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N-{[7-chloro-5-(2,5-dimethoxyphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-1,5-dimethyl-1H-pyrazole-3-carboxamide
N-[(5,6-dimethyl-1H-1,3-benzodiazol-2-yl)methyl]-2-[1-(2-methoxyethyl)-3-(3-methoxyphenyl)-2,5-dioxopyrrolidin-3-yl]-N-methylacetamide
1-methyl-1-[(3-methylthiophen-2-yl)methyl]-3-{5-[2-(morpholin-4-yl)ethyl]-1,3,4-thiadiazol-2-yl}urea
(3S,4S)-1-{[4-(propan-2-yl)-1,3-thiazol-2-yl]methyl}-4-[4-(pyridin-2-yl)piperazin-1-yl]pyrrolidin-3-ol
N-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-N,1-dimethyl-3-(2-methylpropyl)-1H-pyrazole-5-carboxamide
N,2-dimethyl-N-{[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl}-1,3-benzothiazole-5-carboxamide
N-({5-cyclohexyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-2-hydroxyacetamide
(2S)-3-phenyl-2-(2-{tricyclo[9.4.0.03,8]pentadeca-1(11),3(8),4,6,12,14-hexaen-2-yl}acetamido)propanamide
(1R,5R)-6-[(3-phenyl-1H-pyrazol-4-yl)methyl]-3-(pyridine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
N-[4-({4-[(2-methylphenyl)methyl]-5-oxo-1,4-diazepan-1-yl}methyl)phenyl]acetamide
(3S,4S)-1-(benzenesulfonyl)-4-{[2-(3,4-dimethoxyphenyl)ethyl](methyl)amino}pyrrolidin-3-ol
1-{4-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-2-(1H-1,2,4-triazol-1-yl)propan-1-one
butyl 2-(3-phenyl-1,2,4-oxadiazol-5-yl)pyrrolidine-1-carboxylate
3-{[(1-{5-ethyl-2,3-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}piperidin-3-yl)oxy]methyl}pyridine
1-({1-[6-(3-methylpiperidin-1-yl)pyridine-3-carbonyl]piperidin-4-yl}methyl)pyrrolidin-2-one
(3aS,6aR)-5-(5-chloropyridin-2-yl)-3-[3-(morpholin-4-yl)propyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
N-{[2-(dimethylamino)-6H,7H,8H-cyclopenta[g]quinolin-3-yl]methyl}-N-[2-(dimethylamino)ethyl]cyclohexanecarboxamide
methyl({1-[1-(thiolan-3-yl)piperidin-4-yl]-1H-1,2,3-triazol-4-yl}methyl)amine
(2S,4R)-4-(4-cyanobenzamido)-N-(3-phenylpropyl)pyrrolidine-2-carboxamide
ethyl 1-[5-(3-methyl-1,2,4-oxadiazol-5-yl)pyridin-2-yl]piperidine-3-carboxylate
1-({3-[4-(piperidin-1-yl)piperidine-1-carbonyl]-1,2-oxazol-5-yl}methyl)piperidin-4-ol
N-({6-cyclopentyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-2-(pyridin-3-yl)acetamide
N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-5,7-dimethylpyrazolo[1,5-a]pyrimidine-2-carboxamide
2-({[(3R,4R)-1-(5-chlorothiophene-2-carbonyl)-4-(hydroxymethyl)pyrrolidin-3-yl]methyl}(methyl)amino)ethan-1-ol
2-[(1S,5R)-3-(3,4-dimethylbenzoyl)-7-oxo-3,6-diazabicyclo[3.2.2]nonan-6-yl]-N,N-dimethylacetamide
N-{2-[3-cyclopropyl-1-(quinolin-8-yl)-1H-1,2,4-triazol-5-yl]ethyl}-N-methylmethanesulfonamide
N-ethyl-1-[(4-methylphenyl)methyl]-5-oxo-N-(pyridin-4-ylmethyl)pyrrolidine-3-carboxamide
3-{5-[(4-phenylphenyl)methyl]-1,3,4-oxadiazol-2-yl}-N-(pyridin-3-ylmethyl)propanamide
2-(4-ethylpiperazin-1-yl)-N-{1-[(2-fluorophenyl)methyl]piperidin-3-yl}-N-methylacetamide
3-[(3S,7S,8aS)-3-[(1R)-1-hydroxyethyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(2,3-dichlorophenyl)urea
5-{[(1S,5R)-3-[(4-methyl-1H-imidazol-5-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}-2,1,3-benzothiadiazole
N-({1-[(2-phenyl-1,3-thiazol-5-yl)methyl]piperidin-3-yl}methyl)-1H-indazole-3-carboxamide
[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl][1-(5-methyl-1-phenyl-1H-pyrazol-4-yl)ethyl]amine
2-(dimethylamino)-8-{[5-(oxan-2-yl)furan-2-yl]methyl}-1,3,8-triazaspiro[4.5]dec-1-en-4-one
methyl 1-[(3R,5S)-5-{[2-(4-fluorophenyl)ethyl]carbamoyl}-1-[(4-methoxy-3-methylphenyl)methyl]pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate
(2R,3R,6R)-5-cyclopentyl-3-(2-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
4-[4-cyclopropyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-ethylpiperidine
2-{3-methyl-5-[2-oxo-6-(propan-2-yl)-1,2-dihydropyridin-3-yl]-1H-1,2,4-triazol-1-yl}acetic acid
2-(1-{thieno[3,2-d]pyrimidin-4-yl}pyrrolidin-3-yl)benzoic acid
(1R,3S)-3-(2-hydroxyethoxy)-7-(thiophen-3-ylmethyl)-7-azaspiro[3.5]nonan-1-ol
N-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-2-(pyridin-4-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
N-({3-methoxy-4-[2-(4-methyl-1,3-thiazol-5-yl)ethoxy]phenyl}methyl)-2-(3-methyl-1H-pyrazol-1-yl)-N-[(3S)-2-oxoazepan-3-yl]acetamide
2-[carbamoyl(methyl)amino]-N-[(3R,4S)-4-cyclopropyl-1-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]pyrrolidin-3-yl]acetamide
7-(5-methyl-2-phenylfuran-3-carbonyl)-2,7-diazaspiro[4.4]nonane-1,3-dione
N-{[2-(2,4-dimethoxy-3-methylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-N-(prop-2-yn-1-yl)cyclohexanamine
(2S)-2-hydroxy-N-{[2-(2-methyl-1H-imidazol-1-yl)phenyl]methyl}-2-phenylacetamide
3-(4-{[5-methyl-2-(naphthalen-1-yl)-1,3-oxazol-4-yl]methyl}piperazin-1-yl)propanamide
7-methoxy-N,4-dimethyl-N-[2-(2-methylpiperidin-1-yl)ethyl]quinazolin-2-amine
N-(1-methoxypropan-2-yl)-4-{[1-(pyridin-2-ylmethyl)piperidin-4-yl]oxy}benzamide
N-{2-[4-({[(3-hydroxy-4-methoxyphenyl)methyl](methyl)amino}methyl)-5-methyl-1,3-oxazol-2-yl]phenyl}methanesulfonamide