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2-(4-{[1-(2-fluorophenyl)-1H-pyrazol-4-yl]methyl}-1-methylpiperazin-2-yl)ethan-1-ol
N-(2-methyl-1-{7-[(2,4,5-trimethylphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}propyl)methanesulfonamide
N-[4-(oxolan-2-yl)butyl]-1,4-dithiepan-6-amine
N-[(2S,4R,6S)-2-[2,5-dimethoxy-4-(methylsulfanyl)phenyl]-6-ethyloxan-4-yl]acetamide
N-{1-[(2-fluorophenyl)methyl]piperidin-3-yl}-3-(morpholin-4-yl)benzamide
N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-3-(2-oxopyrrolidin-1-yl)propanamide
8-[(4-chloro-2-fluorophenyl)methyl]-1-methyl-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
1-(6-methyl-2-phenylpyrimidin-4-yl)-N-[2-(pyrazin-2-yl)ethyl]piperidin-4-amine
1-{4-[hydroxy(1-methyl-1H-imidazol-2-yl)methyl]piperidin-1-yl}-2-(2,5,7-trimethyl-1H-indol-3-yl)ethan-1-one
4-chloro-2-({3-[4-(2,6-difluorophenyl)-1H-pyrazol-5-yl]piperidin-1-yl}methyl)phenol
N-[2-(2,3-dihydro-1H-indol-1-yl)ethyl]-3,5-dimethyl-4-oxo-3H,4H-thieno[2,3-d]pyrimidine-6-carboxamide
5-[(4-benzylpiperidin-1-yl)methyl]-N-(2,3-dihydroxypropyl)-1,2-oxazole-3-carboxamide
3-{4-[3-(morpholin-4-yl)pyrrolidin-1-yl]-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-2-yl}-1H-indole
N-methyl-N-[(2-phenyl-1,3-thiazol-4-yl)methyl]oxane-4-carboxamide
5-[3-(aminomethyl)pyrrolidin-1-yl]-2-[(4-ethyl-2-methyl-1,3-thiazol-5-yl)methyl]-2,3-dihydropyridazin-3-one
{1-ethyl-5-[2-(pyrrolidin-1-ylmethyl)-1,3-thiazol-5-yl]-1H-1,2,4-triazol-3-yl}(phenyl)methanol
1-[2-({[3-(2-chlorophenyl)-1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}amino)ethyl]piperidin-2-one
[1-(1-phenylcyclopropanecarbonyl)-3-(prop-2-en-1-yl)piperidin-3-yl]methanol
(2R,3S,6R)-5-methyl-3-(4-methylphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
1-(4-chlorobenzoyl)-N-[3-(dimethylamino)propyl]-N-methylpiperidin-3-amine
6,7-dimethoxy-3-[(2,3,6-trifluorophenyl)methyl]-3,4-dihydroquinazolin-4-one
4-[1-(2H-1,3-benzodioxol-5-ylmethyl)piperidin-4-yl]pyridine
1-(4-{[(2-methoxyethyl)(propan-2-yl)amino]methyl}phenoxy)-3-(4-methylpiperazin-1-yl)propan-2-ol
methyl 6-(butan-2-yl)-2-{[2-(2-fluorophenyl)ethyl]sulfamoyl}-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
N-[(8-methoxyquinolin-5-yl)methyl]-N-methyl-3-(4-methyl-1,3-thiazol-5-yl)propanamide
4,4,4-trifluoro-1-{4-[4-methyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}butan-1-one
4-benzyl-3-ethyl-1-{[5-(propan-2-yl)-1,3,4-oxadiazol-2-yl]methyl}-1,4-diazepan-5-one
1-[(4-methylphenyl)amino]-N-[1-(1-propyl-1H-1,2,4-triazol-5-yl)ethyl]cyclopentane-1-carboxamide
N-{3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]propyl}adamantane-1-carboxamide
N-[6,6-dimethyl-1-(4-methylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-2-(pyridin-3-yl)acetamide
1-{[5-(4,6-dimethoxypyrimidin-2-yl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}-3,3-dimethylurea
4-(4-methylphenoxy)-1-(3-phenylpropyl)piperidine-4-carboxylic acid
2-amino-6-(furan-2-yl)-4-(8-methoxy-3,4-dihydro-2H-1,5-benzodioxepin-7-yl)pyridine-3-carbonitrile
2-[3-phenyl-5-(1,2,3,6-tetrahydropyridin-4-ylmethyl)-1H-1,2,4-triazol-1-yl]pyridine
4-benzyl-3-[1-(3-methoxypropanoyl)piperidin-4-yl]-4,5-dihydro-1H-1,2,4-triazol-5-one
2-{1-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]-3-oxopiperazin-2-yl}-N-(2-methylpropyl)acetamide
3-(1-{2-[2,4-dimethyl-5-(1H-1,2,4-triazol-1-ylmethyl)phenyl]-1H-imidazol-1-yl}ethyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
3-[2-(3-fluorophenyl)-3-oxopiperazine-1-carbonyl]-5-methoxybenzoic acid
N-[(3S,4R)-1-(5-hydroxypyrazine-2-carbonyl)-4-(4-methylphenyl)pyrrolidin-3-yl]cyclopropanecarboxamide
5-({5-cyclopropanecarbonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}carbonyl)-4-methyl-1,3-thiazol-2-amine
N-{[4-methyl-2-(propan-2-yl)-1,3-thiazol-5-yl]methyl}-2-[1-(propan-2-yl)piperidin-4-yl]acetamide
7-[(3-hydroxybutyl)sulfamoyl]-N-(propan-2-yl)-1,2,3,4-tetrahydroisoquinoline-2-carboxamide
1-[4-(1-butyl-1H-imidazol-2-yl)piperidine-1-carbonyl]cyclopropan-1-amine
N-{imidazo[1,2-a]pyridin-3-ylmethyl}-1-[4-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)phenyl]piperidin-4-amine
1-[(2-fluorophenyl)methyl]-5-{2-[(pyridin-3-ylmethyl)amino]ethyl}pyrrolidin-2-one
methyl 5-[3-(2-oxo-2,3-dihydro-1H-1,3-benzodiazol-1-yl)propanoyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxylate
4-{4-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}pyridin-2-amine
3-[(1H-indol-3-ylmethyl)[(5-methylthiophen-2-yl)methyl]amino]propan-1-ol
N,3-dimethyl-1-propyl-N-(4,5,6,7-tetrahydro-1H-indazol-3-ylmethyl)-1H-pyrazole-4-carboxamide
1-[(6,7-dimethyl-1H-1,3-benzodiazol-2-yl)methyl]-N-(furan-2-ylmethyl)piperidine-4-carboxamide