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1-{5-chloro-2-[(1-cyclopentylpiperidin-4-yl)oxy]benzoyl}piperidin-3-ol
N-{2-[(1-cyclopropyl-5-oxopyrrolidin-3-yl)formamido]ethyl}-4-fluorobenzamide
1-{[1-(cyclohexylmethyl)-2-methanesulfonyl-1H-imidazol-5-yl]methyl}piperidine-3-carboxamide
3-(2-chlorophenoxy)-1-(furan-2-ylmethyl)azetidine
N-(3,4-dimethoxyphenyl)-1-[2-(2-methylphenyl)benzoyl]piperidin-3-amine
N-cycloheptyl-3-{[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl](methyl)amino}propanamide
dimethyl(2-{2-[1-(7-methyl-1-benzofuran-2-carbonyl)piperidin-4-yl]-1H-imidazol-1-yl}ethyl)amine
N-[2-(1H-1,3-benzodiazol-2-yl)ethyl]-2-[4-(propan-2-yl)morpholin-2-yl]acetamide
8-(5-ethyl-1,2-oxazole-3-carbonyl)-2-methyl-octahydro-1H-pyrazino[1,2-a]piperazin-1-one
3-({3-[2-(4-methoxyphenyl)ethyl]piperidin-1-yl}methyl)pyridine
(3R,4R)-3-cyclopropyl-1-[1-(4-fluorophenyl)piperidin-4-yl]-4-methylpyrrolidin-3-ol
4-({4-methyl-5-[1-(4-methyl-1,2,5-oxadiazole-3-carbonyl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}methyl)morpholine
4-methyl-N-(oxolan-2-ylmethyl)-N-({3-[2-(thiophen-2-yl)ethoxy]phenyl}methyl)benzene-1-sulfonamide
N-{2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]ethyl}-2-(1-oxo-1,2-dihydrophthalazin-2-yl)acetamide
[(5-tert-butyl-1H-pyrazol-3-yl)methyl](oxolan-2-ylmethyl)(pyridin-2-ylmethyl)amine
4-(1H-pyrazol-1-ylmethyl)-1-[3-(1H-1,2,4-triazol-1-yl)propyl]piperidine
1-[(1S,5R)-3-benzoyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-(2-fluorophenyl)ethan-1-one
N-(2-fluoroethyl)-6-(4-methoxyphenyl)-8-oxo-7-(prop-2-en-1-yl)-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
N-(2-hydroxy-2-phenylethyl)-N-methyl-1-(3-phenylpropyl)-1H-1,2,3-triazole-4-carboxamide
5-[4-(adamantan-1-yl)piperazine-1-carbonyl]-1-methyl-1,2-dihydropyridin-2-one
6,7-dimethoxy-4-methyl-N-[3-(1H-1,2,3,4-tetrazol-5-yl)propyl]quinolin-2-amine
5-(diethylamino)-N-methyl-1-(2-phenylethyl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
1-[4-(2-methyl-1H-imidazol-1-yl)phenyl]-N-[2-(pyrazin-2-yl)ethyl]piperidin-4-amine
4-{1-[(3-methyl-1H-pyrazol-5-yl)methyl]pyrrolidin-3-yl}-2-[4-(1H-pyrazol-5-yl)phenyl]pyridine
2-methoxy-4-(4-phenyl-4H-1,2,4-triazol-3-yl)phenol
(3R,4R)-3-cyclopropyl-4-methyl-1-{1-[4-(propan-2-yloxy)phenyl]cyclopentanecarbonyl}pyrrolidin-3-ol
1-ethyl-3-{[3-(2-fluorophenoxy)azetidin-1-yl]methyl}piperidine
4-(dimethyl-1,2-oxazole-4-carbonyl)-1,4-oxazepan-6-ol
4-methyl-3-{4-[2-(4-methyl-1H-imidazol-5-yl)-1H-imidazol-1-yl]phenyl}-4H-1,2,4-triazole
1-[2-(4-methoxyphenyl)ethyl]-5-(3-methoxypropanoyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
1-{2-methyl-5-[2-(3-methyl-1,2-oxazol-5-yl)pyrrolidine-1-carbonyl]phenyl}imidazolidin-2-one
4-[4-(2-methoxyphenyl)piperidin-1-yl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-2-amine
N-[(1-methanesulfonylpiperidin-3-yl)methyl]-3-(2-methyl-1H-indol-1-yl)propanamide
[(2-butyl-5-chloro-1H-imidazol-4-yl)methyl][(1,3-dimethyl-1H-pyrazol-4-yl)methyl]methylamine
2-methyl-8-{[4-(pyrimidin-2-yloxy)phenyl]methyl}-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
4-[(6-chloro-2-fluoro-3-methylphenyl)methyl]-1-methylpiperazine-2-carboxylic acid
3-[({3-methyl-[1,2]oxazolo[5,4-d]pyrimidin-4-yl}amino)methyl]-1λ6-thiolane-1,1-dione
1-[1-(2,3-difluoro-6-methoxybenzoyl)piperidin-4-yl]-3-phenylpropan-1-ol
2,3,6-trimethyl-N-{2-[(pyridin-3-yl)amino]ethyl}quinoline-4-carboxamide
N-(1-{imidazo[2,1-b][1,3,4]thiadiazol-6-yl}ethyl)-1,3-dimethyl-2,6-dioxo-1,2,3,6-tetrahydropyrimidine-4-carboxamide
1-(2-methoxyethyl)-6-oxo-N-[2-(4-phenylpyrimidin-2-yl)ethyl]piperidine-3-carboxamide
(1-{[2-(cyclopentyloxy)phenyl]methyl}-3-(2-methoxyethyl)piperidin-3-yl)methanol
2-(2-fluoro-3-methylphenyl)-2-{4-[(3-methoxyphenyl)methyl]piperazin-1-yl}acetic acid
8-methoxy-N-[(4-methoxy-3,5-dimethylpyridin-2-yl)methyl]-N-methyl-3,4-dihydro-2H-1-benzopyran-3-carboxamide
(3S,4R)-1-[3-(3-methyl-1H-pyrazol-1-yl)propanoyl]-4-(2-methylphenyl)pyrrolidine-3-carboxylic acid
1-(6-{[2-(trifluoromethyl)morpholin-4-yl]sulfonyl}-3,4-dihydro-2H-1,4-benzoxazin-4-yl)ethan-1-one
8-[(2-chloro-6-fluorophenyl)methyl]-1-(2-methoxyethyl)-3-[(3-methoxyphenyl)methyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
6-methoxy-4-oxo-N-[(2E)-3-phenylprop-2-en-1-yl]-N-propyl-1,4-dihydroquinoline-3-carboxamide
{[3-(3-fluoro-4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}(methyl)[2-(morpholin-4-yl)ethyl]amine
1-cyclopentyl-N5-(diphenylmethyl)-N3,N3-diethyl-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide