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2-(3-methylpiperidin-1-yl)-5-[4-(pyridin-3-yloxy)piperidine-1-carbonyl]pyridine
5-{[(3S,4R)-3,4-dihydroxy-4-methylpiperidin-1-yl]methyl}-4H,7H-[1,2,4]triazolo[1,5-a]pyrimidin-7-one
4-[2-(1-methyl-1H-1,3-benzodiazol-2-yl)pyrrolidine-1-carbonyl]-1,2-dihydroquinolin-2-one
7-(1-benzothiophen-3-yl)-4-(3-methylthiophene-2-carbonyl)-9-(oxolan-3-yloxy)-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-[(3R,5S)-5-(ethylcarbamoyl)-1-(furan-2-carbonyl)pyrrolidin-3-yl]-1H-pyrrole-3-carboxamide
3-[1-(2,1,3-benzoxadiazol-4-ylmethyl)piperidin-4-yl]-4-ethyl-4,5-dihydro-1H-1,2,4-triazol-5-one
methyl 6-benzoyl-2-[(3-methylphenyl)sulfamoyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
2-{5-[(3-propyl-1,2,4-oxadiazol-5-yl)methyl]-3H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl}pyridine
2-methyl-4-[3-(naphthalen-1-yl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-5-carbonyl]-1,3-thiazole
ethyl 4-{5H,6H,7H,8H-imidazo[1,5-a]pyrazine-7-carbonyl}-3,5-dimethyl-1H-pyrrole-2-carboxylate
N-{1-[(2-fluorophenyl)methyl]piperidin-3-yl}-5-methyl-1,3-oxazole-4-carboxamide
N3-[(2-ethyl-3-methyl-1H-indol-5-yl)methyl]piperidine-1,3-dicarboxamide
N-ethyl-N-[(4-methoxyphenyl)methyl]-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
2-(5-methyl-1H-pyrazol-1-yl)-1-{3-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}ethan-1-one
methyl 3-{[1-(4-methoxyphenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-yl]carbamoyl}propanoate
N-[(2R,3R)-2-methoxy-1'-(1H-pyrazol-3-ylmethyl)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-(methylsulfanyl)acetamide
{4-[(1-{[6-(dimethylamino)pyridin-3-yl]methyl}pyrrolidin-3-yl)methyl]phenyl}methanol
1-(4-{5-[(dimethylamino)methyl]-4-ethyl-4H-1,2,4-triazol-3-yl}piperidin-1-yl)-3-(pyridin-2-yl)propan-1-one
1-(5-methoxyfuran-2-carbonyl)-4-(2-methylpyridin-4-yl)-1,4-diazepane
1-(2-methylpropyl)-N-(pyridin-3-ylmethyl)-5-(pyridine-3-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
5-(2-tert-butylpyrimidin-4-yl)-2-ethoxybenzoic acid
1-(4-methoxyphenyl)-3-methyl-4-(4-oxo-4-phenylbutyl)piperazin-2-one
N-(1-methylpiperidin-4-yl)-5-[4-(morpholin-4-yl)piperidine-1-carbonyl]pyridin-2-amine
3-(2-chlorophenyl)-4-{5H,6H,7H,8H,9H-imidazo[1,5-a][1,4]diazepine-8-carbonyl}-5-methyl-1,2-oxazole
5-[3-(1H-pyrazol-3-yl)phenyl]pyrimidin-2-amine
1-[4-hydroxy-4-(hydroxymethyl)piperidin-1-yl]-2-(2-methyl-1H-1,3-benzodiazol-5-yl)ethan-1-one
1-[1'-(1,3-dimethyl-1H-pyrazole-4-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]propan-1-one
4-({[1-(propan-2-yl)-1H-pyrazol-4-yl]formamido}methyl)benzoic acid
[1-(5-methyl-1-phenyl-1H-pyrazol-4-yl)ethyl]({[3-(methylsulfanyl)phenyl]methyl})amine
2-{2-[3-(trifluoromethyl)phenyl]acetyl}-2,7-diazaspiro[4.5]decan-6-one
2-[(2,6-dichlorophenyl)methyl]-5-(4-methyl-1,4-diazepane-1-carbonyl)pyrimidin-4-ol
N-methyl-2-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]-N-[(2-phenyl-1,3-thiazol-4-yl)methyl]acetamide
3-(2H-1,3-benzodioxol-5-yl)-5-cyclobutyl-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine
5-{1-[2-(cyclohex-1-en-1-yl)acetyl]pyrrolidin-2-yl}-N-(pyridin-4-yl)thiophene-2-carboxamide
2-(4-{5-methyl-1-[5-methyl-4-(thiophen-2-yl)pyrimidin-2-yl]-1H-pyrazole-4-carbonyl}piperazin-1-yl)phenol
3-(2H-1,3-benzodioxol-5-yl)-5-[(5-methylfuran-2-yl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
N-[(5-fluoro-2-methylphenyl)methyl]-2-{1-[(4-methoxy-2,3-dimethylphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
N'-(2,3-dimethylphenyl)-N-[(2-fluorophenyl)methyl]-N-(1-methoxypropan-2-yl)propanediamide
(3S,4R)-4-(2H-1,3-benzodioxol-5-yl)-1-[2-(2-methoxyethoxy)acetyl]pyrrolidine-3-carboxylic acid
7-{2-amino-3-ethyl-3H-imidazo[4,5-b]pyridine-6-carbonyl}-2-methyl-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-one
2-methyl-7-[3-(methylsulfanyl)propyl]-N-(oxolan-3-ylmethyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
4-methyl-6-[3-(3-methylphenyl)piperidin-1-yl]pyrimidin-2-amine
methyl 2-(piperidine-1-sulfonyl)-6-(4,4,4-trifluorobutanoyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
2-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl]pyridine-3-carbonitrile
N-methyl-N-(2-methylpropyl)-5-[(quinolin-8-yloxy)methyl]-1,2-oxazole-3-carboxamide
1-methyl-5-({5-propanoyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}carbonyl)-1,2-dihydropyridin-2-one
methyl 3-{4-[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl]butanamido}azepane-1-carboxylate
1-[3-({3-[2-(pyridin-2-yl)pyrrolidine-1-carbonyl]-1H-pyrazol-5-yl}methoxy)phenyl]ethan-1-one
4-[(4-methoxy-2,5-dimethylphenyl)methyl]-7-(pyridin-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
2-methoxy-4-{4-[1-(morpholin-4-yl)ethyl]phenyl}pyridine-3-carbonitrile