate
methyl 1-{[(1,4-dimethyl-1H-pyrazol-5-yl)carbamoyl]methyl}-1H-indazole-3-carboxylate
4-{[1-(2-methoxyacetyl)piperidin-4-yl]oxy}-N-[3-(pyridin-3-yl)propyl]benzamide
(3S,4R)-1-[4-(azepan-1-yl)-4-oxobutanoyl]-4-phenylpyrrolidine-3-carboxylic acid
2-methyl-4-(3-{2-methyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carbonyl}phenyl)butan-2-ol
(1R,5R)-3-(5-propyl-1,2-oxazole-3-carbonyl)-3,9-diazabicyclo[3.3.2]decan-10-one