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N-{[4-benzyl-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]methyl}-3-(3,5-dimethyl-1H-pyrazol-1-yl)propanamide
4-[2-(3-methoxyphenyl)pyrrolidine-1-carbonyl]-3-(3-methylphenyl)-1H-pyrazole
N-(2-hydroxyethyl)-1-[2-(piperazin-1-yl)ethyl]-N-(1,3-thiazol-2-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
1-(2H-1,3-benzodioxol-5-ylmethyl)-4-[1-(1-ethyl-1H-pyrazole-4-carbonyl)piperidin-3-yl]piperazine
2-[(4-methyl-1,3-thiazol-5-yl)methyl]-5-(morpholin-4-yl)-2,3-dihydropyridazin-3-one
N-benzyl-N-(3-hydroxy-2-methylpropyl)-3-(trimethyl-1H-pyrazol-1-yl)propanamide
N-butyl-6-oxo-1-{[3-(trifluoromethyl)phenyl]methyl}piperidine-3-carboxamide
N-(1H-indol-2-ylmethyl)-4-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]butanamide
N-(3,4-dimethylphenyl)-1-(1H-imidazol-4-ylmethyl)piperidin-3-amine
N-{1-[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]ethyl}cyclopentanecarboxamide
2-cyclohexyl-6-[4-(thiophen-2-ylmethyl)piperazine-1-carbonyl]-1,3-benzoxazole
methyl[(1-methylpyrrolidin-2-yl)methyl]({3-[4-(trifluoromethyl)phenyl]-1,2,4-oxadiazol-5-yl}methyl)amine
(2S,4S)-1-{[4-(diethylamino)phenyl]methyl}-N-(pyridin-3-ylmethyl)-4-({[3-(trifluoromethyl)phenyl]methyl}amino)pyrrolidine-2-carboxamide
3-(azepane-1-carbonyl)-1-ethyl-N-[2-(2-fluorophenyl)ethyl]-4,5,6,7-tetrahydro-1H-indazol-5-amine
7-chloro-N-cyclopropyl-3,5-dimethyl-N-(pyridin-2-ylmethyl)-1-benzofuran-2-carboxamide
4-fluoro-3-hydroxy-N-(3-hydroxypropyl)-N-[(5-methylthiophen-2-yl)methyl]benzamide
[(6,7-dimethyl-1H-1,3-benzodiazol-2-yl)methyl][(3-methylthiophen-2-yl)methyl]amine
5-(5-fluoro-4-methoxypyrimidin-2-yl)-8-methylquinoline
7-(pyridin-3-yl)-4-(quinoxalin-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
8-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-1-(3-methylbutyl)-3-(pyridin-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-[(4-methoxyphenyl)methyl]-4-(3-methylphenyl)-4H-1,2,4-triazole
N-{1-[5-methyl-1-(2-methylphenyl)-1H-pyrazol-4-yl]ethyl}-2-oxo-6-phenyl-1,2-dihydropyridine-3-carboxamide
1-{4-[2-methoxy-4-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)phenoxy]piperidin-1-yl}ethan-1-one
8-(2H-1,3-benzodioxol-5-ylmethyl)-1-methyl-3-[3-(pyridin-4-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-(furan-2-ylmethyl)-N-(1-hydroxybutan-2-yl)-1-(4-methylphenyl)cyclopropane-1-carboxamide
ethyl 5-{[4-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)piperazin-1-yl]methyl}-2-oxo-2,3-dihydro-1H-imidazole-4-carboxylate
N-({3-methyl-7-[2-(3-oxo-2,3-dihydro-1H-isoindol-1-yl)acetyl]-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-2H-1,3-benzodioxole-5-carboxamide
5-[(dimethylsulfamoyl)amino]-N,1-dimethyl-2-(2-methylpropyl)-N-(thiophen-3-ylmethyl)-1H-1,3-benzodiazole-7-carboxamide
N-cyclopropyl-1-{1-[3-(5-methylfuran-2-yl)butyl]piperidin-4-yl}-1H-1,2,3-triazole-4-carboxamide
4-({3-[2-hydroxy-3-(morpholin-4-yl)propoxy]phenyl}methyl)piperazine-1-carboxamide
1-[2-methyl-6-(propan-2-yl)pyrimidin-4-yl]-N-[(3-propyl-1,2-oxazol-5-yl)methyl]piperidin-4-amine
1-[(1s,4s)-4-hydroxycyclohexanecarbonyl]-4-[3-(trifluoromethyl)phenyl]piperidin-4-ol
N-(6-hydroxy-6-methylheptan-2-yl)-2-(2-phenylethyl)-1,3-benzoxazole-5-carboxamide
ethyl 3-[({6-ethyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)amino]pyrrolidine-1-carboxylate
N-[(1-methylpiperidin-4-yl)methyl]-N-(2-phenylethyl)spiro[2.4]heptane-1-carboxamide
4-chloro-2-{6-[(2-methoxyethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}phenol
5-[4-(2-phenylethyl)piperidine-1-carbonyl]-2,1,3-benzoxadiazole
N-(3-hydroxypropyl)-N-methyl-1-[1-(2-phenylethyl)piperidin-4-yl]piperidine-3-carboxamide
9-[2-(2-amino-4,6-dimethylpyrimidin-5-yl)acetyl]-2-(3-methoxypropyl)-2,9-diazaspiro[5.5]undecan-3-one
1-(2-methoxyethyl)-N-{2-[methyl(phenyl)carbamoyl]phenyl}-5-oxopyrrolidine-3-carboxamide
1-{2-[(3-fluorophenyl)methyl]morpholin-4-yl}-3-(4-methoxyphenyl)propan-1-one
1-[(3R,4R)-3-(hydroxymethyl)-4-(morpholin-4-ylmethyl)pyrrolidin-1-yl]-3-(5-methyl-1H-1,2,4-triazol-3-yl)propan-1-one
3-(2-hydroxyethyl)-1-(2-methoxy-6-methylphenyl)-3-[(trimethyl-1H-pyrazol-4-yl)methyl]urea
3-(2-methoxyphenyl)-1-[3-(pyridin-3-ylmethoxy)piperidin-1-yl]propan-1-one
(4aS,7aR)-1-[(3-chloro-4-fluorophenyl)methyl]-4-(2-methoxyethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-{[1-(1-methyl-1H-1,3-benzodiazol-2-yl)-3-(oxan-4-yl)-1H-1,2,4-triazol-5-yl]methyl}acetamide
(dicyclopropylmethyl)({[2-(2,4-dimethoxy-3-methylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl})methylamine
1-[(1-ethylpyrrolidin-3-yl)methyl]-4-phenyl-3-(piperidin-4-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
1-[(5-methylfuran-2-yl)methyl]-3-(prop-2-en-1-yl)piperidine-3-carboxylic acid
N-{2-[2-(hydroxymethyl)piperidin-1-yl]ethyl}-3-methoxy-4-[(1-methylpiperidin-4-yl)oxy]benzamide