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7-{[3-(furan-2-yl)phenyl]methyl}-3-phenyl-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine
7-({[3-(1H-imidazol-1-yl)propyl](pyridin-3-ylmethyl)amino}methyl)-4-methyl-2H-chromen-2-one
{2-[4-(4-ethoxyphenyl)-1H-imidazol-2-yl]-2-methylpropyl}dimethylamine
ethyl 1-[4-(1H-1,2,3,4-tetrazol-1-ylmethyl)benzoyl]piperidine-2-carboxylate
3-(4-methoxy-3,5-dimethylbenzoyl)-1-[3-(1H-pyrazol-1-yl)benzoyl]piperidine
N-(cyclopropylmethyl)-1-{2-[(3-fluorophenyl)methyl]-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl}-N-propylpiperidine-4-carboxamide
(4aS,7aR)-N-(2-methylphenyl)-6,6-dioxo-4-pentyl-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide
2,4-difluoro-3-methoxy-N-methyl-N-[(5-propyl-1H-pyrazol-3-yl)methyl]benzamide
3-(2-phenylethyl)-1-[4-(1H-1,2,3,4-tetrazol-1-ylmethyl)benzoyl]piperidine
N-{2-[cyclopentyl(methyl)amino]ethyl}-N,5-dimethyl-1-propyl-1H-pyrazole-4-carboxamide
N-[2-(4-methyl-1H-imidazol-2-yl)ethyl]-3-propyl-1H-pyrazole-5-carboxamide
4-[2,2-dimethyl-1-(thiophen-2-yl)cyclopropaneamido]-N-ethylpiperidine-1-carboxamide
N-(1-{2-[cyclohexyl(methyl)amino]-4-methylpyrimidin-5-yl}ethyl)-3-ethyl-1H-pyrazole-5-carboxamide
1-(3-methoxyphenyl)-4-[2-(propan-2-yl)-1,3-thiazole-4-carbonyl]piperazin-2-one
N-[(5-cyclopropyl-1,2,4-oxadiazol-3-yl)methyl]-N-ethyl-3,5,7-trimethyl-1H-indole-2-carboxamide
N-methyl-N-(4,5,6,7-tetrahydro-1,2-benzoxazol-3-ylmethyl)imidazo[2,1-b][1,3]thiazole-6-carboxamide
1-(thiophen-3-ylmethyl)-4-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepin-3-yl}piperidine
N-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-N-methyl-1-{6-methylthieno[2,3-d]pyrimidin-4-yl}piperidin-4-amine
3-{1-[1-(furan-2-ylmethyl)piperidine-4-carbonyl]piperidin-3-yl}benzoic acid
1-[2-(6-methoxynaphthalen-2-yl)morpholine-4-carbonyl]cyclobutan-1-amine
N-[(dimethyl-1,3-thiazol-2-yl)methyl]-5-(2,5-dimethylphenoxymethyl)-1,2-oxazole-3-carboxamide
2-(5-{[methyl(propan-2-yl)amino]methyl}-1H-1,2,3,4-tetrazol-1-yl)-N-{[1-(2-phenylethyl)piperidin-4-yl]methyl}acetamide
3-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-N-[(5-methyl-1H-1,2,4-triazol-3-yl)methyl]benzamide
8-(4-aminopyrimidin-2-yl)-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
4-(5-{1-[3-(1H-pyrazol-1-yl)propyl]pyrrolidin-2-yl}thiophene-2-carbonyl)morpholine
2-(2-{[(1S,2S)-2-hydroxycyclohexyl]amino}-4-(morpholin-4-yl)pyrimidin-5-yl)-2-methylpropanoic acid
N-[(1-{[(pyrazin-2-yl)carbamoyl]methyl}-1,2,5,6-tetrahydropyridin-3-yl)methyl]pyrrolidine-1-carboxamide
4-{[1-(dimethylsulfamoyl)piperidin-4-yl]oxy}-N-[1-(4-fluorophenyl)ethyl]benzamide
5-methyl-N-[1-(2-phenylethyl)piperidin-3-yl]-1,3-oxazole-4-carboxamide
1-[5-(3-cyclopropyl-1,2,4-oxadiazol-5-yl)pyridin-2-yl]-4-(pyridin-2-ylmethyl)-1,4-diazepane
3-{[(3-fluoro-4-methylphenyl)carbamoyl]methyl}-N-(thiophen-2-ylmethyl)morpholine-4-carboxamide
2-{1-[3-(1H-imidazol-1-yl)propyl]-4-phenyl-1H-imidazol-5-yl}benzonitrile
methyl 2-({[3-(2,5-dimethylthiophen-3-yl)-1-(2-fluorophenyl)-1H-pyrazol-4-yl]methyl}(methyl)amino)acetate
(3S,4R)-4-(hydroxymethyl)-1-{[5-(1H-pyrazol-3-yl)furan-2-yl]methyl}piperidin-3-ol
1-(1-{1-[(2-fluorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}-4-phenylpiperidin-4-yl)ethan-1-one
N-(2-methylbutan-2-yl)-2-[6-oxo-4-(piperazin-1-yl)-1,6-dihydropyridazin-1-yl]acetamide
cyclohexyl(4-{[1-(pyrimidin-2-yl)-1H-pyrrol-2-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl)methanol
1-(3,5-dimethylphenyl)-4-{2-[3-oxo-1-(propan-2-yl)piperazin-2-yl]acetyl}piperazin-2-one
6-(10-methoxy-3,4,5,6-tetrahydro-2H-1,5-benzoxazocine-5-carbonyl)piperazin-2-one
6-[(dimethyl-1,2-oxazol-4-yl)methoxy]-4-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-1-(2-methylpropyl)-1,4-diazepan-2-one
N-[(2-ethyl-3,5-dimethyl-1H-indol-7-yl)methyl]-2-(4-oxo-1,4-dihydroquinolin-1-yl)acetamide
1-[4-(4-{[2-(pyridin-3-yloxy)ethyl]amino}piperidin-1-yl)phenyl]pyrrolidin-2-one
dimethyl[(5-{1-phenyl-1H,4H-pyrazolo[3,4-d]imidazol-5-yl}thiophen-3-yl)methyl]amine
N-(2-hydroxyethyl)-3-[5-(pyridin-3-ylmethyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]propanamide
N-[1-(7-{[4-(diethylamino)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)ethyl]-2,5-difluorobenzamide
[(3R,4R)-4-[(4-methyl-1,4-diazepan-1-yl)methyl]-1-{2-methylthieno[3,2-d]pyrimidin-4-yl}pyrrolidin-3-yl]methanol
(1R,5R)-6-(2,4-dimethylpyrimidine-5-carbonyl)-N,N-dimethyl-3,6-diazabicyclo[3.2.2]nonane-3-sulfonamide
1-{1-[1-(4,7-dimethylquinazolin-2-yl)piperidine-4-carbonyl]piperidin-3-yl}propan-1-one
5-{1-[2-(5-cyclopropyl-1,2,4-oxadiazol-3-yl)ethyl]-1H-imidazol-2-yl}-2-hydroxybenzoic acid
3-methyl-2-oxo-1-(2-phenylethyl)-2,3-dihydro-1H-1,3-benzodiazole-5-carboxylic acid