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3-[5-(4-methoxypyrimidin-2-yl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]-1-(pyrrolidin-1-yl)propan-1-one
2-ethoxy-N-methyl-N-[(1-phenylpyrrolidin-3-yl)methyl]pyridine-3-carboxamide
2-[3,5-difluoro-4-(pyrrolidin-1-ylmethyl)phenoxy]-5-(trifluoromethyl)pyridine
N-{[1-(methoxymethyl)cyclopropyl]methyl}-N'-(4-methylphenyl)propanediamide
1-[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-5-[2-({[3-(trifluoromethyl)phenyl]methyl}amino)ethyl]pyrrolidin-2-one
1-(4-carboxy-1H-imidazole-5-carbonyl)-3-ethylpiperidine-3-carboxylic acid
1-[6-(2-fluorophenyl)imidazo[2,1-b][1,3]thiazole-3-carbonyl]-4-(furan-2-carbonyl)-1,4-diazepane
N-[2-(5-methyl-1H-1,3-benzodiazol-2-yl)ethyl]-4-(trimethyl-1H-pyrazol-4-yl)pyrimidin-2-amine
3-[1-(3-cyclohexyl-1H-pyrazol-4-yl)-N-(2-phenylethyl)formamido]propanamide
2-{4-[4-ethyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}ethan-1-amine
4-[4-(ethoxycarbonyl)-4-(2-phenylethyl)piperidine-1-carbonyl]pyridin-1-ium-1-olate
3-ethyl-5-{1H,2H,3H,4H,9H-pyrido[3,4-b]indole-2-carbonyl}-1,2-oxazole
1-methyl-4-[2-oxo-2-(3-propoxypiperidin-1-yl)ethyl]-2,3,4,5-tetrahydro-1H-1,4-benzodiazepine-2,5-dione
2-{7-cyclopentyl-6-oxo-2,7-diazaspiro[4.5]decan-2-yl}-5,6-dimethylpyridine-3-carbonitrile
N-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-1-(7-methanesulfonyl-4-methylquinazolin-2-yl)pyrrolidine-2-carboxamide
(2S,4S)-4-(3-chlorobenzamido)-N-ethyl-1-(oxan-4-yl)pyrrolidine-2-carboxamide
2-(3-fluoro-4-hydroxyphenyl)-1-[4-(2-methoxyphenoxy)piperidin-1-yl]ethan-1-one
6-cyclopentyl-N,1-dimethyl-N-[(4-methyl-1H-imidazol-2-yl)methyl]-1H-pyrazolo[3,4-d]pyrimidin-4-amine
3-[methyl({5-[4-(trifluoromethyl)phenyl]-1,2,4-triazin-3-yl})amino]propane-1,2-diol
6-[4-(cyclopropylmethyl)-3-(propan-2-yl)-1,4-diazepan-1-yl]pyridine-2-carbonitrile
2-methyl-N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-4-phenylpyrimidine-5-carboxamide
N-cyclobutyl-4-{[(3S,4S)-3-(dimethylamino)-4-hydroxypyrrolidin-1-yl]sulfonyl}benzamide
6-[(diethylamino)methyl]-N-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]pyrazolo[1,5-a]pyrimidine-3-carboxamide
1-(2-methoxyphenyl)-2,2-dimethyl-4-(oxolan-3-ylmethyl)piperazine
4-(1-aminocyclopropanecarbonyl)-7-(2-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
[(3R,4R)-1-(2,4-dimethoxybenzoyl)-4-(morpholin-4-ylmethyl)pyrrolidin-3-yl]methanol
2-[(1S,5R)-6-{[4-(difluoromethoxy)phenyl]methyl}-3,6-diazabicyclo[3.2.2]nonan-3-yl]-N,N-dimethylacetamide
1-{2-[(3-fluorophenyl)methyl]morpholin-4-yl}pent-4-en-1-one
1-{2-oxo-2-[3-(pyrrolidine-1-carbonyl)piperidin-1-yl]ethyl}-1,2-dihydroquinoxalin-2-one
(2S)-N-[2-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)ethyl]-2-methoxy-2-phenylacetamide
(3R)-N-ethyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
N-{[2-(2-methoxyphenyl)-1,3-thiazol-5-yl]methyl}-5,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
4,5-dimethyl 1-[(3S,5S)-5-[(1,3-dihydro-2-benzofuran-5-yl)carbamoyl]-1-[(2E)-3-(furan-2-yl)prop-2-en-1-yl]pyrrolidin-3-yl]-1H-1,2,3-triazole-4,5-dicarboxylate
2-(4-acetylphenoxy)-1-{7-[(4-acetylpiperazin-1-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl}ethan-1-one
4-{1-[cyclopropyl(1-methyl-1H-1,2,4-triazol-5-yl)methyl]-4-phenyl-1H-imidazol-5-yl}phenol
1,3-dimethyl-5-{2H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}-1H-pyrazolo[3,4-d][1,3]thiazole
N-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-N-methyloxolane-2-carboxamide
1-[(2-methoxypyridin-3-yl)methyl]-4-[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]piperazine
2-{[2-(pyridin-4-yl)-1H-imidazol-1-yl]methyl}-3-(thiophen-3-yl)propan-1-ol
N-{1-oxo-1-[3-oxo-2-(prop-2-en-1-yl)-2,9-diazaspiro[5.5]undecan-9-yl]propan-2-yl}methanesulfonamide
4-{1-[(4-fluoro-3-methoxyphenyl)methyl]piperidin-4-yl}-5-(3-methylphenyl)-2-(pyridin-4-yl)pyrimidine
2-[(2R,3R)-3-[benzyl(methyl)amino]-2-hydroxy-2,3-dihydrospiro[indene-1,4'-piperidine]-1'-yl]acetic acid
1-ethyl-3-(2-methylpropyl)-N-{1-[2-(trifluoromethyl)phenyl]ethyl}-1H-pyrazole-5-carboxamide
4-(1-{[2-methanesulfonyl-1-(3-methoxypropyl)-1H-imidazol-5-yl]methyl}piperidin-4-yl)pyridine
3-(propan-2-yl)-4-{5-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}piperazin-2-one
1,3-dimethyl-5-{[3-(propan-2-yl)-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazol-6-yl]methyl}imidazolidine-2,4-dione
1-[5-(ethylsulfanyl)thiophene-2-carbonyl]-4-(1-methyl-1H-imidazol-2-yl)piperidine
2-cyclohexyl-1-[(1S,5R)-3-(pyrazine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
5-amino-4-chloro-N-[1-(dimethyl-1,3-thiazol-4-yl)ethyl]-N-methyl-1H-pyrazole-3-carboxamide
N-{1-[2-(methylsulfanyl)ethyl]piperidin-4-yl}quinoxaline-5-carboxamide