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1-[(1-ethyl-5-methyl-1H-pyrazol-4-yl)methyl]-N-[4-(1H-indol-2-yl)phenyl]piperidine-4-carboxamide
(1R,3S)-3-[(2,1,3-benzothiadiazol-5-ylmethyl)(methyl)carbamoyl]cyclopentane-1-carboxylic acid
N-[(2R,3R)-2-methoxy-1'-{[4-(propan-2-yl)-1,3-thiazol-2-yl]methyl}-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]thiophene-2-carboxamide
{[3-(2-fluoro-4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}(furan-3-ylmethyl)methylamine
methyl (2S,4S)-1-[(4-ethylphenyl)methyl]-4-(2-methyl-1,2,3,4-tetrahydroisoquinoline-3-amido)pyrrolidine-2-carboxylate
8-[(2,3-difluorophenyl)methyl]-2-(2-methoxyethyl)-2,8-diazaspiro[5.5]undecan-3-one
ethyl 3-benzyl-1-[(2-methyl-1,3-thiazol-5-yl)methyl]piperidine-3-carboxylate
3-(2-phenyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-N-{[1-(pyrimidin-2-yl)piperidin-3-yl]methyl}propanamide
2-[(3-ethyl-1H-1,2,4-triazol-5-yl)sulfanyl]-N,N-bis(pyridin-3-ylmethyl)acetamide
6-[(2-fluorophenyl)methoxy]-1-[(4-methoxyphenyl)methyl]-4-[5-oxo-1-(pyridin-3-ylmethyl)pyrrolidine-3-carbonyl]-1,4-diazepan-2-one
2-(dimethylamino)-2-(3-fluorophenyl)-N-methyl-N-(1H-pyrazol-3-ylmethyl)acetamide
N-[(5-methylfuran-2-yl)methyl]-2-(4H-1,2,4-triazol-4-yl)pyridine-4-carboxamide
4,5-dimethyl-3-{[5-(pyridin-3-yl)-1,3,4-oxadiazol-2-yl]methyl}-2,3-dihydro-1,3-oxazol-2-one
6-{2-[4-(3-chloro-4-fluorophenyl)-1H-1,2,3-triazol-1-yl]ethyl}-2-methylpyrimidin-4-ol
2-{4-[(5-ethylpyridin-2-yl)methyl]piperazin-1-yl}pyridine-3-carbonitrile
2-[1-(2-ethyl-4-methyl-1,3-oxazole-5-carbonyl)piperidin-3-yl]-1H-1,3-benzodiazole
1-(4-{[3-(1H-indol-1-yl)propyl]amino}-2-methyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl)ethan-1-one
N-[2-(azepan-1-yl)-2-phenylethyl]-1-(methoxymethyl)cyclobutane-1-carboxamide
[(4S)-4-amino-5-{4-[(4-fluorophenyl)methyl]piperidin-1-yl}-5-oxopentyl]urea
1-(2-fluoro-4-methoxyphenyl)-2-{pyrazolo[1,5-a]pyrimidine-3-carbonyl}-1H,2H,3H,4H,9H-pyrido[3,4-b]indole
2-{1-[4-(propan-2-yloxy)benzoyl]pyrrolidin-2-yl}pyridine
3-{7-[(3,4-difluorophenyl)methyl]-2,7-diazaspiro[4.5]decane-2-carbonyl}pyridin-1-ium-1-olate
3-{[1-(5-methylpyrazine-2-carbonyl)piperidin-4-yl]oxy}-N-(pyridin-2-ylmethyl)benzamide
2-(1-methyl-1H-pyrrol-3-yl)-N-({1-[(3-methylphenyl)methyl]pyrrolidin-3-yl}methyl)acetamide
N-(2-methoxyethyl)-2-(3-oxo-2,3-dihydro-1,2-benzothiazol-2-yl)-N-(oxolan-2-ylmethyl)acetamide
1-(4-{[4-(4-fluorophenyl)-1,4-diazepan-1-yl]methyl}phenyl)ethan-1-one
N-[1-(2-methoxyphenyl)-5-oxopyrrolidin-3-yl]-1-methyl-1H-pyrazolo[1,5-a]imidazole-7-carboxamide
N-[1-(2,4-difluorophenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-3-(3-methyl-1H-pyrazol-1-yl)propanamide
(2S)-2-{[5-(3-cyclopropyl-1,2,4-oxadiazol-5-yl)pyridin-2-yl]amino}-4-(methylsulfanyl)butan-1-ol
N-(2-methylprop-2-en-1-yl)-2-(3-oxo-1-{[3-(trifluoromethyl)phenyl]methyl}piperazin-2-yl)acetamide
4-{[1-(dimethylsulfamoyl)piperidin-4-yl]oxy}-N-[(2R)-2-hydroxypropyl]benzamide
N-[2-(2-oxo-1,3-oxazolidin-3-yl)ethyl]-2-[2,6,6-trimethyl-1-(2-methylpropyl)-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl]acetamide
2-{1-[(2-fluoro-4-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-[(5-methylpyrazin-2-yl)methyl]acetamide
N-[(1-methyl-1H-pyrazol-4-yl)methyl]-N-(2-methylpropyl)-1,1-dioxo-1λ6-thiane-4-carboxamide
methyl 4-(5-{[4-(5-chloropyridin-2-yl)piperazin-1-yl]methyl}-1,2,4-oxadiazol-3-yl)benzoate
1-[4-(3-benzyl-1H-pyrazol-5-yl)piperidin-1-yl]pentane-1,2-dione
3-benzyl-8-[(4-methoxyphenyl)methyl]-1-(3-methoxypropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-[1-(furan-2-ylmethyl)piperidin-4-yl]-6-(4H-1,2,4-triazol-4-yl)pyridine-3-carboxamide
2-(2-hydroxypropyl)-9-(3-methyl-1,2-oxazole-5-carbonyl)-2,9-diazaspiro[5.5]undecan-3-one
1-(1-cyclobutylpiperidin-3-yl)-4-phenylpiperazine
2-(4-{1-[2-(1-methylpyrrolidin-2-yl)ethyl]-1H-1,2,3-triazol-4-yl}phenoxy)pyrimidine
(4aS,8aR)-1-(4-hydroxybutyl)-6-(3-methoxypyrazin-2-yl)-decahydro-1,6-naphthyridin-2-one
N-[2-(1H-imidazol-4-yl)ethyl]-2,3-dihydro-1-benzothiophene-2-carboxamide
4-{1-[(4-ethoxyphenyl)methyl]piperidin-4-yl}pyrimidine
(2,1,3-benzoxadiazol-4-ylmethyl)[(1-cyclohexylpiperidin-3-yl)methyl](pyridin-3-ylmethyl)amine
(3S,4S)-1-(benzenesulfonyl)-4-{methyl[(7-methyl-1H-1,3-benzodiazol-2-yl)methyl]amino}pyrrolidin-3-ol
4-(4-ethoxyphenyl)-3-(1-methylpiperidin-3-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
(2E)-1-{3-[4-(2H-1,3-benzodioxol-5-ylmethyl)piperazin-1-yl]piperidin-1-yl}-3-(pyridin-2-yl)prop-2-en-1-one
2-(3-{[3-(3,4-dimethoxybenzoyl)piperidin-1-yl]methyl}-1H-indol-1-yl)acetamide
1-{2-[(1R,5R)-6-benzyl-3,6-diazabicyclo[3.2.2]nonan-3-yl]-2-oxoethyl}-1,2-dihydropyridin-2-one