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N-(1-{2-[2-(butan-2-yl)phenoxy]acetyl}piperidin-4-yl)methanesulfonamide
5-[(1R,3S,5S)-3-(4-fluoro-3-methylphenyl)-8-azabicyclo[3.2.1]octane-8-carbonyl]-1-methyl-1,2-dihydropyridin-2-one
(3S,4S)-1-[(1R,5S,6S)-3-azabicyclo[3.1.0]hexane-6-carbonyl]-4-(naphthalen-2-yl)piperidin-3-ol
N-[2-(2-fluorophenyl)-1-[1-(2-methylpropyl)piperidin-4-yl]ethyl]-N-methylthiophene-2-carboxamide
N-(2,1,3-benzothiadiazol-5-ylmethyl)-2-(1,1-dioxo-1λ6-thiolan-3-yl)acetamide
1-{[5-(methoxymethyl)furan-2-yl]methyl}-N-methyl-N-[2-(pyridin-2-yl)ethyl]piperidin-3-amine
5-[(2-chlorophenyl)methyl]-5-[1-(2,2-dimethylpropanoyl)piperidin-4-yl]-3-(2-methoxyethyl)imidazolidine-2,4-dione
(1S,4S)-2-benzyl-5-[5-(propan-2-yl)-1,2-oxazole-3-carbonyl]-2,5-diazabicyclo[2.2.1]heptane
4-{[4-methyl-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]methyl}-1-[3-(5-methylfuran-2-yl)butyl]piperidine
methyl({[5-methyl-2-(3-methylthiophen-2-yl)-1,3-oxazol-4-yl]methyl}){[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl}amine
2-{1-[1-(propan-2-yl)piperidin-4-yl]-4-[(2,3,4-trimethoxyphenyl)methyl]piperazin-2-yl}ethan-1-ol
1-[2-(4-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]-3-(piperidin-1-yl)propan-1-one
1-[4-(1-butyl-1H-imidazol-2-yl)piperidin-1-yl]-3-(1H-pyrrol-1-yl)propan-1-one
N-ethyl-N-[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl]-3-(1-methyl-1H-pyrrol-2-yl)-1H-pyrazole-5-carboxamide
1-[(2-methyl-1,3-thiazol-4-yl)methyl]-4-{[4-(1H-pyrazol-1-ylmethyl)phenyl]methyl}piperazine
N,1-dimethyl-N-[(3-methylthiophen-2-yl)methyl]-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
(3S,4R)-1-[(7-methoxy-2-oxo-1,2-dihydroquinolin-3-yl)methyl]-4-phenylpyrrolidine-3-carboxylic acid
5-(4-cyclohexyl-1,4-diazepane-1-carbonyl)-N-methyl-N-(1,2-oxazol-3-ylmethyl)pyridin-2-amine
2-methoxy-N-[1-methyl-5-(4-phenylazepane-1-carbonyl)-2-(pyridin-3-yl)-1H-1,3-benzodiazol-7-yl]acetamide
2-methyl-4-(1H-pyrazol-1-yl)-6-(2,3,4-trimethoxyphenyl)pyrimidine
9-methoxy-7-(8-methoxy-4-methylquinolin-2-yl)-4-(thiophen-2-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
1'-[5,6-dimethyl-2-(pyrrolidin-1-yl)pyrimidin-4-yl]-5-methyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
4-{1-[(3-propyl-1,2,4-oxadiazol-5-yl)methyl]piperidine-3-carbonyl}morpholine
4-{[2-(3,4-dimethoxyphenyl)ethyl]amino}-N-ethyl-N-(2-hydroxyethyl)-5-methylthieno[2,3-d]pyrimidine-6-carboxamide
N-ethyl-N-(pyridin-4-ylmethyl)-1-(4,5,6,7-tetrahydro-1-benzothiophene-3-carbonyl)piperidin-3-amine
3-methyl-6-[5-(2-methylbutyl)-1,2,4-oxadiazol-3-yl]pyridazine
methyl 5-{3-[2-(2,4-difluorophenyl)ethyl]piperidin-1-yl}-5-oxopentanoate
1-[2-(1-methyl-1H-1,3-benzodiazol-2-yl)pyrrolidin-1-yl]-2-[1-(propan-2-yl)piperidin-4-yl]ethan-1-one
(1R,5R)-6-(2-methoxyethyl)-3-[2-(pyrrolidin-1-yl)benzoyl]-3,6-diazabicyclo[3.2.2]nonane
3-(4-fluorophenyl)-1-[1-(2-hydroxyethyl)-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-5-yl]-3-phenylpropan-1-one
ethyl(2-methylprop-2-en-1-yl){[3-(pyrazin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}amine
1-{2,7-dimethylpyrazolo[1,5-a]pyrimidine-5-carbonyl}-3-(4-fluorophenoxymethyl)piperidine
4-(1-benzyl-1H-pyrazole-4-carbonyl)-1-cyclohexyl-6-(pyridin-4-ylmethoxy)-1,4-diazepan-2-one
(3R,4R)-1-(6-chloroquinolin-4-yl)-4-ethylpiperidine-3,4-diol
2-{[(1-{5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}piperidin-4-yl)oxy]methyl}pyridine
N-[(1,1-dioxo-1λ6-thiolan-3-yl)methyl]-2-(pyrrolidin-1-yl)-5,6,7,8-tetrahydroquinazoline-4-carboxamide
[(4-cyclopropyl-5-{1-[(2-ethylpyrimidin-5-yl)methyl]piperidin-4-yl}-4H-1,2,4-triazol-3-yl)methyl]dimethylamine
methyl 3-acetamido-5-{[(2-fluorophenyl)methyl]amino}-1-methyl-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
(3S,4S)-3-({1-[2-(dimethylamino)-6-ethylpyrimidin-4-yl]piperidin-4-yl}amino)-4-hydroxy-1λ6-thiolane-1,1-dione
(3R,4R)-4-[4-(2-fluorophenyl)piperazin-1-yl]-1-(4,4,4-trifluorobutyl)piperidin-3-ol
2-{[(4-chloro-1-methyl-1H-indazol-3-yl)methyl](pyridin-3-ylmethyl)amino}butan-1-ol
N'-cyclopentyl-N-{[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]methyl}butanediamide
N-[(3S,4R)-1-[(1-benzyl-1H-imidazol-2-yl)methyl]-4-propylpyrrolidin-3-yl]methanesulfonamide
5-(1-benzofuran-2-yl)-3-[4-(2-chlorophenyl)piperazin-1-yl]-1,2,4-triazine
5-cyclobutanecarbonyl-1'-(2-phenylethyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
1-[(3-methoxyphenyl)methyl]-4-[(1R,2R)-2-phenylcyclopropanecarbonyl]piperazin-2-one
1-({4-[3-cyclopropyl-1-(2,2,2-trifluoroethyl)-1H-1,2,4-triazol-5-yl]phenyl}methyl)-5-methyl-1H-1,2,3,4-tetrazole
(2S,4S)-N-ethyl-4-[3-(1H-pyrazol-1-yl)propanamido]-1-(pyridin-3-ylmethyl)pyrrolidine-2-carboxamide
2-{1-[3-(1H-pyrazol-1-ylmethyl)benzoyl]piperidine-3-carbonyl}pyridine
(1S,4S)-2-(2-chlorophenyl)-5-{[2-(prop-2-en-1-yloxy)phenyl]methyl}-2,5-diazabicyclo[2.2.1]heptan-3-one