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N-[2-(dimethylamino)ethyl]-N-({1-[(2-fluorophenyl)methyl]piperidin-3-yl}methyl)-2-(2-oxopyrrolidin-1-yl)acetamide
5-ethyl-2,3-dimethyl-N-[(4-propyl-4H-1,2,4-triazol-3-yl)methyl]pyrazolo[1,5-a]pyrimidin-7-amine
1-(6-fluoro-4-methylquinazolin-2-yl)-N-(thiophen-2-ylmethyl)azepan-4-amine
2-benzyl-9-{[2-(methoxymethyl)pyrimidin-5-yl]methyl}-2,9-diazaspiro[5.5]undecan-3-one
5-fluoro-2-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-N,N-dimethylpyrimidin-4-amine
N-(1-{7-[(4-methoxy-3-methylphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}-3-methylbutyl)-5-(methoxymethyl)furan-2-carboxamide
N-{[5-(dimethylcarbamoyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}-2,4-dimethyl-1,3-thiazole-5-carboxamide
1-(cyclopropylmethyl)-N-(1,3-thiazol-2-ylmethyl)-5-(thiophene-3-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
N-[(1S,3aS,6aS)-octahydropentalen-1-yl]-2-oxo-6-(propan-2-yl)-1,2-dihydropyridine-3-carboxamide
(4aS,8aR)-6-(3-phenyl-1,2-oxazole-4-carbonyl)-decahydro-1,6-naphthyridine-4a-carboxylic acid
(3S,4S)-1-(2,2-diphenylethyl)-4-[4-(pyridin-2-yl)piperazin-1-yl]pyrrolidin-3-ol
1-[(diethylcarbamoyl)methyl]-N-(2-{imidazo[2,1-b][1,3]thiazol-6-yl}ethyl)-1H-1,2,3-triazole-4-carboxamide
N-({2-[benzyl(methyl)amino]pyridin-3-yl}methyl)-1-methyl-5-oxopyrrolidine-3-carboxamide
(4aR,8aS)-6-[(3-ethoxy-4-methoxyphenyl)methyl]-1-(2-methoxyethyl)-decahydro-1,6-naphthyridin-2-one
1-(methoxymethyl)-N-{[1-methyl-2-(methylsulfanyl)-1H-imidazol-5-yl]methyl}cyclobutane-1-carboxamide
N-[(1-benzyl-1H-pyrazol-4-yl)methyl]-2-(pyridin-3-yl)pyrimidine-5-carboxamide
N-[1-(4-methoxyphenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-yl]-2-(methylsulfanyl)acetamide
5-(4-methoxyphenyl)-N-{[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-1,2,4-triazin-3-amine
N-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-2-(6-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidin-5-yl)acetamide
N-(piperidin-4-yl)-1-[1-(pyridin-4-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
1-[2-(1-{[3-(2-aminoethyl)phenyl]methyl}piperidin-4-yl)ethyl]pyrrolidin-2-one
8-(furan-3-carbonyl)-2-(pyridin-4-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
N-[(1-{[2,4-dimethyl-6-(1H-pyrazol-1-yl)phenyl]methyl}piperidin-3-yl)methyl]-4-fluorobenzamide
1-[(3,4-difluorophenyl)methyl]-3-hydroxy-3-({methyl[(4-methyl-1,3-thiazol-2-yl)methyl]amino}methyl)piperidin-2-one
2-{2-[2-(5-ethylfuran-2-yl)-1H-imidazol-1-yl]phenyl}ethan-1-ol
N-benzyl-1-(prop-2-en-1-yl)-3-(pyrrolidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
2-ethyl-N-(4-methylphenyl)-3-oxo-2,9-diazaspiro[5.5]undecane-9-carboxamide
7-cyclohexyl-2-(4-methylpiperazine-1-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
2-[2-(2-methoxy-4-methylphenoxymethyl)-1,3-oxazole-4-carbonyl]-1,2,3,4-tetrahydroisoquinoline
3-({[2-(3-fluorophenyl)ethyl]amino}methyl)-5,6,7-trimethoxy-N,N-dimethylquinolin-2-amine
methyl[3-(5-methylfuran-2-yl)butyl]{2-[4-(thiomorpholine-4-carbonyl)-1H-1,2,3-triazol-1-yl]ethyl}amine
(1S,5R)-6-[1-(difluoromethyl)-1H-pyrazole-3-carbonyl]-3-(3-phenylpropyl)-3,6-diazabicyclo[3.2.2]nonane
[(3R,5R)-1-[5-(propan-2-yl)thiophene-3-carbonyl]-5-(pyrrolidin-1-ylmethyl)piperidin-3-yl]methanol
1-[(2-methyl-1,3-thiazol-4-yl)methyl]-4-[2-(1H-pyrazol-1-ylmethyl)phenyl]-1H-1,2,3-triazole
methyl 1-{2-[benzyl(methyl)amino]-2,3-dihydro-1H-indene-2-carbonyl}piperidine-4-carboxylate
2-[1-(4-chloro-1,3-dimethyl-1H-pyrazole-5-carbonyl)piperidin-3-yl]-4-methyl-1H-1,3-benzodiazole
9-[(5-cyclopentyl-1,2,4-oxadiazol-3-yl)methyl]-1-oxa-9-azaspiro[5.5]undecan-5-ol
2-methoxy-N-{[1-(oxan-4-yl)piperidin-3-yl]methyl}pyrimidine-5-carboxamide
1-methyl-N-[(1R,4S,6S)-spiro[bicyclo[2.2.1]heptane-7,1'-cyclopropan]-2-en-6-ylmethyl]-1H-pyrazolo[1,5-a]imidazole-7-carboxamide
ethyl 1-[(2-fluorophenyl)methyl]-4-{[3-(trifluoromethyl)phenyl]methyl}piperidine-4-carboxylate
2-(dimethylamino)-N-{[3-(3-fluorophenyl)-1,2-oxazol-5-yl]methyl}-2-(3-methylphenyl)acetamide
8-methyl-N-[2-(1-methyl-1H-pyrazol-5-yl)ethyl]-4-oxo-1,4-dihydroquinoline-3-carboxamide
4-(3,5-dimethyl-1H-pyrazol-1-yl)-N-methyl-N-[3-(1-methyl-1H-imidazol-2-yl)propyl]benzamide
2-(3-methylbut-2-en-1-yl)-8-(quinoline-7-carbonyl)-2,8-diazaspiro[4.5]decan-3-one
3-[5-(2-methylbutanoyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]propanoic acid
1-{[2-methyl-5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-yl]amino}-3-(pyrrolidin-1-yl)propan-2-ol
3-[5-(1H-indol-3-ylmethyl)-1,3,4-oxadiazol-2-yl]-N-methyl-N-(thiophen-3-ylmethyl)propanamide
2-methyl-4-[(1-phenyl-1H-pyrazol-4-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
1-(4-fluorophenyl)-4-[1-(1-methylcyclohexanecarbonyl)piperidin-3-yl]piperazine
{[2-(cycloheptanesulfonyl)-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}[(4-ethylphenyl)methyl]methylamine