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N-methyl-3-(4,5,6,7-tetrahydro-2H-indazol-3-yl)-N-[1-(1,3-thiazol-2-yl)ethyl]propanamide
N-[(7S,8aS)-2-methyl-octahydropyrrolo[1,2-a]piperazin-7-yl]-5-(3-fluorophenoxymethyl)-1H-pyrazole-3-carboxamide
N-[3-(methylsulfanyl)phenyl]-2-[2-(morpholin-4-yl)ethyl]piperidine-1-carboxamide
1-[4-(1,3-benzothiazol-2-yl)-1,4-diazepane-1-carbonyl]cyclopropan-1-amine
N-({7-[3-(1H-indol-3-yl)propanoyl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)furan-2-carboxamide
3-{3-[(1-methylpiperidin-4-yl)methyl]-1,2,4-oxadiazol-5-yl}-6-(pyridin-4-yl)-1,2-dihydropyridin-2-one
5-ethyl-5-{1-[3-(5-methylfuran-2-yl)-1H-pyrazole-5-carbonyl]piperidin-4-yl}imidazolidine-2,4-dione
4-(4-{[2-(cyclohex-1-en-1-yl)ethyl]amino}-5-methylthieno[2,3-d]pyrimidine-6-carbonyl)-1,4-diazepane-1-carbaldehyde
4-ethyl-3-{1-[(1-ethyl-5-methyl-1H-pyrazol-4-yl)sulfonyl]piperidin-4-yl}-4,5-dihydro-1H-1,2,4-triazol-5-one
(1R,5R)-3-benzoyl-6-{[2-(ethylsulfanyl)pyrimidin-5-yl]methyl}-3,6-diazabicyclo[3.2.2]nonane
1-{1-[1-(2-amino-9H-purin-6-yl)piperidin-4-yl]-1H-1,2,3-triazol-4-yl}ethan-1-ol
[(3S,5R)-1-(1H-1,3-benzodiazol-2-ylmethyl)-5-[(4-methyl-1,4-diazepan-1-yl)methyl]piperidin-3-yl]methanol
1-methyl-4-({2-[5-methyl-2-(1H-pyrazol-1-yl)phenyl]-1H-imidazol-1-yl}methyl)piperidin-4-ol
1-(cyclopropylmethyl)-3-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
4-(3-{[4-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]formamido}propyl)-1,2,5-oxadiazole-3-carboxylic acid
2-amino-4-[4-methoxy-3-(1H-1,2,4-triazol-1-ylmethyl)phenyl]-5-methyl-6-(propan-2-yl)pyridine-3-carbonitrile
(5S,9aS,9bS)-5-(2-fluorophenyl)-2-(2-phenylethyl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
7-[(2-fluoro-5-methoxyphenyl)methyl]-2-(1H-pyrazole-4-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
1-(morpholine-4-carbonyl)-4-[3-(propan-2-yl)-1H-pyrazol-1-yl]piperidine-4-carboxylic acid
methyl 4-{[9-methoxy-7-(quinolin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]methyl}benzoate
2-[5-(propan-2-yl)-1,2-oxazol-3-yl]-N-[1-(thiophen-2-ylmethyl)-1H-pyrazol-5-yl]pyrrolidine-1-carboxamide
4-[(1-{1-[(4-fluorophenyl)methyl]piperidin-4-yl}-1H-1,2,3-triazol-4-yl)methyl]morpholine
2-(dimethylamino)-2-(2-methylphenyl)-1-[4-(thiomorpholin-4-yl)piperidin-1-yl]ethan-1-one
1-{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1H-imidazole
(4aR,7aS)-1-cyclobutanecarbonyl-4-(6-methylpyridine-2-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
5-[(2R,3R,6R)-3-(2-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carbonyl]pyridin-2-amine
1-[2-(dimethylamino)ethyl]-N-[1-(furan-2-ylmethyl)piperidin-4-yl]-5-oxopyrrolidine-3-carboxamide
3-(2-{3-[(2-methoxyphenyl)methyl]-1-methyl-1H-1,2,4-triazol-5-yl}ethyl)-3,4-dihydroquinazolin-4-one
2-[4-({[(3S,4R)-4-hydroxyoxolan-3-yl](methyl)amino}methyl)phenoxy]acetic acid
3-{2-[(5-ethylpyrimidin-2-yl)amino]-1-hydroxyethyl}phenol
N-(furan-2-ylmethyl)-1-(prop-2-en-1-yl)-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
5-[5-methyl-6-(4H-1,2,4-triazol-4-yl)pyridin-3-yl]-1,2,3,4-tetrahydroisoquinoline
4-({[1-(dimethylcarbamoyl)piperidin-3-yl]formamido}methyl)benzoic acid
1-[4-(2-ethoxyphenyl)piperazin-1-yl]-3-(trimethyl-1H-pyrazol-4-yl)propan-1-one
3-[2-({2-phenyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl}amino)ethyl]-1,3-oxazolidin-2-one
1-cycloheptyl-N-[2-(4-phenyl-1,3-thiazol-2-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
(3S,4R)-1-[(4-methanesulfonylphenyl)methyl]-4-(2-methylphenyl)pyrrolidine-3-carboxylic acid
[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl](methyl){[5-(oxan-2-yl)thiophen-2-yl]methyl}amine
2-methoxy-6-{[2-(2-methoxyethyl)morpholin-4-yl]methyl}phenol
1-ethyl-2-[(4-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}piperazin-1-yl)methyl]-1H-1,3-benzodiazole
(1S,5R)-6-methyl-3-[(5-methyl-2,1,3-benzothiadiazol-4-yl)sulfonyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
(1-{[2-(morpholin-4-yl)-1,3-thiazol-5-yl]methyl}-3-(2-phenylethyl)piperidin-3-yl)methanol
5-[4-(2-phenylethyl)piperidine-1-carbonyl]-2-(1H-pyrazol-4-yl)pyridine
2-amino-N-[(1-benzyl-1H-pyrazol-4-yl)methyl]-4-methylpyrimidine-5-carboxamide
N-{[1-(pyrrolidine-1-sulfonyl)piperidin-3-yl]methyl}-1H-indole-2-carboxamide
4-methoxy-2-({3-[2-(methylsulfanyl)benzoyl]piperidin-1-yl}methyl)phenol
1-(2-ethoxyphenyl)-4-{[5-methyl-2-(5-methylthiophen-2-yl)-1,3-oxazol-4-yl]methyl}piperazine
1-[5-({6-methylimidazo[2,1-b][1,3]thiazol-5-yl}methyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carbonyl]pyrrolidine
3-({ethyl[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]amino}methyl)-7-methoxy-1,2-dihydroquinolin-2-one
(4S,6R)-4-{[1-(2-fluorophenyl)-3-(2-methylpropyl)-1H-1,2,4-triazol-5-yl]methyl}-6-methyl-1,3-diazinane-2-thione