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4-(1-{1-[(2,4-dimethylphenyl)methyl]piperidin-4-yl}-1H-1,2,3-triazole-4-carbonyl)morpholine
6-(2-chlorophenyl)-N-{2-[(3-methyl-1H-1,2,4-triazol-5-yl)sulfanyl]ethyl}imidazo[2,1-b][1,3]thiazole-3-carboxamide
(1S,5R)-6-(2-ethylpyrimidine-5-carbonyl)-3-(pyrazine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
7-[2-(3-fluorophenyl)piperidine-1-carbonyl]-1,2,3,4-tetrahydroquinoxalin-2-one
N-cyclopropyl-3-[1-methyl-5-(pyrrolidine-1-sulfonyl)-1H-1,3-benzodiazol-2-yl]propanamide
(1S,5R)-6-[2-methyl-5-(propan-2-yl)furan-3-carbonyl]-3-(pyridine-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
(1S,5R)-3-(2H-1,3-benzodioxol-5-ylmethyl)-3,9-diazabicyclo[3.3.2]decan-10-one
(2R,3R)-3-amino-1'-(quinolin-2-ylmethyl)-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
1-[(2-fluoro-4-methoxyphenyl)methyl]piperidine-4-carbonitrile
1-ethyl-N-methyl-3-(piperidine-1-carbonyl)-N-(thiophen-3-ylmethyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
9-{[2-(butylsulfanyl)pyrimidin-5-yl]methyl}-1,4-dimethyl-1,4,9-triazaspiro[5.5]undecane
3-(2-methoxyethyl)-1-[2-(trifluoromethyl)benzoyl]piperidine-3-carboxylic acid
1-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]-4-{[1,2,4]triazolo[4,3-a]pyrimidin-5-yl}piperazine
1-(1'-{[3-(propan-2-yl)-1,2-oxazol-5-yl]methyl}-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl)propan-1-one
4-{[1-(3-chloro-2-fluorobenzoyl)pyrrolidin-3-yl]methyl}benzoic acid
1-(6-{4-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyridin-2-yl)ethan-1-ol
N-[2-(2-oxoimidazolidin-1-yl)ethyl]-5-(oxolan-2-yl)thiophene-2-carboxamide
2-[(2H-1,3-benzodioxol-5-yloxy)methyl]-N-[(4-fluorophenyl)methyl]-N-methyl-1,3-oxazole-4-carboxamide
2-(2-{4-[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]-1H-1,2,3-triazol-1-yl}propyl)pyrazine
7-(5-chloropyridin-2-yl)-4-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
3-{3-benzyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl}quinoline
2-[2-(ethylsulfanyl)-1,3-thiazol-4-yl]-N-{[4-(hydroxymethyl)oxan-4-yl]methyl}acetamide
2-(2-hydroxyphenyl)-N-{[2-(4-methylpiperazin-1-yl)pyridin-3-yl]methyl}acetamide
N-[2-(dimethylamino)ethyl]-N-({1-[(2-methoxyphenyl)methyl]piperidin-3-yl}methyl)-2-oxo-2-phenylacetamide
N-[(2R)-1-(benzyloxy)-3-hydroxypropan-2-yl]-1-cyclohexyl-1H-1,2,3-triazole-4-carboxamide
7-cyclohexyl-2-[2-(2-methyl-1H-imidazol-1-yl)acetyl]-2,7-diazaspiro[4.5]decan-6-one
N-[(3S,7S,8aS)-3-methyl-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-4-bromobenzamide
dimethyl({[4-(4-methylphenyl)-5-(pyridin-2-yl)-1H-imidazol-2-yl]methyl}sulfamoyl)amine
N-(1-{7-[(4-hydroxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-3-methoxypropanamide
N-[1-(furan-2-carbonyl)piperidin-3-yl]-1-(2-methoxyacetyl)piperidine-4-carboxamide
3-{5-hydroxy-1-oxa-9-azaspiro[5.5]undecane-9-carbonyl}-1-methyl-6-(propan-2-yl)-1,2-dihydropyridin-2-one
N-{[4-(cycloheptyloxy)-3-methoxyphenyl]methyl}-3-methoxy-N-(pyridin-2-ylmethyl)benzamide
N-[(4-ethoxyphenyl)methyl]-N-(2-methoxyethyl)-2-(methylamino)pyridine-4-carboxamide
[1-(5-fluoroquinazolin-4-yl)piperidin-4-yl](1-methyl-1H-imidazol-2-yl)methanol
N-({1-[(2-methoxyphenyl)methyl]piperidin-4-yl}methyl)-N-(2-methylpropyl)-2-(propan-2-yl)-1,3-thiazole-4-carboxamide
N-methyl-N'-(5-methyl-1,2-oxazol-3-yl)-N-{[3-(3-methylphenyl)-1,2,4-oxadiazol-5-yl]methyl}ethanediamide
methyl 2-[8-(oxan-4-yl)-2,4-dioxo-1-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decan-3-yl]acetate
1-(2-{[ethyl(pyridin-4-ylmethyl)amino]methyl}-5-methoxyphenoxy)-3-(pyrrolidin-1-yl)propan-2-ol
4-(1H-pyrazol-1-yl)-1-[3-(trimethyl-1H-pyrazol-4-yl)propanoyl]piperidine-4-carboxylic acid
N-cyclopentyl-6-methyl-N-({1-[2-(2-methylphenyl)ethyl]piperidin-4-yl}methyl)pyridine-2-carboxamide
(8R,9aS)-2-(2,3-dihydro-1H-inden-2-yl)-8-hydroxy-octahydro-1H-pyrido[1,2-a]piperazine-1,4-dione
2-amino-4-[2-(cyclopentylmethyl)-1H-imidazol-4-yl]-6-(1H-pyrrol-2-yl)pyridine-3-carbonitrile
(1S,5R)-3-methyl-6-{[4-(pyridin-2-ylmethoxy)phenyl]methyl}-3,6-diazabicyclo[3.2.2]nonane
5-[3-(3,4-dimethoxybenzoyl)piperidine-1-carbonyl]-N-methylpyrimidin-2-amine
3-[(2R,3R,6R)-5-[(2-fluoro-4-methoxyphenyl)methyl]-1,5-diazatricyclo[5.2.2.02,6]undecan-3-yl]phenol
N-(3,4-diethyl-1-methyl-1H-pyrazol-5-yl)-4-[(2-methyl-1,3-thiazol-4-yl)methyl]piperazine-1-carboxamide
N-[2-(2-oxoimidazolidin-1-yl)ethyl]-2-(pyrrolidin-1-yl)-5,6,7,8-tetrahydroquinazoline-4-carboxamide
2-fluoro-6-(4-phenoxybutyl)benzamide
2-(cyclohex-1-en-1-yl)-1-[3-(4-methoxy-3,5-dimethylbenzoyl)piperidin-1-yl]ethan-1-one
2-{[(3,4-dihydro-2H-1-benzopyran-3-yl)amino]methyl}quinolin-4-ol