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4,6-dimethyl-2-[({5-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]furan-2-yl}methyl)sulfanyl]pyrimidine
6-{5-hydroxy-1-oxa-9-azaspiro[5.5]undecane-9-carbonyl}-1,3-dimethyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
3-(3-fluorophenyl)-N-{[3-(pyrimidin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-1H-pyrazole-4-carboxamide
5-[3-(1-methyl-1H-pyrrol-2-yl)-1H-pyrazol-5-yl]-3-[(methylsulfanyl)methyl]-1,2,4-oxadiazole
1-(5-{[6-(hydroxymethyl)-1,4-oxazepan-4-yl]methyl}-1-methyl-1H-pyrrol-3-yl)ethan-1-one
5-[(3-cyclohexylpyrrolidin-1-yl)methyl]-3-phenyl-1,2,4-oxadiazole
8-fluoro-2-({[(3-methyloxetan-3-yl)methyl]amino}methyl)quinolin-4-ol
5-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl}-1-methyl-3-(2-methylpropyl)-1H-pyrazole
1-(6-ethoxy-4-methylquinazolin-2-yl)-N-[(4-phenyl-1,3-thiazol-5-yl)methyl]piperidin-4-amine
3-[(1S,5R)-3-(3-phenylpropyl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-1H-indazole
1-[(2,5-difluorophenyl)methyl]-N-[2-(3-methoxyphenyl)phenyl]piperidine-4-carboxamide
9-{[2-(butan-2-yloxy)phenyl]methyl}-2-(2-hydroxyethyl)-2,9-diazaspiro[5.5]undecan-3-one
(3R,4R)-4-(morpholin-4-yl)-1-[(2E)-3-phenylprop-2-en-1-yl]piperidin-3-ol
8-[(4-methoxypyridin-2-yl)methyl]-2-methyl-2,8-diazaspiro[4.5]decane-3-carboxylic acid
8-methoxy-2-[3-(piperidin-1-ylmethyl)piperidin-1-yl]quinoline
1-benzyl-N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-1H-pyrazole-4-carboxamide
4-[(4-fluorophenyl)methyl]-1-{[3-(3-methylbutyl)-1,2,4-oxadiazol-5-yl]methyl}piperidine
3-(3-chlorobenzoyl)-1-(3-phenylprop-2-yn-1-yl)piperidine
5-fluoro-N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]-1H-indole-2-carboxamide
(1S,5R)-3-[2-(3,4-dimethoxyphenyl)acetyl]-6-propyl-3,6-diazabicyclo[3.2.2]nonan-7-one
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-(furan-2-ylmethyl)piperidin-3-ol
1-(carbamoylmethyl)-N-[2-(2-chloro-6-methylphenoxy)ethyl]piperidine-4-carboxamide
3-(morpholine-4-sulfonyl)-N-[3-(1H-1,2,3-triazol-1-yl)propyl]benzamide
1-[3-(dimethylcarbamoyl)propanoyl]-N-[3-(4-fluorophenyl)phenyl]piperidine-3-carboxamide
4-(2-amino-4-methyl-1,3-benzothiazole-6-carbonyl)-1-(4-methylphenyl)piperazin-2-one
4-[3-(3,5-dimethyl-1H-pyrazol-1-yl)azetidin-1-yl]-6-methyl-2-(piperidin-1-yl)pyrimidine
4-hydroxy-N-{[4-(hydroxymethyl)oxan-4-yl]methyl}-N-methyl-2-(4-methylphenyl)pyrimidine-5-carboxamide
2,3,6-trimethyl-4-[3-(1H-pyrazol-5-yl)piperidine-1-carbonyl]quinoline
3-[1-(5,6-dimethyl-2-oxo-1,2-dihydropyridin-3-yl)-N-methylformamido]-N-methylbutanamide
8-[(5-chloro-3-ethyl-1-methyl-1H-pyrazol-4-yl)methyl]-2-(dimethylamino)-1,3,8-triazaspiro[4.5]dec-1-en-4-one
4-(4-methyl-1H-pyrazol-1-yl)-1-(4,5,6,7-tetrahydro-1,2-benzoxazole-3-carbonyl)piperidine-4-carboxylic acid
2-(4-methoxyphenyl)-5-{[3-(4H-1,2,4-triazol-3-yl)piperidin-1-yl]methyl}pyrimidine
3-{2-[(1R,3R,5S)-3-(4-fluoro-3-methylphenyl)-8-azabicyclo[3.2.1]octan-8-yl]-2-oxoethyl}imidazolidine-2,4-dione
N-{[5-(methoxymethyl)-1,2,4-oxadiazol-3-yl]methyl}-1H-pyrrolo[2,3-b]pyridin-6-amine
methyl 1-{ethyl[(1-methylpyrrolidin-3-yl)methyl]carbamoyl}cyclopropane-1-carboxylate
4-ethyl-3-[1-(4-methoxy-2-methylbenzoyl)piperidin-4-yl]-4,5-dihydro-1H-1,2,4-triazol-5-one
methyl 5-{[(2,6-difluorophenyl)methyl]amino}-1-[2-(1H-indol-3-yl)ethyl]-3-(3-methoxypropanamido)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
N-[(3,4-difluorophenyl)methyl]imidazo[1,2-a]pyridine-6-carboxamide
10-methoxy-5-{5-methyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carbonyl}-3,4,5,6-tetrahydro-2H-1,5-benzoxazocine
1-{3-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-2-(pyridin-4-yl)ethan-1-one
1-[4-({[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl](methyl)amino}methyl)-2-methoxyphenoxy]-3-[methyl(propan-2-yl)amino]propan-2-ol
1-(2,6-difluorobenzoyl)-4-[4-(pyrrolidine-1-carbonyl)piperidin-1-yl]piperidine
2-(3-fluoro-4-methylbenzoyl)-7-(oxan-4-yl)-2,7-diazaspiro[4.5]decan-6-one
N-[(5-cyclopropyl-1H-pyrazol-3-yl)methyl]-1-[6-methyl-2-(pyrrolidin-1-yl)pyrimidin-4-yl]piperidin-4-amine
3-(2-methylphenyl)-3-phenyl-N-[2-(pyridin-3-yl)ethyl]propanamide
2-(3-chloro-4-hydroxyphenyl)-N-methyl-N-[2-(oxan-2-yl)ethyl]acetamide
N-[(2S,4R,6S)-2-benzyl-6-[1-(2-methoxyethyl)-1H-imidazol-2-yl]oxan-4-yl]acetamide
N-{[2-(1H-imidazol-1-yl)phenyl]methyl}-6-methyl-2-(pyridin-3-yl)pyrimidin-4-amine
2-[2-(trifluoromethyl)morpholin-4-yl]pyridine-3-carboxylic acid
2-oxo-N-phenyl-2-[4-(1,2,3,4-tetrahydronaphthalen-2-yl)piperazin-1-yl]acetamide