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3-(1,1-dioxo-2,3-dihydro-1λ6-thiophen-3-yl)-1-(trimethyl-1H-pyrazol-4-yl)urea
3,4,5-trimethoxy-N-({5-[4-(methylsulfanyl)phenyl]-2,3-dihydro-1-benzofuran-2-yl}methyl)benzamide
methyl 2-(4-{3-[(2-phenylethyl)carbamoyl]piperidin-1-yl}piperidin-1-yl)acetate
4-(2-methoxyethoxy)-1-({5-methyl-2-[4-(methylsulfanyl)phenyl]-1,3-oxazol-4-yl}methyl)piperidine
1-(1-{5-methyl-6-[(2-methylpyridin-3-yl)oxy]pyrimidin-4-yl}piperidin-3-yl)pyrrolidin-2-one
(2S,4S)-4-[4-({[(3-chlorophenyl)carbamoyl]amino}methyl)-1H-1,2,3-triazol-1-yl]pyrrolidine-2-carboxylic acid
(3aS,6aR)-3-[2-(3-chlorophenyl)ethyl]-5-(1H-pyrrole-2-carbonyl)-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
1-(5-methyl-1,2-oxazole-3-carbonyl)-3-phenylpyrrolidin-3-ol
N-(5-cyano-1,3-thiazol-2-yl)-3-{[(1R,3S,5S)-3-hydroxy-8-azabicyclo[3.2.1]octan-8-yl]methyl}benzamide
3-[1-(2-chlorobenzenesulfonyl)piperidin-4-yl]-N-cyclopropylpropanamide
2-[2-(2,4-difluorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]ethan-1-ol
1-[(2,4-dimethoxy-3-methylphenyl)methyl]-3-(2-methoxyphenoxy)azetidine
N-cyclobutyl-1-(4-fluorophenyl)-2,2-dimethylcyclopropane-1-carboxamide
4-({4-methyl-5-[1-(pyrazin-2-yl)piperidin-3-yl]-4H-1,2,4-triazol-3-yl}methyl)morpholine
methyl 3-(3,5-dimethyl-1H-pyrrole-2-carbonyl)-7-oxo-9-[2-(thiophen-2-yl)ethoxy]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
3-(2H-1,3-benzodioxol-5-yl)-1-{5-hydroxy-1-oxa-9-azaspiro[5.5]undecan-9-yl}propan-1-one
2-(dimethylamino)-N-{[4-(5-methyl-1,2,4-oxadiazol-3-yl)phenyl]methyl}-2-(4-methylphenyl)acetamide
N-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]quinoxaline-6-carboxamide
(3R,4S)-3,4-dimethyl-1-{[3-(morpholin-4-yl)phenyl]methyl}piperidin-4-ol
1-(2,2-dimethylpropyl)-3-hydroxy-3-{[4-(2-methoxyphenyl)piperazin-1-yl]methyl}piperidin-2-one
3-chloro-5-({3-[3-(pyridin-2-ylmethoxy)piperidine-1-carbonyl]-1,2-oxazol-5-yl}methoxy)pyridine
N-[1-(3-fluorophenyl)-4-(2-oxo-1,3-oxazolidin-3-yl)-1H-indazol-3-yl]oxolane-3-carboxamide
ethyl 4-[(4-methoxyphenyl)methyl]-1-(thiophene-2-sulfonyl)piperidine-4-carboxylate
N-ethyl-N-(oxan-4-ylmethyl)-4-(piperidin-3-ylmethyl)benzamide
2-(2-methoxyphenyl)-8-methyl-5-[(6-methylpyridin-2-yl)methyl]-2,3,4,5-tetrahydro-1,5-benzothiazepine
6-(2-oxo-1,2-dihydropyridin-3-yl)-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(15),3(8),6,11,13-pentaen-4-one
N-methyl-N-[1-(pyrazin-2-yl)propan-2-yl]-1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carboxamide
(2S,4S)-1-[(3-chlorophenyl)methyl]-N-methyl-4-[(naphthalen-2-ylmethyl)amino]pyrrolidine-2-carboxamide
(2S,4R)-4-amino-1-[3-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)propanoyl]-N-ethylpyrrolidine-2-carboxamide
(3S,4R)-1-{[4-(3-hydroxy-3-methylbut-1-yn-1-yl)phenyl]methyl}-4-(3-methylthiophen-2-yl)piperidin-3-ol
(1S,6R)-9-[2-(3-fluoro-4-hydroxyphenyl)acetyl]-3,9-diazabicyclo[4.2.1]nonan-4-one
2-{4-[2-(ethoxymethyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl]morpholin-2-yl}ethan-1-ol
4-[(1-{[1-(6-methylpyridazin-3-yl)piperidin-3-yl]methyl}-1H-1,2,3-triazol-4-yl)methyl]thiomorpholine
methyl 4-[({[(2S)-5-oxopyrrolidin-2-yl]methyl}(pyridin-3-ylmethyl)carbamoyl)amino]benzoate
1-(4-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-2-yl}phenyl)-3-(propan-2-yl)urea
benzyl(cyclobutylmethyl){[6-(4-methyl-1,4-diazepane-1-carbonyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl}amine
ethyl 1-[(3-{[1-(naphthalene-2-sulfonyl)piperidin-4-yl]oxy}phenyl)methyl]piperidine-2-carboxylate
1-[5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-yl]-4-[1-(pyrrolidin-1-yl)ethyl]piperidine
3-({[(3-cyclohexyl-1H-pyrazol-4-yl)methyl]amino}methyl)-N,N-diethylpyridin-2-amine
N6-methyl-N6-[(3-phenyl-1,2-oxazol-5-yl)methyl]-9H-purine-2,6-diamine
2-{[3-(3-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]methyl}-5-methoxy-4H-pyran-4-one
2-[4-(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)piperazin-1-yl]-1,3-benzoxazole
N-ethyl-1-[3-(morpholin-4-yl)propyl]-6-oxo-N-[2-(1H-pyrazol-1-yl)ethyl]piperidine-3-carboxamide
N-{3-[2-(hydroxymethyl)pyridin-4-yl]phenyl}acetamide
3-(3-hydroxy-3-methylbutyl)-N-[2-(4H-1,2,4-triazol-4-yl)ethyl]benzamide
1-{6-[4-(hydroxymethyl)phenyl]pyridin-3-yl}ethan-1-one
(4aS,8aR)-6-(1-methyl-1H-imidazole-5-carbonyl)-1-[2-(thiophen-2-yl)ethyl]-decahydro-1,6-naphthyridin-2-one
2-[2-(propan-2-yl)-1H-imidazol-1-yl]-N-{pyrazolo[1,5-a]pyrimidin-3-ylmethyl}propanamide
N-[(1R,3S)-3-(4-ethoxypiperidine-1-carbonyl)cyclopentyl]-4-methyl-1H-imidazole-2-carboxamide
3-[2-(4-fluorophenyl)morpholine-4-carbonyl]-1,5,6-trimethyl-1,2-dihydropyridin-2-one