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(1S,5R)-6-[2-methoxy-5-(1H-pyrazol-1-yl)benzenesulfonyl]-3-methyl-3,6-diazabicyclo[3.2.2]nonane
(3aS,6aS)-2-cyclopropanecarbonyl-5-[(2-methoxyphenyl)carbamoyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-{3-[4-({[(2-fluorophenyl)methyl]amino}methyl)-2-methoxyphenoxy]-2-hydroxypropyl}piperidin-4-ol
8-[(8-methoxy-3,4-dihydro-2H-1,5-benzodioxepin-7-yl)methyl]-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
5-chloro-2-({6-[(2R,6S)-2,6-dimethylmorpholine-4-carbonyl]imidazo[2,1-b][1,3]thiazol-5-yl}methyl)-1,2,3,4-tetrahydroisoquinoline
ethyl 1-[(3-acetylphenyl)methyl]-3-[(3-methoxyphenyl)methyl]piperidine-3-carboxylate
[5-({3-[2-(2,6-difluorophenyl)ethyl]piperidin-1-yl}methyl)furan-2-yl]methanol
4-{2-[3-(2-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]ethyl}morpholine
2-[3-ethyl-4-(propan-2-yl)piperazin-1-yl]-5-methoxypyrimidine
N-[(4-methoxyphenyl)methyl]-2-{3-oxo-1-[(4-phenylphenyl)methyl]piperazin-2-yl}acetamide
2-(naphthalen-2-yloxy)-N-[2-(2-oxo-1,3-oxazolidin-3-yl)ethyl]propanamide
1-(2-methoxyethyl)-3-[(3-methoxyphenyl)methyl]-8-(naphthalen-1-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
5-ethyl-2-{4-[2-(1H-pyrazol-1-yl)ethyl]piperidin-1-yl}pyrimidine
N-(1-{1-[(5-acetylthiophen-3-yl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)-4-phenylbutanamide
(2R,6R)-4-(4-chlorobenzoyl)-10-methoxy-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
methyl (2S,4R)-1-methyl-4-(4-methyl-3,4-dihydro-2H-1,4-benzoxazine-7-sulfonamido)pyrrolidine-2-carboxylate
1-[4-(2H-1,3-benzodioxol-5-yl)pyrimidin-2-yl]-5-cyclopropyl-N-[(4-fluorophenyl)methyl]-1H-pyrazole-4-carboxamide
6-cyclopentyl-2-(4-{[methyl(pyridin-2-ylmethyl)amino]methyl}phenyl)-3,4-dihydropyrimidin-4-one
(4aS,8aR)-2-{[1-butyl-2-(ethanesulfonyl)-1H-imidazol-5-yl]methyl}-decahydroisoquinoline
N-[2-(2-oxopiperidin-1-yl)ethyl]-2-(3-phenylpropyl)-1,3-benzoxazole-5-carboxamide
1-[(3R,4R)-4-cyclobutyl-4-hydroxy-3-methylpiperidin-1-yl]-2-(pyrrolidin-1-yl)ethan-1-one
N-({1-[(2-methoxyphenyl)methyl]piperidin-4-yl}methyl)-N-(2-methylpropyl)pyridine-2-carboxamide
3-{2-[2-(6-methyl-1H-1,3-benzodiazol-2-yl)pyrrolidin-1-yl]-2-oxoethyl}-1,3-oxazolidin-2-one
1-(cyclohexylmethyl)-N-[2-(4,6-dimethylpyrimidin-2-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
2-amino-6-{2-[(4S)-4-hydroxy-3,3,4-trimethylpiperidin-1-yl]-2-oxoethyl}-3,4-dihydropyrimidin-4-one
5-[(5-methyl-2-phenyl-1,3-oxazol-4-yl)methyl]-3-(oxolan-3-yl)-1,2,4-oxadiazole
N-methyl-3-(2-oxo-1,2-dihydropyridin-1-yl)-N-[(2-phenyl-1,3-thiazol-4-yl)methyl]propanamide
N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-4-methyl-3-(2-oxoimidazolidin-1-yl)benzamide
1-methanesulfonyl-4-{5-[1-(piperidin-1-yl)ethyl]furan-2-carbonyl}piperazine
(2S)-2-amino-N-(2-methylpropyl)-N-(3-phenylprop-2-yn-1-yl)-3-(1,3-thiazol-4-yl)propanamide
4-methyl-5-oxo-N-[3-(pyridin-3-yloxy)propyl]oxolane-3-carboxamide
5-({ethyl[2-(pyridin-2-yl)ethyl]amino}methyl)-N-phenyl-1,3-thiazol-2-amine
N-(3-hydroxy-2,2-dimethylpropyl)-2-[methyl(2-phenylethyl)amino]-2,3-dihydro-1H-indene-2-carboxamide
9-[2-(benzenesulfonyl)ethyl]-2-ethyl-2,9-diazaspiro[5.5]undecan-3-one
(2R,3R)-3-(dimethylamino)-1'-[(4,5-dimethylfuran-2-yl)methyl]-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
1-(1-{5H,6H-benzo[h]quinazolin-2-yl}-5-(methoxymethyl)-1H-pyrazole-4-carbonyl)-4-ethylpiperazine
N-(1-{1-[3-(2-chlorophenyl)propanoyl]piperidin-4-yl}-2-(2,4-difluorophenyl)ethyl)-N-methylpropanamide
N-[(3S,4R)-1-(8-methoxyquinolin-2-yl)-4-(propan-2-yl)pyrrolidin-3-yl]methanesulfonamide
5,6-dimethyl-2-oxo-N-[2-(pyrrolidine-1-sulfonyl)ethyl]-1,2-dihydropyridine-3-carboxamide
5-{1-[(2-fluorophenyl)methyl]-1H-pyrazol-3-yl}-4-methyl-N-[(3,4,5-trimethoxyphenyl)methyl]-1,3-thiazol-2-amine
4-[(4-{4H,5H,6H,7H-thieno[3,2-c]pyridine-5-carbonyl}furan-2-yl)methyl]morpholine
4-{4-[2-(1-ethyl-1H-imidazol-2-yl)-1H-imidazol-1-yl]piperidine-1-carbonyl}morpholine
(2S)-2-amino-N-{[2-(2-fluorophenoxy)pyridin-3-yl]methyl}-3-(4-hydroxyphenyl)propanamide
4-[3-(1-methoxyethyl)phenyl]-6-(pyrrolidin-1-yl)pyrimidin-2-amine
N-[2-(3,6-dioxo-1,2,3,6-tetrahydropyridazin-1-yl)ethyl]-2-(7-fluoro-2-methyl-1H-indol-3-yl)acetamide
2-methyl-N-{[5-(2-methylpropyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}-6-oxo-1,6-dihydropyrimidine-5-carboxamide
2-(2-fluorophenoxy)-N-(oxan-4-yl)pyridin-3-amine
2-ethyl-5-{3-[(2-methylphenyl)methoxy]azetidine-1-carbonyl}pyrimidine
(2S,4S)-N-ethyl-1-[(3-hydroxyphenyl)methyl]-4-[3-(methylsulfanyl)propanamido]pyrrolidine-2-carboxamide
2-{2-[1-(5-chloro-2-hydroxybenzoyl)piperidin-4-yl]-1H-imidazol-1-yl}acetamide