提示: 按住Ctrl键可以同时选择多个官能团
1-[1,3-dioxo-2-(pyridin-3-ylmethyl)-2,3-dihydro-1H-isoindol-4-yl]-N-methyl-N-(2-phenylethyl)piperidine-4-carboxamide
2-methyl-3-[2-oxo-2-(pyrrolidin-1-yl)ethyl]-1-(oxolan-2-ylmethyl)-4,5,6,7-tetrahydro-1H-indol-4-one
1-{2-[(6-methoxypyrimidin-4-yl)oxy]hex-5-en-1-yl}piperidine-4-carboxylic acid
4-(5-chloro-2-ethoxyphenyl)-6-methyl-2,3-dihydropyridazin-3-one
N-[(3S,4R)-1-(3,5-difluoropyridine-2-carbonyl)-4-(4-methoxyphenyl)pyrrolidin-3-yl]acetamide
9-[(2R)-2-amino-2-cyclohexylacetyl]-2-(pyridin-4-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
(1S,5R)-6-(1-ethyl-5-methyl-1H-pyrazole-3-carbonyl)-3-(pyridin-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
1-[4-({5-methyl-2-[4-(methylsulfanyl)phenyl]-1,3-oxazol-4-yl}methyl)piperazin-1-yl]ethan-1-one
methyl (2S,4R)-4-(dimethylamino)-1-[(8-methoxy-2H-chromen-3-yl)methyl]pyrrolidine-2-carboxylate
(1S,5R)-6-[(1-ethyl-1H-pyrazol-4-yl)methyl]-3-[(4-methoxyphenyl)methyl]-3,6-diazabicyclo[3.2.2]nonane
3-{5-[(2,5-dimethoxyphenyl)methyl]-1,3,4-oxadiazol-2-yl}-N-[2-(3-methoxyphenyl)ethyl]propanamide
N-{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]methyl}-2-oxo-N-(oxolan-2-ylmethyl)propanamide
1-(2-methoxyethyl)-4-[1-(3-phenylphenyl)piperidin-4-yl]piperazine
N-[2-(dimethylsulfamoyl)ethyl]-2-{imidazo[2,1-b][1,3]thiazol-6-yl}acetamide
[(3R,4S)-1-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-4-(morpholin-4-ylmethyl)pyrrolidin-3-yl]methanol
N3-cyclooctyl-4-oxo-1-(oxolan-2-ylmethyl)-N5-(pyridin-2-ylmethyl)-1,4-dihydropyridine-3,5-dicarboxamide
methyl 9-[(4-fluorophenyl)methoxy]-7-oxo-3-(1,3-thiazol-2-ylmethyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
8-[2-(5-methyl-3-oxo-2,3-dihydro-1H-pyrazol-4-yl)acetyl]-3-(3-methylbutyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
2-(5-methyl-1H-pyrazol-1-yl)-1-[6-(morpholine-4-sulfonyl)-1,2,3,4-tetrahydroisoquinolin-2-yl]ethan-1-one
4-(3-fluorophenoxy)-1-(pyridin-4-yl)piperidine-4-carboxylic acid
1-({3-[(1S,4S)-2-azabicyclo[2.2.1]heptane-2-carbonyl]-1H-pyrazol-5-yl}methyl)-2-methyl-1H-1,3-benzodiazole
3-[2-(4-chlorophenyl)morpholine-4-carbonyl]-1-ethyl-4,6-dimethyl-1,2-dihydropyridin-2-one
1-{1-[3-(1-methyl-1H-pyrazol-5-yl)propanoyl]piperidin-4-yl}-2,3-dihydro-1H-1,3-benzodiazol-2-one
2-{4-[(4-fluorophenyl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}-1-phenoxypropan-2-ol
N-methyl-3-(6-methyl-2-oxo-1,2-dihydropyridin-1-yl)-N-(quinolin-5-ylmethyl)propanamide
1-{2-[(3aS,6aS)-octahydropyrrolo[2,3-c]pyrrol-1-yl]-2-oxoethyl}-3-methyl-1,2-dihydroquinoxalin-2-one
2-methyl-4-(4-{1-[2-methyl-5-(1H-1,2,3,4-tetrazol-5-yl)phenyl]-1H-imidazol-2-yl}phenyl)but-3-yn-2-ol
5-[4-(3-methoxybenzoyl)piperazine-1-carbonyl]-1-methyl-1,2-dihydropyridin-2-one
3-acetyl-N-benzyl-N-(cyclobutylmethyl)-1H-pyrazole-5-carboxamide
1-cyclopentyl-5-oxo-N-[3-(1H-1,2,4-triazol-1-yl)propyl]pyrrolidine-3-carboxamide
N,N-dimethyl-2-phenyl-2-(2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1H-imidazol-1-yl)acetamide
(1R,3S)-3-(2-aminoethoxy)-7-{[4-(difluoromethoxy)phenyl]methyl}-7-azaspiro[3.5]nonan-1-ol
[1-ethyl-5-({2-[(oxolan-2-ylmethyl)amino]pyrimidin-5-yl}methyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-3-yl]methanol
4-[3-(1H-1,2,3,4-tetrazol-1-yl)-1H-pyrazole-4-carbonyl]-2-(trifluoromethyl)morpholine
(1R,5S,6R)-3-[(4-methoxy-3-methylphenyl)methyl]-N-[2-(1H-pyrazol-4-yl)ethyl]-3-azabicyclo[3.1.0]hexane-6-carboxamide
2-cyclobutanecarbonyl-7-[(3,4-difluorophenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one
1-(4-{3-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidine-1-carbonyl}phenyl)ethan-1-one
5-cyclopropanecarbonyl-1'-[(3-fluorophenyl)methyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
2-amino-4-(3,5-difluorophenyl)-6-(furan-2-ylmethyl)-5,6,7,8-tetrahydro-1,6-naphthyridine-3-carbonitrile
1-[4-(3-phenylpropyl)-1,4-diazepan-1-yl]-2-(pyridin-3-yl)ethan-1-one
N-[(3,4-dimethoxyphenyl)methyl]-N-methyl-2-{[methyl(1,2-oxazol-3-ylmethyl)amino]methyl}quinazolin-4-amine
1-(2-methoxy-4-methyl-1,3-thiazole-5-carbonyl)-4-(4-phenyl-1H-pyrazol-5-yl)piperidine
N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide
N-[(5-fluoro-2-methylphenyl)methyl]-1,3-dimethyl-6-(pyridin-2-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
1-methyl-N-[1-(3-methylphenyl)cyclopropyl]-2-oxo-1,2-dihydroquinoline-3-carboxamide
5-[(2S)-2-hydroxypropanoyl]-N-(pyridin-2-ylmethyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
{2-[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]ethyl}({[2-(pyrrolidine-1-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl})amine
(4S)-1-[(1-benzyl-1H-imidazol-5-yl)methyl]-3,3,4-trimethylpiperidin-4-ol
N-(3,4-dihydro-1H-2-benzopyran-1-ylmethyl)-3-phenyl-1,2-oxazole-5-carboxamide
5-(1H-1,3-benzodiazol-1-ylmethyl)-N-(thiophen-3-ylmethyl)-1H-pyrazole-3-carboxamide