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N-(1-{4-[(1S,4S)-2-azabicyclo[2.2.1]heptane-2-carbonyl]phenyl}-1H-pyrazol-4-yl)pyridine-3-carboxamide
(3R,4R)-4-(2-ethyl-4-methyl-1H-imidazol-5-yl)-1-methyl-N-[2-(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)ethyl]pyrrolidine-3-carboxamide
N-(1-{imidazo[2,1-b][1,3,4]thiadiazol-6-yl}ethyl)-5-methyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
3-[3-(oxolan-3-yl)propyl]-1-[2-(propan-2-yloxy)phenyl]urea
2-ethoxy-5-[2-(ethoxymethyl)pyrimidin-4-yl]benzoic acid
2-amino-4-[1-(pyrimidin-2-yl)-1H-pyrrol-2-yl]-5,6,7,8-tetrahydroquinoline-3-carbonitrile
(2R,3S,6R)-5-[(4-methyl-1H-imidazol-5-yl)methyl]-3-(4-methylphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
N,2,6-trimethyl-N-[(1-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidin-4-yl)methyl]pyrimidine-4-carboxamide
1-(1-cyclopropanecarbonylpiperidin-4-yl)-N-[(2-methylphenyl)methyl]piperidine-3-carboxamide
{1-[(5-ethylfuran-2-yl)methyl]-4-(2-phenoxyethyl)piperidin-4-yl}methanol
1-{3-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-2-(propan-2-yloxy)ethan-1-one
(1R,5S)-6-({2-methylimidazo[1,2-a]pyridin-3-yl}methyl)-3,6-diazabicyclo[3.2.2]nonane
3,5-dimethyl-2-(4-{5-methyl-[1,2,4]triazolo[1,5-a]pyrimidin-7-yl}piperazine-1-carbonyl)-1H-indole
(3S,4S)-3-{[(2-ethoxynaphthalen-1-yl)methyl](methyl)amino}-4-hydroxy-1λ6-thiolane-1,1-dione
3-(1-{[2-(4-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}pyrrolidin-2-yl)-4-methyl-1,2,5-oxadiazole
3-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl}-1-ethylpyrrolidine
3-(4-{[(2S)-4-methyl-2-(propan-2-yl)piperazin-1-yl]methyl}-1H-pyrazol-1-yl)propanoic acid
2-{1-[(2-fluorophenyl)methyl]-2-methyl-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl}-N-(2-hydroxyethyl)-N-methylacetamide
7-methyl-4-(oxolan-2-ylmethyl)-3,4-dihydro-2H-1,4-benzothiazin-3-one
1-(2-methyl-4-{4-[2-(pyridin-4-yl)ethyl]piperazin-1-yl}-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl)ethan-1-one
2-{1-[(3,5-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-[2-(2-methoxyphenyl)ethyl]acetamide
N-[(5-{[6-(dimethylamino)pyridin-3-yl]methyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl)methyl]cyclobutanecarboxamide
5-(propan-2-yl)-4-{4-[3-(pyrrolidine-1-carbonyl)piperidin-1-yl]piperidin-1-yl}pyrimidine
(2S)-1-acetyl-N-cyclopentyl-N-({1-[2-(2-methylphenyl)ethyl]piperidin-4-yl}methyl)pyrrolidine-2-carboxamide
N-{[2-(1H-imidazol-1-yl)phenyl]methyl}-1-(2-methylpropyl)piperidin-4-amine
2-{2-[(3-methoxyphenyl)methyl]morpholine-4-carbonyl}-N,N-dimethylaniline
2-{3-[(2-methoxyphenyl)methoxy]phenyl}-2-(morpholin-4-yl)acetic acid
2-[4-(2-methoxypyridine-4-carbonyl)piperazin-1-yl]-1-(piperidin-1-yl)ethan-1-one
(3S)-1-benzyl-3-(2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1H-imidazol-1-yl)piperidine
4-[4-(1,2-benzothiazol-3-yl)piperazin-1-yl]pyrimidine-5-carboxylic acid
3-methoxy-N-[1-(3-methyl-1,2,4-oxadiazol-5-yl)ethyl]-4-[(1-methylpiperidin-4-yl)oxy]benzamide
N-[(3-chloro-1-benzothiophen-2-yl)methyl]-N-methyl-2,8-diazaspiro[4.5]decane-3-carboxamide
5-(2H-1,3-benzodioxol-5-yl)-N-(2,3-dihydro-1H-inden-1-yl)-1,2,4-triazin-3-amine
4-(4-fluorophenyl)-1-{[4-(3-hydroxy-3-methylbutyl)phenyl]methyl}piperidin-4-ol
1-(4-fluorophenyl)-4-[1-(5-methoxyfuran-2-carbonyl)piperidin-3-yl]piperazine
6-[1-(4-chlorobenzenesulfonyl)piperidin-3-yl]-2-methyl-3,4-dihydropyrimidin-4-one
N-{[3-(4-fluorophenyl)-1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl}-N-methyloxan-4-amine
3-[6-ethyl-2-(pyrrolidin-1-yl)pyrimidin-4-yl]aniline
N-methyl-6-oxo-N-[3-(1H-pyrazol-1-yl)propyl]-1,4,5,6-tetrahydropyridazine-3-carboxamide
(2R,3R,6R)-3-(2-methoxyphenyl)-N,N-dimethyl-1,5-diazatricyclo[5.2.2.02,6]undecane-5-sulfonamide
2-{[(2-chlorophenyl)methyl]sulfanyl}-N-[1-(2-methoxyethyl)-5-oxopyrrolidin-3-yl]acetamide
N-butyl-3-cyclohexyl-N-(pyridin-3-ylmethyl)-1H-pyrazole-4-carboxamide
N-[(5-cyclopentyl-1,2,4-oxadiazol-3-yl)methyl]-N,1,3-trimethyl-2,6-dioxo-1,2,3,6-tetrahydropyrimidine-4-carboxamide
2-[(3,5-difluorophenyl)methyl]-8-[3-(1H-1,2,3,4-tetrazol-1-yl)propanoyl]-2,8-diazaspiro[4.5]decan-3-one
(1R,7S)-N-methyl-4-oxo-3-[4-(propan-2-yl)phenyl]-N-(1,3-thiazol-2-ylmethyl)-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
1-[(4-fluorophenyl)methyl]-4-{[(3-hydroxyphenyl)methyl]amino}pyrrolidin-2-one
(2S,4R)-1-(2,3-dihydro-1H-inden-2-yl)-N-(2-methoxyethyl)-4-[(naphthalen-1-ylmethyl)amino]pyrrolidine-2-carboxamide
(butan-2-yl)({[3-(1H-pyrazol-1-ylmethyl)phenyl]methyl})(pyridin-4-ylmethyl)amine
2-[1-(2,2-dimethylpropyl)-3-oxopiperazin-2-yl]-N-[(4-propyl-4H-1,2,4-triazol-3-yl)methyl]acetamide
2-cyclopropyl-N-{1-[5-methyl-1-(2-methylphenyl)-1H-pyrazol-4-yl]ethyl}acetamide