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2-cyclohexyl-7-[(3-methoxyphenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one
N-(furan-2-ylmethyl)-5-hydroxy-N-(3-methylbutan-2-yl)pyrazine-2-carboxamide
N-[(3S,4R)-1-{2-[(2R,6S)-2,6-dimethylmorpholin-4-yl]-2-oxoethyl}-4-(4-methylphenyl)pyrrolidin-3-yl]acetamide
4-methyl-2-(propan-2-yl)-N-{[1-(propan-2-yl)pyrrolidin-3-yl]methyl}pyrimidine-5-carboxamide
6-{3-[benzyl(methyl)amino]piperidin-1-yl}pyridine-2-carbonitrile
1-(1-{imidazo[2,1-b][1,3]thiazole-6-carbonyl}pyrrolidin-3-yl)-3,5-dimethyl-1H-pyrazole
7,7-dimethyl-2-[2-(1H-pyrazol-1-yl)phenyl]-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
3-[3-(2-methoxyphenyl)-1,2,4-oxadiazol-5-yl]-1-(propan-2-yl)piperidine
3-(2-{2-methyl-1-azatricyclo[6.3.1.04,12]dodeca-2,4,6,8(12)-tetraen-3-yl}ethyl)-1-(1-methyl-1H-1,2,4-triazol-3-yl)urea
5-[1-(4,5,6,7-tetrahydro-1,3-benzothiazole-2-carbonyl)pyrrolidin-2-yl]thiophene-2-carboxamide
2-methyl-6-({3-[3-(pyridin-3-yl)phenyl]-1H-pyrazol-1-yl}methyl)pyridine
N-[(4,6-dimethylpyrimidin-2-yl)methyl]-5-(naphthalen-1-yl)-1,2,4-triazin-3-amine
4-[(2R,3R,6R)-3-(3-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carbonyl]pyridin-3-ol
N-ethyl-5-[3-(pyridin-3-ylmethoxy)piperidine-1-carbonyl]pyrimidin-2-amine
3-[6-amino-4-(2,1,3-benzoxadiazol-4-yl)-5-cyanopyridin-2-yl]-1H-pyrazole-5-carboxylic acid
N-{[2-(4-methylpiperazin-1-yl)pyridin-3-yl]methyl}-4-(1H-pyrazol-4-yl)butanamide
8-[3-(5-methyl-1H-1,2,4-triazol-3-yl)propanoyl]-3-(pentan-2-yl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
2-[5-(methanesulfonylmethyl)pyridin-2-yl]benzoic acid
2-phenyl-1-(1-{[1,2,3,4]tetrazolo[1,5-a]pyridine-6-carbonyl}piperidin-4-yl)ethan-1-ol
1-(3-methylpiperidine-3-carbonyl)-4-(4-phenyl-1H-pyrazol-5-yl)piperidine
6-[4-(4-ethyl-1H-pyrazol-5-yl)piperidin-1-yl]pyrazine-2-carboxamide
(4S)-1-(2,3-dichlorobenzoyl)-4-(methoxymethyl)-3,3-dimethylpiperidin-4-ol
9-{[3-(2-aminoethyl)phenyl]methyl}-2-ethyl-2,9-diazaspiro[5.5]undecan-3-one
3-hydroxy-4-[(2-hydroxyethyl)[(4-{[(2-methoxyphenyl)methyl]amino}-8-methylquinazolin-2-yl)methyl]amino]-1λ6-thiolane-1,1-dione
1-[7-(cyclohexylmethyl)-2,7-diazaspiro[4.5]decan-2-yl]-2,2-dimethylpropan-1-one
N-[2-(2-ethyl-7-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)ethyl]-3-(thiophen-2-yl)propanamide
N-{[1-(cyclohex-2-en-1-yl)-1,2,5,6-tetrahydropyridin-3-yl]methyl}-2-phenoxyacetamide
8-{2-[ethyl(methyl)amino]acetyl}-2-[(2E)-3-phenylprop-2-en-1-yl]-2,8-diazaspiro[4.5]decan-3-one
N-(1-butyl-4-methyl-1H-pyrazol-5-yl)-2,1-benzoxazole-3-carboxamide
N-[2-(1,2,3,4-tetrahydroisoquinolin-2-yl)ethyl]-1H-1,3-benzodiazole-5-carboxamide
2-{1-[(4-fluorophenyl)methyl]-4-{[1-(4-methoxyphenyl)-1H-imidazol-2-yl]methyl}piperazin-2-yl}ethan-1-ol
1-(dimethyl-1,3-thiazole-5-carbonyl)-4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazine
2-methyl-6-{1-[2-(methylamino)pyridine-4-carbonyl]piperidin-4-yl}pyrimidin-4-ol
2-(cyclopropylmethyl)-N-methyl-N-[2-(methylsulfanyl)ethyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
methyl({5-methyl-2-[4-(trifluoromethyl)phenyl]-1,3-oxazol-4-yl}methyl)[1-(1,2-oxazol-3-yl)ethyl]amine
7-(cyclopropylmethyl)-6-(2-fluoro-4-methoxyphenyl)-N-(2-fluoroethyl)-8-oxo-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
N-cyclopentyl-4-{[2-(3,4-dimethoxyphenyl)ethyl]amino}-5-methylthieno[2,3-d]pyrimidine-6-carboxamide
1-{3-[4-(naphthalen-1-yl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}ethan-1-one
5-fluoro-2-(4-{[3-(1H-pyrazol-1-ylmethyl)phenyl]methyl}piperazin-1-yl)pyrimidine
N-tert-butyl-2-[4-(dimethylamino)pyrimidin-2-yl]benzene-1-sulfonamide
N-{2-[2-(pyrimidin-2-yl)-1,3-thiazol-4-yl]ethyl}-1H-pyrrolo[2,3-b]pyridin-6-amine
N-{[3-methyl-7-(4,5,6,7-tetrahydro-1-benzothiophene-3-carbonyl)-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}-1-phenylmethanesulfonamide
(3S,4R)-1-[1-(4-chlorophenyl)cyclobutanecarbonyl]-3-methoxypiperidin-4-amine
1-{2-[1-tert-butyl-3-(thiophen-2-ylmethyl)-1H-1,2,4-triazol-5-yl]ethyl}-5-methyl-1H-1,2,3,4-tetrazole
N-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-5-(4-fluorophenyl)-1,2,4-triazin-3-amine
1-{3,9-diazaspiro[5.5]undecan-3-yl}-2-[(2-hydroxyethyl)(methyl)amino]ethan-1-one
N-{2-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethyl}-2-[3-(trifluoromethyl)phenyl]acetamide
N-{1-[1-methyl-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]piperidin-4-yl}acetamide
N-[(5-cyclopentyl-1,2,4-oxadiazol-3-yl)methyl]-5-oxo-1-[4-(propan-2-yl)phenyl]pyrrolidine-3-carboxamide
2-[(3R,4S)-3-(3-cyanobenzenesulfonamido)-4-cyclopropylpyrrolidin-1-yl]acetamide