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4-ethyl-3-({1-[(2E)-3-(4-fluorophenyl)prop-2-en-1-yl]piperidin-4-yl}methyl)-1-methyl-4,5-dihydro-1H-1,2,4-triazol-5-one
(2S)-4-(benzyloxy)-2-{imidazo[2,1-b][1,3]thiazol-6-ylformamido}butanoic acid
1-methyl-3-[3-methyl-1-(2-methylphenyl)-1H-pyrazol-5-yl]-1-[3-(oxolan-2-yl)propyl]urea
1-(2-{5-cyclopropanecarbonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}-2-oxoethyl)-1,4-dihydropyridin-4-one
2-(2-methoxyethyl)-N-{4-[(2-methylprop-2-en-1-yl)oxy]phenyl}piperidine-1-carboxamide
1-ethyl-8-{[4-(3-hydroxy-3-methylbut-1-yn-1-yl)phenyl]methyl}-3-[3-(pyridin-3-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-[(1S,5R)-3-[5-(methoxymethyl)thiophene-2-carbonyl]-7-oxo-3,6-diazabicyclo[3.2.2]nonan-6-yl]-N,N-dimethylacetamide
1-{2-[3-(2,3-dihydro-1-benzofuran-7-yl)phenoxy]ethyl}-1H-imidazole
4-(dimethylamino)-N-{[2-(2-fluorophenyl)-3-methyl-1H-indol-5-yl]methyl}butanamide
1-(3-methoxypropyl)-3-{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}-1,3,8-triazaspiro[4.5]decane-2,4-dione
(1-benzothiophen-2-ylmethyl)({4-[2-(4-{imidazo[2,1-b][1,3]thiazole-6-carbonyl}piperazin-1-yl)ethoxy]phenyl}methyl)methylamine
6-(3-benzoylpiperidine-1-carbonyl)-2,5-dimethyl-3H,4H-thieno[2,3-d]pyrimidin-4-one
(2R,6S)-2,6-dimethyl-4-(2-{1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl}-2,3-dihydro-1H-inden-2-yl)morpholine
3-amino-N-{[2-(2,4-difluorophenoxy)pyridin-3-yl]methyl}-2-hydroxypropanamide
2-[(1S,5R)-3-[(dimethyl-1,2-oxazol-4-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]-1-(morpholin-4-yl)ethan-1-one
1-methyl-N-[2-(5-methylfuran-2-yl)-2-(morpholin-4-yl)ethyl]-3-propyl-1H-pyrazole-5-carboxamide
N-[1-(2,3-dihydro-1H-inden-2-yl)-5-oxopyrrolidin-3-yl]-2-hydroxy-4-methylbenzamide
(3R,4R)-1-cyclopentanecarbonyl-4-[4-(2-fluorophenyl)piperazin-1-yl]piperidin-3-ol
(4-{[1-(1-ethyl-5-methyl-1H-pyrazole-3-carbonyl)pyrrolidin-3-yl]methyl}phenyl)methanol
4-fluoro-N-({4-methyl-5-[(pyridin-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}methyl)benzamide
4-(1H-pyrazol-3-yl)-N-[2-(pyridin-2-ylsulfanyl)ethyl]benzamide
1-(4-methylphenyl)-4-(2,2,3,3-tetramethylcyclopropanecarbonyl)piperazin-2-one
1-[(1-benzylpiperidin-3-yl)methyl]pyrrolidin-2-one
1-methyl-N-{2-[4-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)morpholin-2-yl]ethyl}piperidine-4-carboxamide
1-propyl-5-[4-(pyridin-4-yl)piperidin-1-yl]-4,5,6,7-tetrahydro-1H-indazole-3-carboxylic acid
N-[2-(dimethylamino)-2-(2-methylphenyl)ethyl]-2-(2-oxopiperidin-1-yl)acetamide
methyl 1-{2-hydroxy-3-[4-({[2-(piperidin-1-yl)ethyl]amino}methyl)phenoxy]propyl}piperidine-4-carboxylate
3-(3-hydroxyquinoxalin-2-yl)-N-[1-(1H-imidazol-1-yl)butan-2-yl]propanamide
1-{[5-methyl-2-(thiophen-2-yl)-1,3-oxazol-4-yl]methyl}-3-(3-methylthiophene-2-carbonyl)piperidine
5-{[benzyl(methyl)amino]methyl}-N-{pyrazolo[1,5-a]pyrimidin-3-ylmethyl}-1,2-oxazole-3-carboxamide
N-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]-2-[(quinolin-8-yloxy)methyl]-1,3-oxazole-4-carboxamide
N-[3-(1H-1,2,3-benzotriazol-1-yl)propyl]-2-[2-(2-fluorophenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]acetamide
1-{1-[(5-ethylpyridin-2-yl)methyl]piperidin-4-yl}-N-(pyridin-3-ylmethyl)piperidine-3-carboxamide
N-[(6-chloro-1H-1,3-benzodiazol-2-yl)methyl]-1-methyl-1H-indole-2-carboxamide
N-(2-methoxyethyl)-1-[1-(4-methylpyridine-3-carbonyl)piperidin-4-yl]piperidine-3-carboxamide
5-({2,4-dimethyl-5H,6H-furo[2,3-d]pyrimidin-6-yl}methyl)-2-phenyl-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
5,6-dimethyl-N-[2-(1-methylpyrrolidin-2-yl)ethyl]thieno[2,3-d]pyrimidin-4-amine
N-{2-methyl-1-[7-({4-[methyl(phenyl)amino]phenyl}methyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]propyl}furan-3-carboxamide
4-{4-[(4-benzyl-1H-1,2,3-triazol-1-yl)methyl]piperidin-1-yl}pyrimidin-2-amine
2-{1-[3-(2-chlorophenyl)propyl]piperidin-2-yl}ethan-1-ol
N-(2-{3-[(6,7-dimethoxy-1,2,3,4-tetrahydroisoquinolin-2-yl)methyl]phenoxy}propyl)cyclohexanecarboxamide
N-[3-(4-chloro-3-methylphenoxy)-2-hydroxypropyl]-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
1-{[3-(2H-1,3-benzodioxol-5-yl)-1H-pyrazol-4-yl]methyl}-4-phenyl-1,4-diazepane
2-[4-(2,4-dimethoxyphenyl)phenyl]-2-methylpropanamide
4-{3-[2-(1-methyl-1H-1,3-benzodiazol-2-yl)-1H-imidazol-1-yl]propyl}piperazin-2-one
3-[3-(3-methoxyphenoxymethyl)piperidine-1-carbonyl]-2-methyl-4,5,6,7-tetrahydro-2H-indazole
2-(3,6-dioxo-1,2,3,6-tetrahydropyridazin-1-yl)-N-[2-(2-phenoxyethoxy)phenyl]acetamide
(1R,5R)-3-[3-(2-methylpropyl)-1,2-oxazole-5-carbonyl]-3,9-diazabicyclo[3.3.2]decan-10-one
(3R,4R)-4-(hydroxymethyl)-1-{6-methyl-2H-[1,3]dioxolo[4,5-g]quinolin-8-yl}piperidin-3-ol
1-[2-fluoro-5-(4H-1,2,4-triazol-4-yl)phenyl]-3-{[1-(2-methoxyethyl)-5-oxopyrrolidin-3-yl]methyl}urea