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2-{4-[(1-ethyl-1H-pyrazol-4-yl)sulfonyl]morpholin-3-yl}-N-phenylacetamide
1-[2-amino-2-(3,5-dimethyl-1H-pyrazol-4-yl)acetyl]-N-[(4-methylphenyl)methyl]piperidine-4-carboxamide
1-[2-(2-chlorophenyl)acetyl]-4-(naphthalen-2-ylmethyl)-1,4-diazepan-5-one
4-(1-methyl-1H-imidazol-2-yl)-1-[2-(1-phenyl-1H-pyrazol-4-yl)ethyl]-1H-1,2,3-triazole
(3S,4S)-1-[(1-methyl-1H-imidazol-2-yl)methyl]-4-propylpyrrolidine-3-carboxylic acid
1-[(1-ethyl-1H-pyrazol-4-yl)methyl]-5,5-diphenylpiperidin-2-one
N-(1-{7-[(5-methylfuran-2-yl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-3-phenylpropanamide
3-{[methyl(pyrazin-2-ylmethyl)amino]methyl}-7-(methylsulfanyl)-1,2-dihydroquinolin-2-one
1-[5-({[(3-chlorophenyl)methyl]amino}methyl)-2-methoxyphenoxy]-3-(pyrrolidin-1-yl)propan-2-ol
N-{1-[1-(2H-1,3-benzodioxol-5-ylmethyl)piperidin-4-yl]-2-(2,4-difluorophenyl)ethyl}-N-methylfuran-2-carboxamide
4-chloro-2-[(1S,5R)-3-[(dimethyl-1,2-oxazol-4-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]phenol
4-(4-ethenylphenyl)benzamide
1-ethyl-N-(3-methylbutyl)-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
1-{1,3-dioxo-2-[(trimethyl-1H-pyrazol-4-yl)methyl]-2,3-dihydro-1H-isoindol-4-yl}-N-(prop-2-en-1-yl)piperidine-4-carboxamide
6-ethoxy-2-{[3-(pyridin-2-yl)azetidin-1-yl]methyl}quinoline
5-methanesulfonyl-2-methyl-N-{2-[2-(propan-2-yl)-1,3-thiazol-4-yl]ethyl}pyrimidin-4-amine
N-cyclopropyl-3-(4-methyl-4H-1,2,4-triazol-3-yl)-N-[(trimethyl-1H-pyrazol-4-yl)methyl]propanamide
1-[3-(4-phenylphenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]ethan-1-one
4-{2-[1-(2-methoxyphenyl)-3-(pyridin-4-yl)-1H-1,2,4-triazol-5-yl]ethyl}morpholine
4-{1-[2-(dimethylamino)ethyl]-1H-imidazol-2-yl}-N-(3-fluorophenyl)piperidine-1-carboxamide
3-[5-(4-fluoro-2-methoxyphenyl)-4-phenyl-1H-imidazol-1-yl]propan-1-ol
N-{[6-(trifluoromethyl)pyridin-3-yl]methyl}-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
5-(2H-1,3-benzodioxol-5-ylmethyl)-5-methyl-1-{2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]ethyl}piperidin-2-one
1-(3-fluorophenyl)-3-{1-[1-(2-oxopropanoyl)piperidin-4-yl]-1H-pyrazol-5-yl}urea
N-[1-(3,4-dimethylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-3-(2-oxopyrrolidin-1-yl)propanamide
2-[4-(pyrrolidine-1-carbonyl)piperidin-1-yl]-5,6,7,8-tetrahydroquinoline-3-carbonitrile
(2S)-3-(4-hydroxyphenyl)-2-{[3-(4H-1,2,4-triazol-4-yl)phenyl]formamido}propanamide
N-methyl-2-{3-oxo-1-[(3-phenoxyphenyl)methyl]piperazin-2-yl}-N-(pyridin-2-ylmethyl)acetamide
1-methyl-3-(2-phenylethyl)piperidine
1-[5-(1H-imidazol-1-ylmethyl)furan-2-carbonyl]-2-(pyrrolidine-1-carbonyl)piperazine
2-[3-(methoxymethyl)phenyl]-2-{4-[(1-methyl-1H-imidazol-2-yl)methyl]piperazin-1-yl}acetic acid
2-({3-methyl-1-[(3-methylphenyl)methyl]-1H-1,2,4-triazol-5-yl}methoxy)acetamide
1-(cyclobutylmethyl)-3-hydroxy-3-{[methyl(2,2,6,6-tetramethylpiperidin-4-yl)amino]methyl}piperidin-2-one
N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-1,2,3-thiadiazole-4-carboxamide
1-(2-methoxyethyl)-3-(3-methoxyphenyl)-3-[2-oxo-2-(4-phenylazepan-1-yl)ethyl]pyrrolidine-2,5-dione
1-[(diethylcarbamoyl)methyl]-N-{5H,6H,7H-pyrrolo[2,1-c][1,2,4]triazol-3-ylmethyl}-1H-1,2,3-triazole-4-carboxamide
(3S,4S)-4-(morpholin-4-yl)-1-[5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-yl]pyrrolidin-3-ol
3-({4-[2,4-dimethyl-6-(1H-pyrazol-1-yl)phenyl]-1H-1,2,3-triazol-1-yl}methyl)-5-(propan-2-yl)-1,2,4-oxadiazole
4-[4-(benzyloxy)butanoyl]-1-(4-methylphenyl)piperazin-2-one
N-({5-methanesulfonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-3-methylpiperidine-3-carboxamide
ethyl 4-{[2-methanesulfonyl-1-(oxolan-2-ylmethyl)-1H-imidazol-5-yl]methyl}piperazine-1-carboxylate
2-phenyl-1-[1-(pyrimidin-2-yl)piperidin-4-yl]ethan-1-ol
1-(4-fluorophenyl)-4-{[2-(pyridin-2-yl)pyrimidin-5-yl]methyl}-1,4-diazepane
N-[4-(3-fluorophenyl)phenyl]-1-(pyridin-4-ylmethyl)pyrrolidine-2-carboxamide
4-(1-ethylpiperidine-2-carbonyl)-7-(1,2,3,4-tetrahydroisoquinolin-2-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
(3R,5S)-N-butyl-5-(3-fluorophenoxymethyl)-1-[(4-hydroxyphenyl)methyl]piperidine-3-carboxamide
2-(4-{[3-(4-methoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl}piperazin-1-yl)-N-(propan-2-yl)acetamide
2-{3-[4-(1H-imidazol-2-yl)piperidine-1-carbonyl]phenyl}-2,3-dihydro-1H-isoindole
4,4,4-trifluoro-1-[3-(3-phenylpropanoyl)piperidin-1-yl]butan-1-one
2-(dimethylamino)-N-{[4-(3-fluorophenyl)oxan-4-yl]methyl}-4-methylpyrimidine-5-carboxamide