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6-(2-chlorophenyl)-N,7-dimethyl-8-oxo-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
1-(cyclohexylmethyl)-3-hydroxy-3-[({2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}amino)methyl]piperidin-2-one
3-{[benzyl(ethyl)amino]methyl}-N,8-dimethyl-N-(2-phenylethyl)imidazo[1,2-a]pyridine-2-carboxamide
methyl 1-(benzyloxy)-8-(2,3-dihydro-1-benzofuran-5-ylmethyl)-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylate
8-(3-methylbenzoyl)-3-phenyl-1,8-diazaspiro[4.5]decan-2-one
5-(morpholin-4-ylmethyl)-N-{[3-(trifluoromethoxy)phenyl]methyl}-1,2-oxazole-3-carboxamide
N-{[4-(2,3-dihydro-1H-inden-2-yloxy)-3-methoxyphenyl]methyl}-N-(oxolan-2-ylmethyl)quinoline-8-sulfonamide
2-amino-4-(2-methyl-1H-imidazol-4-yl)-6-[4-(trifluoromethyl)phenyl]pyridine-3-carbonitrile
6-methoxy-3-(2-{1-methyl-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazin-2-yl}-2-oxoethyl)-2,3-dihydro-1H-indol-2-one
N-methyl-N-[2-(4-methylphenoxy)ethyl]-6-oxo-1-(pyridin-2-ylmethyl)piperidine-3-carboxamide
(2R,6R)-4-(3-hydroxybenzoyl)-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
4-[3-({4-[1-(pyrrolidin-1-yl)ethyl]piperidin-1-yl}methyl)imidazo[1,2-a]pyridine-2-carbonyl]morpholine
2-methoxy-1-(4-{2-[2-(1H-pyrazol-1-yl)ethyl]piperidine-1-carbonyl}piperidin-1-yl)ethan-1-one
N-({7-[(3,4-dimethylphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)-3-fluorobenzamide
1-butyl-4-[3-(4H-1,2,4-triazol-4-yl)benzoyl]piperazin-2-one
{[1-(2-chlorophenyl)-1H-pyrazol-4-yl]methyl}({1-[1-(3-fluorophenyl)-5-methyl-1H-pyrazol-4-yl]ethyl})amine
2-(furan-3-ylmethyl)-7-(oxan-4-yl)-2,7-diazaspiro[4.5]decan-6-one
3-acetamido-N-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]-N-(prop-2-en-1-yl)propanamide
N-cyclobutyl-3-{[(1-ethylpiperidin-2-yl)methyl]sulfamoyl}benzamide
8-{[6-(dimethylamino)pyridin-3-yl]methyl}-1-methyl-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
2-hydroxy-N-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}-2-[4-(trifluoromethyl)phenyl]acetamide
2-[(1-cyclopentylpiperidin-4-yl)oxy]-5-methoxy-N-[3-(morpholin-4-yl)propyl]benzamide
3-[1-(3-ethyl-5-methyl-1,2-oxazole-4-carbonyl)piperidin-4-yl]-N-(pyridin-3-ylmethyl)propanamide
(4aS,7aR)-1-(5-chloropyridine-2-carbonyl)-4-propyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-amino-N-[3-(3,5-dimethyl-1H-pyrazol-4-yl)propyl]-6-methylpyrimidine-4-carboxamide
2-amino-6-(2,5-dimethylthiophen-3-yl)-4-[2-(methoxymethyl)pyrimidin-5-yl]pyridine-3-carbonitrile
N-[(2-chlorophenyl)methyl]-N-(2-methoxyethyl)-2,5-dimethyl-1,3-thiazole-4-carboxamide
6-(7-chloro-2,3,4,5-tetrahydro-1,4-benzoxazepine-4-carbonyl)-2,3,4,5-tetrahydropyridazin-3-one
3-(2-hydroxy-4,6-dimethylpyrimidin-5-yl)-1-[3-(1H-imidazol-1-ylmethyl)piperidin-1-yl]propan-1-one
(1s,4s)-4-[3-(3-ethylphenoxy)azetidine-1-carbonyl]cyclohexan-1-ol
5-methyl-N-({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)-N-(pyridin-3-ylmethyl)pyrazine-2-carboxamide
2-(3-methyl-1H-pyrazol-1-yl)-N-[1-(pyrimidin-2-yl)piperidin-3-yl]acetamide
4-hydroxy-N-[1-(1-methyl-1H-pyrazol-5-yl)propyl]-2-(1H-1,2,4-triazol-1-ylmethyl)pyrimidine-5-carboxamide
[3-(3-{[(3aR,6aS)-5-methyl-octahydropyrrolo[3,4-c]pyrrol-2-yl]methyl}phenoxy)propyl]dimethylamine
N-methyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-2-(pyrimidin-5-yl)quinoline-4-carboxamide
N-{[2-(1H-1,3-benzodiazol-1-yl)pyridin-3-yl]methyl}-2-{imidazo[1,2-a]pyridin-3-yl}acetamide
N-{[2-(4-cyclobutaneamidophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-2-(methylsulfanyl)-1,3-thiazole-4-carboxamide
5-(3-cyclopropyl-1,2,4-oxadiazol-5-yl)-N-[2-(pyrazin-2-yl)ethyl]pyridin-2-amine
4-{2-[(6-chloropyridazin-3-yl)oxy]hex-5-en-1-yl}morpholine
2-{3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidin-1-yl}quinoxaline
2-{1-[1-methyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]piperidin-4-yl}-1,2,3,4-tetrahydroisoquinoline
7-fluoro-3-{1-[2-(1-methylpyrrolidin-2-yl)ethyl]-1H-imidazol-2-yl}-1,2-dihydroquinolin-2-one
1-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-4-(1H-imidazol-1-ylmethyl)piperidine
1,3-dimethyl-N-{[4-(piperidine-1-carbonyl)phenyl]methyl}-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
4-benzyl-3-{1-[(1-methyl-1H-imidazol-2-yl)methyl]piperidin-4-yl}-4,5-dihydro-1H-1,2,4-triazol-5-one
2-[4-(1-benzothiophene-5-carbonyl)-1-(furan-2-ylmethyl)piperazin-2-yl]ethan-1-ol
ethyl 1-(4-oxo-4-phenylbutanoyl)-3-(2-phenoxyethyl)piperidine-3-carboxylate
N-methyl-N-[(5-methylfuran-2-yl)methyl]-1-{1-[(6-methylpyridin-2-yl)methyl]piperidin-4-yl}piperidine-4-carboxamide
1-{[5-chloro-1-methyl-3-(5-methyl-1,2-oxazol-3-yl)-1H-pyrazol-4-yl]methyl}azepan-3-amine
1-(3,4-difluorophenyl)-3-(2-methoxyethyl)-5-[(oxolan-2-ylmethoxy)methyl]-1H-1,2,4-triazole