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N-[1-(1-methyl-1H-1,2,4-triazol-5-yl)ethyl]-2-(1-propylpiperidin-4-yl)acetamide
2-{4-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}-1-phenoxypropan-2-ol
methyl 2-{8-[4-(1H-indol-3-yl)butan-2-yl]-1-(2-methoxyethyl)-2,4-dioxo-1,3,8-triazaspiro[4.5]decan-3-yl}acetate
N-(2-{7-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-2-phenoxyacetamide
N,3,6,7-tetramethyl-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-1-benzofuran-2-carboxamide
3-methyl-8-[1-(2-phenylethyl)piperidin-4-yl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
2-(3-acetyl-1H-indol-1-yl)-N-{5H,6H,7H-pyrrolo[2,1-c][1,2,4]triazol-3-ylmethyl}butanamide
N-methyl-2-(2-oxo-1,2-dihydroquinolin-1-yl)-N-{[2-(1H-pyrazol-1-yl)phenyl]methyl}acetamide
1-[(3,4-dimethoxypyridin-2-yl)methyl]-4-ethyl-3-(piperidin-4-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
N-methyl-2-{4-[2-(pyridin-3-yl)-1H-imidazol-1-yl]phenoxy}acetamide
1-[2-(cyclopropylmethyl)-7-methyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl]piperidine-3-carbonitrile
4-[4-(3-methylphenyl)-1H-pyrazol-5-yl]-1-(oxolan-3-ylmethyl)piperidine
4-{7-[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}thiomorpholine
N-({3-[2-(dimethylamino)ethoxy]phenyl}methyl)-5-methyl-N-(pyridin-2-ylmethyl)thiophene-2-carboxamide
5-fluoro-2-(3-{[2-(2-methoxyethyl)morpholin-4-yl]methyl}phenyl)-6-methyl-3,4-dihydropyrimidin-4-one
14-(3-cyclohexyl-1H-pyrazol-4-yl)-2,8,11-triazatricyclo[7.5.0.02,7]tetradeca-1(9),3,5,7-tetraen-12-one
1-[4-(1-butyl-1H-imidazol-2-yl)piperidin-1-yl]-2-(morpholin-3-yl)ethan-1-one
2-(butylsulfanyl)-6-[4-(morpholine-4-carbonyl)piperazin-1-yl]pyrimidin-4-amine
(1r,4r)-4-{[(trimethylpyrimidin-4-yl)amino]methyl}cyclohexane-1-carboxamide
(1s,4s)-4-[4-(3-phenylpropyl)-1,4-diazepane-1-carbonyl]cyclohexan-1-ol
4-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]-1-(3-ethoxybenzoyl)piperidine
7-(1-benzothiophen-3-yl)-4-[(2S)-3-hydroxy-2-methylpropyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
8-chloro-2-({4-[(4-methyl-4H-1,2,4-triazol-3-yl)methyl]piperidin-1-yl}methyl)quinoline
1-[(2-methyl-1,3-oxazol-4-yl)methyl]-8-[5-(trifluoromethyl)pyridin-2-yl]-1,8-diazaspiro[4.5]decane
1-(2-benzylmorpholin-4-yl)-3-(1,2-oxazolidin-2-yl)propan-1-one
8-(1-methoxypropan-2-yl)-1-(2-methylpropyl)-3-[3-(pyridin-3-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-(3-phenylpropyl)-5-{2H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl}piperidin-2-one
1-{7-[(5-methyl-1,2-oxazol-3-yl)sulfamoyl]-1,2,3,4-tetrahydroisoquinoline-2-carbonyl}cyclopropane-1-carboxamide
5-fluoro-N-{2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]ethyl}quinazolin-4-amine
(5S,9aS,9bS)-5-(3-methyl-1-propyl-1H-pyrazol-4-yl)-2-[(2-methylphenyl)methyl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
4-(4-methyl-1H-pyrazol-1-yl)-1-(quinolin-5-ylmethyl)piperidine-4-carboxylic acid
ethyl 1-[(5-acetylthiophen-3-yl)methyl]-3-[(3-methoxyphenyl)methyl]piperidine-3-carboxylate
(2-{2-[1-(5-chloro-2-fluorobenzoyl)piperidin-3-yl]-1H-imidazol-1-yl}ethyl)dimethylamine
1-(2-chloro-4-fluoro-5-methylphenyl)-3-ethyl-3-[(3S,4R)-4-hydroxyoxolan-3-yl]urea
5-[3-(5-methyl-1H-pyrazol-1-yl)propanoyl]-1-(2-phenylethyl)-N-(pyridin-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
(4aR,7aS)-1-(2-methoxyacetyl)-4-[2-(2,6,6-trimethylcyclohex-1-en-1-yl)ethyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
{1-[7-fluoro-3-({[(3,4,5-trimethoxyphenyl)methyl]amino}methyl)quinolin-2-yl]piperidin-3-yl}methanol
N4,6-dimethyl-N2-{[4-(4-methylphenyl)-5-(pyridin-2-yl)-1H-imidazol-2-yl]methyl}pyrimidine-2,4-diamine
ethyl 1-(1H-indole-2-carbonyl)-4-[(4-methoxyphenyl)methyl]piperidine-4-carboxylate
(3S,4S)-1-[2-(dimethylamino)pyridine-3-carbonyl]-4-(propan-2-yl)pyrrolidine-3-carboxylic acid
2-(benzyloxy)-1-{3-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidin-1-yl}ethan-1-one
(3aS,6aS)-5-[(4-chlorophenyl)methyl]-1-oxo-2-(prop-2-en-1-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
{[3-(diphenylmethyl)-1,2,4-oxadiazol-5-yl]methyl}(methyl)[2-(oxan-2-yl)ethyl]amine
1-(1,3-thiazol-2-yl)-4-[3-(4H-1,2,4-triazol-4-yl)benzoyl]piperazine
4-(1-methyl-1H-imidazol-2-yl)-1-[4-(2-methyl-2H-1,2,3,4-tetrazol-5-yl)benzoyl]piperidine
1,8-bis(2-phenylethyl)-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
4-[(2,6-dichloro-3-hydroxyphenyl)methyl]-1-phenylpiperazin-2-one
N-[(5-chloro-1H-1,3-benzodiazol-2-yl)methyl]-2-cyclohexyl-N-methyl-1,3-benzoxazole-6-carboxamide
4-[3-(4-methoxyphenoxymethyl)piperidin-1-yl]-4-oxobutanamide
N-[(1-cyclopentylpiperidin-4-yl)methyl]-2-methyl-N-(pyridin-3-ylmethyl)-1,3-benzothiazole-5-carboxamide