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(2R,4S)-4-hydroxy-1-[(6-methylpyridin-2-yl)methyl]piperidine-2-carboxylic acid
4-(1H-1,3-benzodiazol-1-yl)-1-(thiophen-3-ylmethyl)piperidine-4-carboxylic acid
(1R,3S)-3-methoxy-7-[(4-methoxypiperidin-1-yl)sulfonyl]-7-azaspiro[3.5]nonan-1-ol
1-{[2-(propan-2-yl)-1,3-oxazol-4-yl]methyl}-4-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepin-3-yl}piperidine
2-tert-butyl-4-hydroxy-N-methyl-N-[2-(2-methyl-1H-indol-1-yl)ethyl]pyrimidine-5-carboxamide
5-({3-cyclopropyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}methyl)-2-(propan-2-yl)pyrimidine
1-(1-cyclopentylpiperidin-4-yl)-N-cyclopropylpiperidine-3-carboxamide
4-{[3-(3-methoxyphenyl)-1,2-oxazol-5-yl]methyl}-1-(1H-pyrazol-3-ylmethyl)piperidin-4-ol
2-{1-[(5-methylfuran-2-yl)methyl]-4-{[1-(2-methylpropyl)-1H-1,3-benzodiazol-2-yl]methyl}piperazin-2-yl}ethan-1-ol
3-[1-(but-2-ynoyl)piperidin-4-yl]-N-(3-methylphenyl)propanamide
methyl (2S,4R)-1-[(2-fluorophenyl)methyl]-4-(quinoline-2-amido)pyrrolidine-2-carboxylate
4-[(2-methoxynaphthalen-1-yl)methyl]-7-(thiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N-benzyl-N-ethyl-6-(4-fluorophenyl)imidazo[2,1-b][1,3]thiazole-3-carboxamide
1-{[1-(3,4-dimethylphenyl)-1H-pyrazol-4-yl]methyl}-3-[(2-methyl-1H-imidazol-1-yl)methyl]piperidine
4-[5-benzyl-1-(2-phenylethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl]morpholine
5-acetyl-N-({5-acetyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-2,4-dimethyl-1H-pyrrole-3-carboxamide
1-(3-methoxy-4-methylphenyl)-3-[1-(3-methyl-1H-pyrazol-5-yl)propan-2-yl]urea
(4aR,7aS)-1-(cyclopropylmethyl)-4-(3-ethoxybenzoyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-[4-({methyl[1-(pyrazin-2-yl)propan-2-yl]amino}methyl)phenyl]acetamide
3-[(3R,4S)-1-(5-ethyl-1H-pyrrole-2-carbonyl)-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propan-1-ol
2-[6-(methylcarbamoyl)pyridin-2-yl]benzoic acid
1-[(4-fluorophenyl)methyl]-2-methyl-3-[2-(1,2-oxazolidin-2-yl)-2-oxoethyl]-4,5,6,7-tetrahydro-1H-indol-4-one
3-[3-({[3-(pyridin-4-yl)propyl]amino}methyl)-1H-indol-1-yl]propanamide
N-[(3S,7S,8aS)-3-methyl-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-4-methoxybenzamide
2,6,8-trimethyl-N-[2-(4H-1,2,4-triazol-4-yl)ethyl]quinoline-4-carboxamide
2,4-dimethyl-5-{[2-(4-methyl-1H-imidazol-5-yl)-1H-imidazol-1-yl]methyl}-1,3-thiazole
1-[4-(piperidin-1-yl)benzoyl]-4-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidine
N-[(1-ethyl-1H-pyrazol-4-yl)methyl]-N-(2-methoxyethyl)-1-methyl-1H-indole-4-carboxamide
1-[3-(3-butyl-4H-1,2,4-triazol-4-yl)phenyl]ethan-1-one
methyl 8-(3-methylbut-2-en-1-yl)-2-oxo-1-(prop-2-en-1-yloxy)-1,8-diazaspiro[4.5]decane-4-carboxylate
1-[(2S,4R)-4-[(4,6-dimethylpyrimidin-2-yl)sulfanyl]-1-[(3-fluorophenyl)methyl]pyrrolidine-2-carbonyl]-4-methyl-1,4-diazepane
1-(3-ethyl-5-methyl-1,2-oxazole-4-carbonyl)-3-(3-fluoro-4-phenylbenzoyl)piperidine
2-fluoro-N-methyl-N-({1-[2-(2-methylphenyl)ethyl]piperidin-3-yl}methyl)benzamide
1-[(2S)-1-(piperidin-4-yl)pyrrolidine-2-carbonyl]-4-(pyridin-4-yl)piperazine
methyl (1R,3S,3aR,6aS)-3-(4-hydroxy-3,5-dimethylphenyl)-1,5-dimethyl-4,6-dioxo-octahydropyrrolo[3,4-c]pyrrole-1-carboxylate
2-amino-3-ethyl-N-[(2,4,5-trifluorophenyl)methyl]-3H-imidazo[4,5-b]pyridine-6-carboxamide
2-({[2-(2-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(thiophen-2-ylmethyl)amino)ethan-1-ol
1-methyl-3-(piperidine-1-carbonyl)-N-(2,2,2-trifluoroethyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
3-(5-{[2-methyl-4-(2-methylphenyl)piperazin-1-yl]methyl}thiophen-3-yl)prop-2-yn-1-ol
2-[1-(2,2-dimethylpropyl)-4-{[4-(methylsulfanyl)phenyl]methyl}piperazin-2-yl]ethan-1-ol
N2-[1-methyl-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]-N1-(pyridin-3-yl)ethane-1,2-diamine
N-benzyl-3-(pyridine-2-carbonyl)piperidine-1-sulfonamide
2-{[3-(2H-1,3-benzodioxol-5-ylmethyl)-3-methylpiperidin-1-yl]methyl}-5-methoxy-4H-pyran-4-one
1-methyl-3-{[4-(pyrimidin-2-yl)-1,4-diazepan-1-yl]methyl}-1,2-dihydroquinolin-2-one
N-(2-{[3-methyl-5-(trifluoromethyl)-1H-pyrazol-1-yl]methyl}propyl)-2-(2-oxopiperidin-1-yl)acetamide
6-oxo-1-[3-(2-oxopyrrolidin-1-yl)propyl]-N-[(2-phenyl-1,3-thiazol-4-yl)methyl]piperidine-3-carboxamide
2-methoxy-N-{2-[(4-methyl-1,2,5-oxadiazol-3-yl)oxy]ethyl}-5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide
5-{1-[(2E)-3-[4-(dimethylamino)phenyl]prop-2-en-1-yl]piperidin-4-yl}-5-methylimidazolidine-2,4-dione
2-(3-{[4-(methoxymethyl)-1H-1,2,3-triazol-1-yl]methyl}piperidin-1-yl)pyridine-3-carboxamide
(2S,4S)-1-benzyl-N-ethyl-4-{[(4-methoxynaphthalen-1-yl)methyl]amino}pyrrolidine-2-carboxamide