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2-phenyl-5-{3-phenyl-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-5-carbonyl}-1H-pyrrole
9-(cyclopropylmethyl)-1-methyl-4-(pyridine-3-carbonyl)-1,4,9-triazaspiro[5.6]dodecan-10-one
{[4-ethyl-5-(1-{5-[(methylsulfanyl)methyl]furan-2-carbonyl}piperidin-4-yl)-4H-1,2,4-triazol-3-yl]methyl}dimethylamine
5-{1-[2-(1H-imidazol-4-yl)ethyl]-1H-imidazol-2-yl}-N-(propan-2-yl)pyrimidin-2-amine
4-methyl-6-{3-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyrimidin-2-amine
2-{2-ethyl-[1,3]oxazolo[5,4-d]pyrimidin-7-yl}-7-(2-hydroxyethyl)-2,7-diazaspiro[4.5]decan-6-one
7-(oxan-4-yl)-2-[2-(2H-1,2,3,4-tetrazol-2-yl)acetyl]-2,7-diazaspiro[4.5]decan-6-one
1-{1-[2-(cyclohex-1-en-1-yl)acetyl]piperidin-4-yl}-N-cyclopropylpiperidine-4-carboxamide
N-{[4-(cyclobutylmethoxy)phenyl]methyl}-N-cyclopropyl-4-methylbenzamide
({2,5-dimethyl-3-[(4-methylpiperazin-1-yl)methyl]phenyl}methyl)[(3-ethyl-1,2-oxazol-5-yl)methyl]methylamine
1-{2-[(1R,5R)-3-methanesulfonyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-oxoethyl}-5-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
N-(4-chloro-3-methoxyphenyl)-2-[2-(3-methyl-1,2-oxazol-5-yl)pyrrolidin-1-yl]acetamide
(1S,4S)-2-{2-[(1-methanesulfonylpiperidin-4-yl)oxy]benzoyl}-2-azabicyclo[2.2.1]heptane
10-methoxy-5-[1-methyl-3-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-yl]-3,4,5,6-tetrahydro-2H-1,5-benzoxazocine
1,5-dimethyl-4-{[methyl(pyrazin-2-ylmethyl)amino]methyl}-2-phenyl-2,3-dihydro-1H-pyrazol-3-one
methyl 5-{[(4-ethoxyphenyl)methyl]amino}-1-ethyl-3-(furan-3-amido)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
6-[6-(1H-pyrazol-1-yl)pyrimidin-4-yl]quinoline
2-{4-[(2R,6S)-2,6-dimethylmorpholine-4-carbonyl]-1H-1,2,3-triazol-1-yl}-N,N-diethylacetamide
(2S,4S)-4-amino-1-(2-{[(4-fluorophenyl)methyl](methyl)amino}acetyl)-N-methylpyrrolidine-2-carboxamide
ethyl 5-(1H-indole-6-carbonyl)-1-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
3-[4-(pyrrolidine-1-carbonyl)-1H-1,2,3-triazol-1-yl]-1-(thiophen-2-ylmethyl)piperidine
(4aS,8aR)-1-[2-(cyclohex-1-en-1-yl)ethyl]-6-[3-(1H-1,2,4-triazol-1-yl)propanoyl]-decahydro-1,6-naphthyridin-2-one
1-[(3-chloro-5-fluorophenyl)methyl]-3-(2-methoxyethyl)piperidine-3-carboxylic acid
5-chloro-N-(cyclopropylmethyl)-N-(2-methoxyethyl)naphthalene-1-carboxamide
2-(4-hydroxybenzoyl)-N-methyl-N-(propan-2-yl)-1,2,3,4-tetrahydroisoquinoline-7-sulfonamide
1-[2-(4-chlorophenyl)morpholin-4-yl]-2-(piperazin-1-yl)ethan-1-one
ethyl 1-[3-(methylsulfanyl)propyl]-4-(oxan-2-ylmethyl)piperidine-4-carboxylate
phenyl (7R,9aR)-7-(2-methylpropyl)-6,9-dioxo-octahydro-1H-pyrazino[1,2-a]piperazine-2-carboxylate
(4aS,8aR)-6-(3-methylpyrazin-2-yl)-1-[2-(pyridin-2-yl)ethyl]-decahydro-1,6-naphthyridin-2-one
(3S,5R)-1-[2-(2,5-dimethylphenyl)acetyl]-5-(pyrrolidine-1-carbonyl)piperidine-3-carboxylic acid
2-{1-[(1-cycloheptanecarbonylpiperidin-3-yl)methyl]-1H-1,2,3-triazol-4-yl}ethan-1-ol
7-(2-{[(furan-3-ylmethyl)(methyl)amino]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-5-yl)-[1,2,4]triazolo[4,3-c]pyrimidin-5-amine
(1S,5R)-3-cyclobutanecarbonyl-6-(6-methylpyridine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-4-(1H-pyrazol-3-yl)benzamide
1-(1-{5H,6H-benzo[h]quinazolin-2-yl}-5-(methoxymethyl)-1H-pyrazole-4-carbonyl)-N,N-diethylpyrrolidin-3-amine
4-benzyl-3-[1-(2,2-dimethylpropyl)piperidin-4-yl]-4,5-dihydro-1H-1,2,4-triazol-5-one
ethyl 2-[({[2-(2-methylphenoxy)pyridin-3-yl]methyl}carbamoyl)amino]acetate
6-{[3-(2-methylphenyl)phenyl]methyl}-N-(thiophen-2-ylmethyl)-6-azaspiro[2.5]octane-1-carboxamide
1-(cyclobutylmethyl)-4-[4-cyclopropyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
N-[(2,4-dimethoxyphenyl)methyl]-3-[1-(thiophen-2-ylmethyl)piperidin-3-yl]propanamide
N3-[2-(5,7-difluoro-2-methyl-1H-indol-3-yl)ethyl]piperidine-1,3-dicarboxamide
3-(3-phenyl-1,2,4-oxadiazol-5-yl)-N-{[2-(1H-1,2,4-triazol-1-yl)pyridin-3-yl]methyl}propanamide
1-(4-chlorophenyl)-N-{[1-(1H-pyrazol-3-ylmethyl)piperidin-3-yl]methyl}cyclopropane-1-carboxamide
N-(2-hydroxy-3-phenylpropyl)-2-[(3-methyl-1H-1,2,4-triazol-5-yl)sulfanyl]acetamide
4-[(pyridin-4-ylmethyl)amino]-1-{[2-(trifluoromethyl)phenyl]methyl}pyrrolidin-2-one
2-(furan-2-yl)-1-{pyrazolo[1,5-a]pyridine-3-carbonyl}azepane
4,4,4-trifluoro-N-({1-[2-(2-methoxyphenyl)ethyl]piperidin-4-yl}methyl)-N-methylbutanamide
methyl 6-{2-methyl-3-oxo-4-phenyl-2,9-diazaspiro[5.5]undecan-9-yl}pyrimidine-4-carboxylate
1-ethyl-N,2,5-trimethyl-N-{[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]methyl}-1H-pyrrole-3-carboxamide
N-[2-(5-methyl-1,2-oxazole-4-carbonyl)-1,2,3,4-tetrahydroisoquinolin-7-yl]-1-phenylcyclopropane-1-carboxamide