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N-methyl-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}-2,3-dihydro-1H-indene-5-carboxamide
N-({1-[(1-ethenyl-1H-pyrazol-4-yl)methyl]pyrrolidin-3-yl}methyl)-5-methylpyrazine-2-carboxamide
N-ethyl-2-[4-(pyrimidin-5-yl)phenyl]acetamide
14-(6-methoxy-2H-1,3-benzodioxol-5-yl)-2,8,11-triazatricyclo[7.5.0.02,7]tetradeca-1(9),3,5,7-tetraen-12-one
1-[(2-fluorophenyl)methyl]-4-{[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}piperazin-2-one
7-(3-chlorophenyl)-4-(pyrazine-2-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N-{1-[7-(2,2-diphenylethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]-3-methylbutyl}acetamide
1-(5-chloropyridin-2-yl)-4-{[2-(4-methoxy-3-methylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperazine
(3R,4R)-4-[4-(2-fluorophenyl)piperazin-1-yl]-1-(1,3-thiazol-2-ylmethyl)piperidin-3-ol
(2R,3R)-3-{[2-(4-chlorophenyl)ethyl]amino}-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
2-({4-[4-ethyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}methyl)-6-methylpyridine
4-[5-(4-fluorophenyl)-1,3,4-oxadiazol-2-yl]-1-(oxane-2-carbonyl)piperidine
5-[3-(2-methylpiperidin-1-yl)azetidine-1-carbonyl]thiophene-2-carboxylic acid
N-methyl-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}thian-4-amine
(5S)-5-{[(1H-imidazol-2-ylmethyl)(pyridin-3-ylmethyl)amino]methyl}pyrrolidin-2-one
3-[3-(hydroxymethyl)-4-methylpiperazine-1-carbonyl]naphthalen-2-ol
methyl 1-(3,6,7-trimethyl-1-benzofuran-2-carbonyl)piperidine-4-carboxylate
3-(5-{1-[2-(4-methyl-4H-1,2,4-triazol-3-yl)ethyl]-1H-imidazol-2-yl}thiophen-2-yl)prop-2-yn-1-ol
2-(3-fluoro-4-methoxyphenyl)-5-(methanesulfonylmethyl)pyridine
1-[3-(4-chloro-2-methylbenzoyl)piperidin-1-yl]-3-(pyridin-3-yl)propan-1-one
4-(2,5-dimethoxyphenyl)-3-[1-(1H-pyrazol-1-yl)ethyl]-4H-1,2,4-triazole
3-{[4-(1H-1,2,4-triazol-1-yl)phenyl]methyl}-3H,4H-pyrido[2,3-d]pyrimidin-4-one
N-(2-methylpropyl)-1-(prop-2-en-1-yl)-3-(pyrrolidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
3-(3-fluorophenyl)-1-[2-(piperidin-1-yl)ethyl]-6-(thiophene-3-carbonyl)-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
1-(1-{1-[4-(methylsulfanyl)benzoyl]piperidin-4-yl}-1H-1,2,3-triazol-4-yl)ethan-1-ol
3-(3-acetamidophenyl)-4-methoxy-N-methylbenzamide
4-[(4-methyl-3-phenylpiperazin-1-yl)methyl]-2,1,3-benzoxadiazole
2-(2-chloro-6-methoxyphenyl)-5-[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]pyridine
1-[3-(4-methoxyphenoxymethyl)piperidin-1-yl]-2-(4-methyl-1H-pyrazol-1-yl)ethan-1-one
4-methyl-7-{[(pyrazin-2-yl)amino]methyl}-2H-chromen-2-one
(3aR,6aR)-2-{[(1,3-dimethyl-1H-pyrazol-4-yl)carbamoyl]methyl}-5-methanesulfonyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
4-tert-butyl-N-[2-(1H-pyrazol-4-yl)ethyl]benzamide
methyl 5-{[(2,3-difluorophenyl)methyl]amino}-3-(2-methoxyacetamido)-1-methyl-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
N-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carboxamide
3-[1-(5-methoxy-1-methyl-1H-indole-2-carbonyl)piperidin-4-yl]-1,3-oxazolidin-2-one
1-cyclopropanecarbonyl-N-cyclopropyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]piperidine-4-carboxamide
N-{3-[2-(1-ethylpiperidin-3-yl)-1H-imidazol-1-yl]phenyl}acetamide
4-[4-(2-chlorophenyl)piperidin-4-yl]-N-[2-(pyridin-4-yl)ethyl]pyrimidin-2-amine
(propan-2-yl)(quinolin-4-ylmethyl)[(trimethyl-1H-pyrazol-4-yl)methyl]amine
7-(cyclopropylmethyl)-2-[3-(1H-pyrazol-1-yl)propyl]-2,7-diazaspiro[4.5]decan-6-one
4-(1,3-dimethyl-1H-pyrazol-4-yl)-N-methylpyrimidin-2-amine
1-cyclopentyl-4-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-1,4-diazepane
N-ethyl-N-[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl]-2-{8-methylimidazo[1,2-a]pyridin-3-yl}acetamide
1-[6-(2-chlorophenyl)imidazo[2,1-b][1,3]thiazole-3-carbonyl]-2-(2-methoxyethyl)piperidine
2-amino-4-[1-(pyridin-4-yl)-1H-pyrrol-2-yl]-6-(1H-pyrrol-3-yl)pyridine-3-carbonitrile
2-amino-N-[3-(2,3-dihydro-1H-isoindol-2-yl)propyl]-3-ethyl-3H-imidazo[4,5-b]pyridine-6-carboxamide
4-{[2-(1H-indol-3-yl)ethyl]amino}-N,5-dimethyl-N-(2-methylpropyl)thieno[2,3-d]pyrimidine-6-carboxamide
1-[3-({methyl[2-(oxan-4-yl)ethyl]amino}methyl)phenoxy]-3-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-2-ol
1-(2-chloro-4-fluorobenzenesulfonyl)-3-(4-methyl-1H-pyrazol-5-yl)piperidine
2-methyl-N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)pyrrolidin-3-yl]methyl}-6-oxo-1,6-dihydropyrimidine-5-carboxamide