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N-[(5-methylpyrazin-2-yl)methyl]-4-(1H-pyrazol-5-yl)benzamide
N-[1-(1-methylpiperidin-4-yl)piperidin-3-yl]-1-phenylcyclohexane-1-carboxamide
N-(3-methylphenyl)-3-{1-[4-(thiophen-2-yl)butanoyl]piperidin-4-yl}propanamide
(2R)-N-[3-chloro-4-(dimethylcarbamoyl)phenyl]-2-methylpiperazine-1-carboxamide
N-benzyl-1-methyl-5-(pyridin-3-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
1-cyclohexyl-4-(1H-indol-7-ylmethyl)piperazin-2-one
1-[(4-benzylmorpholin-2-yl)methyl]-4-ethyl-3-(piperidin-4-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
2-chloro-N-[(3,4-dimethoxyphenyl)methyl]-5-(1H-pyrazol-1-yl)benzamide
1-ethyl-5-oxo-N-[(3-phenylphenyl)methyl]pyrrolidine-3-carboxamide
1-({5-methyl-2-[3-(trifluoromethyl)phenyl]-1,3-oxazol-4-yl}methyl)piperidine-3-carboxamide
2-phenyl-N-[(1r,4r)-4-hydroxycyclohexyl]imidazo[1,2-a]pyridine-6-carboxamide
4-(4-methylpiperazin-1-yl)-6-(3,4,5-trimethoxyphenyl)quinazoline
3-[(2R,3R,6R)-3-(4-fluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carbonyl]-6-methyl-1,2-dihydropyridin-2-one
8-(2-ethoxyethyl)-2-[(5-methylpyrazin-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
1-{1-[5-(methoxymethyl)pyrazolo[1,5-a]pyrimidin-7-yl]piperidin-4-yl}-1,4-diazepan-5-one
8-[1-(2-fluorophenyl)cyclopropanecarbonyl]-1-methyl-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
2-(2-aminopyridine-4-carbonyl)-7-methyl-2,7-diazaspiro[4.5]decan-6-one
1-[(3R,4S)-3-amino-4-(propan-2-yl)pyrrolidin-1-yl]-3-(1H-1,2,4-triazol-1-yl)propan-1-one
methyl 5-[2-(pyrimidin-2-ylsulfanyl)acetyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxylate
1-benzyl-N3-[(3-methylphenyl)methyl]-4-oxo-N5-(prop-2-en-1-yl)-1,4-dihydropyridine-3,5-dicarboxamide
N-[(3S,4R)-1-(5-acetylpyridin-2-yl)-4-propylpyrrolidin-3-yl]methanesulfonamide
3-[(1-acetylpiperidin-4-yl)oxy]-4-methoxy-N-methyl-N-(4,5,6,7-tetrahydro-1H-indazol-3-ylmethyl)benzamide
N-benzyl{[4-(1H-pyrazol-4-yl)phenyl]amino}sulfonamide
N-[(3-methylphenyl)methyl]-4-{[1-(pyridin-2-ylmethyl)piperidin-4-yl]oxy}benzamide
1-(2-chloro-4-fluorophenyl)-3-({1-[ethyl(methyl)amino]cyclopentyl}methyl)urea
1-(2-chloro-5-sulfamoylphenyl)-3-[1-(1-propyl-1H-1,2,4-triazol-5-yl)ethyl]urea
(1R,5R)-3-{3-fluoro-6-methylimidazo[1,2-a]pyridine-2-carbonyl}-6-(3-methylbut-2-en-1-yl)-3,6-diazabicyclo[3.2.2]nonane
N-[(1-methylpiperidin-4-yl)methyl]-3-(1,2-oxazolidin-2-yl)-N-(2-phenylethyl)propanamide
N-methyl-N-(4,5,6,7-tetrahydro-1H-indazol-3-ylmethyl)-2-(thiophen-2-yl)-1,3-thiazole-4-carboxamide
5-methyl-2-{2-[2-(2-methyl-1H-imidazol-1-yl)ethyl]piperidine-1-carbonyl}phenol
N-benzyl-N-(cyclobutylmethyl)-2-{1-[(2-methylphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
3-(5-{[4-(5-methylfuran-2-yl)phenyl]methyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl)propanoic acid
N-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-3-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]propanamide
N-[(3,4-difluorophenyl)methyl]-3-{1-[2-(1H-indazol-3-yl)acetyl]piperidin-3-yl}propanamide
(1R,2R)-2-[3-(5-methylfuran-2-yl)-5-[(pyridin-2-ylsulfanyl)methyl]-1H-1,2,4-triazol-1-yl]cyclohexan-1-ol
5-{2,8-diazaspiro[4.5]decane-3-carbonyl}-4H,5H,6H,7H-[1,3]thiazolo[5,4-c]pyridin-2-amine
(3aR,6aR)-2-methanesulfonyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]-N-propyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxamide
N-cyclooctyl-4-oxo-5-[4-(propan-2-yl)piperazine-1-carbonyl]-1-(pyridin-2-ylmethyl)-1,4-dihydropyridine-3-carboxamide
N-[(1-{2-[(5-methyl-1,3,4-oxadiazol-2-yl)sulfanyl]acetyl}piperidin-3-yl)methyl]-4-phenylbenzamide
(cyclobutylmethyl)(oxolan-2-ylmethyl){[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}amine
8-[2-(pyridin-3-yl)acetyl]-2-(pyridin-4-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
2-(butylsulfanyl)-N4-[(1-methyl-1H-pyrazol-4-yl)methyl]pyrimidine-4,6-diamine
[1-(5-chloropyridin-2-yl)-3-(2-methoxyethyl)piperidin-3-yl]methanol
3-{1-[1-(quinoxalin-2-yl)piperidin-4-yl]-1H-1,2,3-triazol-4-yl}propanoic acid
N-({6-cyclopentyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-4-methyl-1H-pyrrole-2-carboxamide
1-(5-{2-azaspiro[4.4]nonan-2-ylmethyl}-2-methoxyphenoxy)-3-(diethylamino)propan-2-ol
4-[(1-cyclohexyl-1H-imidazol-5-yl)methyl]-2H,3H,4H-pyrido[3,2-b][1,4]oxazin-3-one
1-[(2,3-difluorophenyl)methyl]-3-hydroxy-3-[(4-methyl-1,4-diazepan-1-yl)methyl]piperidin-2-one
N-[(3-methylphenyl)methyl]-2-{1-[(2-methylphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
methyl 3-[(propan-2-yl)[(trimethyl-1H-pyrazol-4-yl)methyl]carbamoyl]propanoate