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N-(2-methoxy-5-methylphenyl)-1,9-dimethyl-10-oxo-1,4,9-triazaspiro[5.6]dodecane-4-carboxamide
6-{2-ethyl-3-oxo-2,9-diazaspiro[5.5]undecane-9-carbonyl}-1,3-dimethyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
4-({4-[6-oxo-4-(pyridin-3-yl)-1,6-dihydropyrimidin-2-yl]phenyl}methyl)-1λ6-thiomorpholine-1,1-dione
3-(ethylsulfanyl)-1-{4-[4-methyl-5-(morpholin-4-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}propan-1-one
(3aR,6aS)-2-ethyl-1-oxo-5-{pyrazolo[1,5-a]pyridine-3-carbonyl}-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-({2,4-dimethyl-5H,6H-furo[2,3-d]pyrimidin-6-yl}methyl)-1,2-dihydroquinoxalin-2-one
(1R,5S)-8-[6-(methoxymethyl)-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl]-3,8-diazabicyclo[3.2.1]octane
11-[(cyclopropylmethyl)amino]-4-(3-phenylpropyl)-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
N-{2-[(2-butyl-6-methylpyrimidin-4-yl)amino]ethyl}-1-methyl-6-oxo-1,6-dihydropyridine-3-carboxamide
N-{1-[4-(3-oxopiperazine-1-carbonyl)phenyl]-1H-pyrazol-4-yl}furan-3-carboxamide
1-methyl-N-[1-(4-methylpyridin-2-yl)propyl]-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
4-[4-(4-fluorophenyl)butanoyl]-1-(3-methoxyphenyl)piperazin-2-one
(2S,4R)-4-(1H-1,3-benzodiazol-2-ylsulfanyl)-1-[(2Z)-2-chloro-3-phenylprop-2-en-1-yl]-N-(propan-2-yl)pyrrolidine-2-carboxamide
(2R)-2-amino-N-[(2-chlorophenyl)methyl]-3-phenyl-N-(prop-2-en-1-yl)propanamide
2-[1-(2,2-dimethylpropyl)-3-oxopiperazin-2-yl]-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}acetamide
2,6-dimethyl-4-[2-(1H-pyrazol-1-ylmethyl)pyrrolidine-1-carbonyl]quinoline
1-(3,5-dimethylphenyl)-3-({1-[(1-methyl-1H-pyrazol-4-yl)methyl]pyrrolidin-3-yl}methyl)urea
N-{[2-(1H-imidazol-1-yl)phenyl]methyl}-4-(1H-1,2,3,4-tetrazol-1-ylmethyl)benzamide
1-ethyl-N-[3-methoxy-4-(3-methylbutanamido)phenyl]-4,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
2-ethoxy-N-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]acetamide
N-cyclopentyl-N-({3-[(4-fluorophenyl)methoxy]phenyl}methyl)-2-(thiophen-3-yl)acetamide
1-[(1-ethyl-1H-pyrazol-4-yl)methyl]-4-{[3-(3-methoxyphenyl)-1,2-oxazol-5-yl]methyl}piperidin-4-ol
[1-(3-ethyl-1,2,4-oxadiazol-5-yl)ethyl][1-(4-methylphenyl)propan-2-yl]amine
2-[2,5-dioxo-3-phenyl-1-(pyridin-4-ylmethyl)pyrrolidin-3-yl]-N-methyl-N-[1-(4-methyl-1,3-thiazol-2-yl)ethyl]acetamide
1-[4-(4-ethylpiperazine-1-carbonyl)phenyl]-N-[(1-methyl-1H-pyrazol-4-yl)methyl]piperidin-4-amine
methyl 4-({[(2,3-dimethyl-1H-indol-5-yl)methyl]amino}methyl)benzoate
3-{2-[3-(1-methyl-1H-imidazol-2-yl)piperidin-1-yl]-2-oxoethyl}-3,4-dihydroquinazolin-4-one
methyl 4-[5-({4-[(2E)-3-phenylprop-2-en-1-yl]piperazin-1-yl}methyl)-1,2,4-oxadiazol-3-yl]benzoate
N-tert-butyl-2-[3-(3-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]acetamide
6-methyl-5-{[2-(morpholin-4-ylmethyl)piperidin-1-yl]methyl}quinoline
2-{1-[(6-methylpyridin-2-yl)methyl]-4-[(2E)-3-phenylprop-2-en-1-yl]piperazin-2-yl}ethan-1-ol
N-ethyl-N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-2-(phenylamino)pyrimidine-5-carboxamide
2-(dimethylamino)-1-[4-(2-hydroxyethyl)piperidin-1-yl]-2-(2-methylphenyl)ethan-1-one
1-[2-(ethylsulfanyl)ethyl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
5-[(4,5-dimethylfuran-2-yl)methyl]-3-(thiophen-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
N-({1-[(2-methoxypyrimidin-5-yl)methyl]pyrrolidin-3-yl}methyl)cyclohexanecarboxamide
1-[1'-(1-cyclopropyl-1H-pyrrole-2-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]-2-methoxyethan-1-one
4-(prop-2-en-1-yl)-3-[2-(1H-pyrazol-1-yl)ethyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
{[2-(2,2-dimethylpropanesulfonyl)-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}[(2-methoxyphenyl)methyl]methylamine
4-({8-methylimidazo[1,2-a]pyridin-2-yl}methyl)-1-[2-(3-methylphenyl)acetyl]-1,4-diazepan-5-one
7-(4-fluorophenyl)-2-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepin-3-yl}-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
N,N,4-trimethyl-3-[({[(propan-2-yl)carbamoyl]methyl}carbamoyl)methyl]-3,4-dihydro-2H-1,4-benzoxazine-6-carboxamide
7-(1-benzothiophen-3-yl)-4-(1,3-thiazol-4-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N-[7-(4-formyl-1,4-diazepane-1-carbonyl)-1-methyl-2-phenyl-1H-1,3-benzodiazol-5-yl]ethane-1-sulfonamide
3-(4-cyclopentylpiperazin-1-yl)-5-(3-fluorophenyl)-1,2,4-triazine
2-[({5-[1-(2-amino-6-methylpyrimidin-4-yl)piperidin-4-yl]-4-methyl-4H-1,2,4-triazol-3-yl}methyl)(methyl)amino]ethan-1-ol
2-methyl-N-[1-(1H-1,2,4-triazol-5-yl)ethyl]-1,3-thiazole-4-carboxamide
3-({1-[(2E)-3-phenylprop-2-en-1-yl]piperidin-4-yl}oxy)-N-(pyridin-3-ylmethyl)benzamide
N-cyclopropyl-3-({1-[(3,4-difluorophenyl)methyl]piperidin-4-yl}oxy)-4-methoxybenzamide
(3R,4R)-1-[(4-hydroxy-3,5-dimethylphenyl)methyl]-4-(4-methylpiperazin-1-yl)piperidin-3-ol