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1-[2-(methoxymethyl)piperidin-1-yl]-3-{5-[(4-phenylphenyl)methyl]-1,3,4-oxadiazol-2-yl}propan-1-one
4-(2-hydroxy-5-methoxyphenyl)-1-[(2-methoxyphenyl)methyl]-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
(3aR,6aR)-2-(2H-1,3-benzodioxole-5-carbonyl)-5-(prop-2-en-1-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
4-{[1-(2-methoxyacetyl)piperidin-4-yl]oxy}-N-[1-(2-methyl-1,3-thiazol-4-yl)ethyl]benzamide
methyl 5-{2-[(3-fluorophenyl)methyl]morpholin-4-yl}-5-oxopentanoate
4-(1H-pyrazol-1-yl)-1-{spiro[2.3]hexane-1-carbonyl}piperidine-4-carboxylic acid
N-({1-[(2E)-3-(furan-2-yl)-2-methylprop-2-en-1-yl]pyrrolidin-3-yl}methyl)-1,3-thiazole-5-carboxamide
5-[1-(3-fluorophenyl)-3-[(1-methylpiperidin-4-yl)methyl]-1H-1,2,4-triazol-5-yl]pyrazin-2-ol
3-(1H-pyrazol-1-yl)-N-[1-(pyridin-3-yl)propan-2-yl]propanamide
1-[(3-methylthiophen-2-yl)methyl]-3-phenylpyrrolidin-3-ol
1-[(3,4-dimethoxyphenyl)methyl]-4-{2-[(4-fluorophenyl)methyl]-3H-imidazo[4,5-b]pyridin-3-yl}piperidine
8-(3-ethyl-1H-indole-2-carbonyl)-2-methyl-2,8-diazaspiro[4.5]decane-3-carboxylic acid
5-{5-[1-(3-chlorophenoxy)ethyl]-1,2,4-oxadiazol-3-yl}-6-methyl-1,2,3,4-tetrahydro-2,7-naphthyridine
1-(3-fluorophenyl)-3-(1-{1-[3-(pyridin-2-yl)propanoyl]piperidin-4-yl}-1H-pyrazol-5-yl)urea
2-chloro-3-{[(furan-2-ylmethyl)(3-methylbutan-2-yl)amino]methyl}-9-methyl-4H-pyrido[1,2-a]pyrimidin-4-one
N-{[1-(1H-imidazol-1-ylmethyl)cyclopropyl]methyl}-2-oxo-2-(1,2,3,4-tetrahydroquinolin-1-yl)acetamide
1-(2-methoxy-4-{[(2-methoxy-2-methylpropyl)amino]methyl}phenoxy)-3-(pyrrolidin-1-yl)propan-2-ol
N-(3,5-dimethoxyphenyl)-2-[4-hydroxy-4-(pyridin-2-yl)piperidin-1-yl]acetamide
N-[2-(dimethylamino)ethyl]-N-methyl-5-[4-(pyridin-3-yloxy)piperidine-1-carbonyl]pyridin-2-amine
N,2,3-trimethyl-N-[3-(1-methyl-1H-pyrazol-4-yl)propyl]quinoxaline-6-carboxamide
3-[(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)sulfamoyl]benzoic acid
(2R)-1-[3-(4-methyl-1,2,3,6-tetrahydropyridine-1-carbonyl)benzenesulfonyl]pyrrolidine-2-carboxamide
3-(3-chlorobenzoyl)-1-(5-methyl-1,3,4-oxadiazol-2-yl)piperidine
N-cyclopropyl-1-{1-[2-(4-methoxyphenyl)acetyl]piperidin-4-yl}piperidine-4-carboxamide
2-{5-[(3,4-difluorophenyl)methyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl}-1H-1,3-benzodiazole
3-{2-oxo-8-[(1R,2R)-2-phenylcyclopropanecarbonyl]-1-oxa-3,8-diazaspiro[4.5]decan-3-yl}propanoic acid
N-(2-{[(3-chlorophenyl)methyl]sulfanyl}ethyl)-5-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxamide
3-(1-butyl-1H-imidazol-2-yl)-1-phenylmethanesulfonylpiperidine
N-ethyl-N-({1-[2-(2-methylphenyl)ethyl]piperidin-4-yl}methyl)cyclopent-1-ene-1-carboxamide
3-methyl-6-(5-{2H,3H-thieno[3,4-b][1,4]dioxin-5-yl}-1,2,4-oxadiazol-3-yl)pyridazine
1-[5-(2,5-dimethylphenoxymethyl)-1,2-oxazole-3-carbonyl]-3-(methoxymethyl)piperidine
(2S,4R)-4-amino-1-[(4-methanesulfonylphenyl)methyl]-N-methylpyrrolidine-2-carboxamide
(1S,5R)-3-benzyl-6-(4-ethenylbenzoyl)-3,6-diazabicyclo[3.2.2]nonane
N-[3-(1H-indazol-1-yl)propyl]-1-[4-methyl-6-(propan-2-yl)quinazolin-2-yl]piperidine-4-carboxamide
2-methyl-6-[(2R,3R,6R)-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carbonyl]-2,3-dihydropyridazin-3-one
3-cyclohexyl-N-{[2-(pyrrolidin-1-yl)-1,3-thiazol-4-yl]methyl}-1H-pyrazole-4-carboxamide
2-methyl-4-[4-(3-phenylpiperazine-1-carbonyl)phenyl]butan-2-ol
2-{5-[2,5-dimethyl-1-(pyridin-3-ylmethyl)-1H-pyrrol-3-yl]-4-phenyl-1H-imidazol-1-yl}-N-methylacetamide
5-(3,4-dimethylphenoxymethyl)-N-methyl-N-(3-methylbutyl)-1,2-oxazole-3-carboxamide
2-(dimethyl-1H-1,2,4-triazol-1-yl)-1-[3-(3-fluoro-4-methoxybenzoyl)piperidin-1-yl]ethan-1-one
N-({1-[(4-hydroxyphenyl)methyl]piperidin-3-yl}methyl)-4-methoxybenzene-1-sulfonamide
4-{5-[(3-oxopiperazin-1-yl)methyl]-1-phenyl-1H-1,2,4-triazol-3-yl}benzamide
ethyl 4-[(3-methoxyphenyl)methyl]-1-[(6-methylpyridin-2-yl)methyl]piperidine-4-carboxylate
2-{2-[3-(1-methyl-1H-imidazol-4-yl)-1,2,4-oxadiazol-5-yl]ethyl}-1H-1,3-benzodiazole
2-butyl-5-chloro-4-{1-[2-(1H-imidazol-4-yl)ethyl]-1H-imidazol-2-yl}-1H-imidazole
3-(2H-1,3-benzodioxol-5-yl)-5-(morpholine-4-sulfonyl)benzoic acid
N-{2-[5-(3-ethoxy-4-methoxyphenyl)-4-phenyl-1H-imidazol-1-yl]ethyl}acetamide
5-(3-{8-chloro-1H,2H,3H,4H,5H-pyrido[4,3-b]indol-2-yl}-3-oxopropyl)imidazolidine-2,4-dione
2-(1-cyclopentyl-3-oxopiperazin-2-yl)-N-{[2-(trifluoromethoxy)phenyl]methyl}acetamide
N-{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-1-[(2-fluorophenyl)methyl]-1H-1,2,3-triazole-4-carboxamide