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N-methyl-2-(methylsulfanyl)-N-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]-1,3-thiazole-4-carboxamide
(3R,4S)-N,N-dimethyl-4-propyl-1-(pyridin-4-yl)pyrrolidin-3-amine
N-[1-(2,5-dimethylphenyl)ethyl]-6-methyl-2-oxo-1,2-dihydropyridine-3-carboxamide
(1R,3S)-3-methoxy-7-[2-(methylsulfanyl)-1,3-thiazole-4-carbonyl]-7-azaspiro[3.5]nonan-1-ol
N-benzyl-5-[4-(2-hydroxyphenyl)piperazin-1-yl]-N,1-dimethyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
3-(but-2-yn-1-yl)-5-(2-phenylethyl)-5-{1-[(2E)-3-phenylprop-2-en-1-yl]piperidin-4-yl}imidazolidine-2,4-dione
2-(2-chloro-4-fluorophenyl)-1-{2-[2-(1H-pyrazol-1-yl)ethyl]piperidin-1-yl}ethan-1-one
2-({3-[5-(benzylsulfanyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidin-1-yl}methyl)-6-ethoxyphenol
2-tert-butyl-4-hydroxy-N-[2-(pyridin-2-ylsulfanyl)ethyl]pyrimidine-5-carboxamide
3-[({1-[2-(2-fluorophenyl)ethyl]piperidin-3-yl}methyl)(methyl)amino]-2,2-dimethylpropan-1-ol
N-methyl-3-(2-oxo-2,3-dihydro-1H-1,3-benzodiazol-1-yl)-N-{[3-(1H-1,2,3,4-tetrazol-5-yl)phenyl]methyl}propanamide
(1S,5R)-3-methyl-6-[2-(4-methylphenoxymethyl)furan-3-carbonyl]-3,6-diazabicyclo[3.2.2]nonane
1-cyclohexyl-N-{[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-N-methyl-1H-1,2,3-triazole-4-carboxamide
N-methyl-N-[1-(4-methyl-1,3-thiazol-2-yl)ethyl]-2-(1H-1,2,4-triazol-3-yl)benzamide
4-{3-[2-(hydroxymethyl)-4-methylpiperazine-1-carbonyl]phenyl}-2-methylbutan-2-ol
4-chloro-2-{[4-(2-methyl-6-propylpyrimidin-4-yl)piperazin-1-yl]methyl}phenol
N-[(5-methylthiophen-2-yl)methyl]-2-(3-oxo-1-{[3-(trifluoromethyl)phenyl]methyl}piperazin-2-yl)acetamide
2-methoxy-4-({methyl[(1-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidin-3-yl)methyl]amino}methyl)phenol
N-{2-[(4-chlorophenyl)methoxy]ethyl}-3-(piperidin-3-yl)benzamide
5-(1-benzofuran-2-sulfonyl)-3-propyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
N-[(3,4-difluorophenyl)methyl]-3-[1-(3-methyl-5,6-dihydro-1,4-dioxine-2-carbonyl)piperidin-3-yl]propanamide
1-(5-chloro-2-methylphenyl)-4-{1-[(2-fluorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}piperazine
3-(2,3,6-trimethylquinoline-4-amido)pyrrolidine-3-carboxylic acid
N-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}-2-(1,2,3,4-tetrahydroisoquinolin-2-ylmethyl)-1,3-oxazole-4-carboxamide
2-methyl-5-[1-(1-phenylethyl)-1H,4H-pyrazolo[3,4-d]imidazol-5-yl]-1,3-thiazole
2-[4-(3-phenylpropyl)-1-(thiophen-2-ylmethyl)piperazin-2-yl]ethan-1-ol
5-fluoro-1-methyl-2-{[3-(4-methylpiperazin-1-yl)pyrrolidin-1-yl]methyl}-1H-indole
N-{imidazo[1,2-a]pyridin-2-ylmethyl}-3-(pyrrolidine-1-carbonyl)benzene-1-sulfonamide
2-methyl-N-(oxolan-2-ylmethyl)-N-(pyridin-2-ylmethyl)imidazo[1,2-a]pyridine-6-carboxamide
1-{[5-(1-benzofuran-5-ylmethyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}-3,3-dimethylurea
N-{2-methyl-1-[7-({4-[methyl(phenyl)amino]phenyl}methyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]propyl}propanamide
(3-{2-[1-(3-chloro-4-fluorobenzoyl)piperidin-3-yl]-1H-imidazol-1-yl}propyl)dimethylamine
N-{2-[(4-chlorophenyl)sulfanyl]ethyl}-3-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanamide
2-{4-[(3-{[1-(2,5-dimethoxybenzenesulfonyl)piperidin-4-yl]oxy}phenyl)methyl]piperazin-1-yl}pyrimidine
5-[1-(oxan-4-ylmethyl)-1H-imidazol-2-yl]-N-propylpyrimidin-2-amine
N-(1H-indol-6-ylmethyl)-3-(3-methoxyphenyl)-1H-pyrazole-4-carboxamide
4-{[3-(2-chlorophenyl)-1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-1,2-dimethylpiperazine
N-[(1R,2R)-2-hydroxycyclohexyl]-1-methyl-3-(2-methylpropyl)-N-propyl-1H-pyrazole-5-carboxamide
N-[2-(N-methylmethanesulfonamido)ethyl]-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
N-{2-[(3-methylpyridin-4-yl)amino]ethyl}-1-benzothiophene-2-carboxamide
N-[(7S,8aS)-2-methyl-octahydropyrrolo[1,2-a]piperazin-7-yl]-2-(5-chloro-1H-1,3-benzodiazol-2-yl)acetamide
N-{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]methyl}-N-[3-(dimethylamino)propyl]-3-ethynylbenzamide
1-benzyl-4-(cyclopropylmethyl)-3-(propan-2-yl)-1,4-diazepan-5-one
6-fluoro-3-[2-methoxy-2-(thiophen-2-yl)ethyl]-3,4-dihydroquinazolin-4-one
N3-butyl-N5-[2-(3-chlorophenyl)ethyl]-1-(2-methoxyethyl)-N3-methyl-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
5-(2,3-dimethoxybenzoyl)-1-(2-methylpropyl)-N-(pyridin-3-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
8-[3-(methylsulfanyl)propanoyl]-3-{2-[4-(propan-2-yl)piperazin-1-yl]ethyl}-1-oxa-3,8-diazaspiro[4.5]decan-2-one
4-[(4aS,8aR)-decahydroisoquinolin-2-ylmethyl]-N-(2-methyl-2H-1,2,3-triazol-4-yl)benzamide
5-(3-hydroxy-3-methylbut-1-yn-1-yl)-N-methyl-N-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)furan-2-carboxamide
1-(pyrimidin-2-yl)-4-(quinolin-6-yloxy)piperidine-4-carboxylic acid