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N-{[2-(2,6-dimethylphenoxy)pyridin-3-yl]methyl}pyridine-3-carboxamide
1-[(1R,2R)-2-phenylcyclopropanecarbonyl]-4-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidine
N,N-diethyl-2-({4-[3-(3-hydroxy-3-methylbut-1-yn-1-yl)benzoyl]-2-oxo-1-(2-phenylethyl)-1,4-diazepan-6-yl}oxy)acetamide
N-[(dimethyl-1,2-oxazol-4-yl)methyl]-N-methyl-2-(3-oxo-2,3-dihydro-1,2-benzothiazol-2-yl)acetamide
7-{[3-(hydroxymethyl)-4-(propan-2-yloxy)phenyl]methyl}-2-methyl-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-one
5-({3-[5-(4-fluorophenyl)-2-methylpyrimidin-4-yl]piperidin-1-yl}methyl)-2-methoxyphenol
ethyl 5-{[(2,2-dimethyloxan-4-yl)amino]methyl}-1-[4-(4-methoxyphenyl)-1,3-thiazol-2-yl]-1H-pyrazole-4-carboxylate
2-(3-{[2-(5-fluoro-1H-1,3-benzodiazol-2-yl)pyrrolidin-1-yl]methyl}phenoxy)acetamide
7-fluoro-2-methyl-N-{[3-(pyrimidin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}quinoline-4-carboxamide
N-methyl-2-(2-oxopyrrolidin-1-yl)-N-[(1-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidin-4-yl)methyl]acetamide
5-ethyl-N-[(5-fluoro-2-methylphenyl)methyl]-4-(pyrrolidin-1-ylmethyl)furan-2-carboxamide
1-(2,5-dimethylbenzoyl)-3-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidine
5,6-dimethoxy-2-[2-(4-methyl-1,2,3,6-tetrahydropyridin-1-yl)-2-oxoethyl]-1,2-dihydroisoquinolin-1-one
methyl 1-(2-{[6-(4-cyclohexylpiperazin-1-yl)pyridazin-3-yl]oxy}acetyl)piperidine-2-carboxylate
4-methyl-2-{1-[3-(2-methylpropyl)-1,2-oxazole-5-carbonyl]piperidin-3-yl}-1H-1,3-benzodiazole
N-ethyl-1-(2-methylpropyl)-4-oxo-5-(4-phenylpiperidine-1-carbonyl)-1,4-dihydropyridine-3-carboxamide
2-[2-({5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}amino)ethyl]-1,2,3,4-tetrahydrophthalazine-1,4-dione
(1S,5R)-3-[4-(1H-imidazol-1-yl)benzoyl]-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
N-[(1-methyl-1H-imidazol-2-yl)methyl]-3-(piperidin-4-ylmethyl)-N-propylbenzamide
N-[4-(1H-1,3-benzodiazol-2-yl)phenyl]-1-[(2,6-difluorophenyl)methyl]piperidine-4-carboxamide
N,4,6-trimethyl-N-[3-(1-methyl-1H-pyrazol-4-yl)propyl]pyrimidin-2-amine
2-(4-{2-amino-3-ethyl-3H-imidazo[4,5-b]pyridine-6-carbonyl}piperazin-1-yl)-N-(propan-2-yl)acetamide
1-(azepan-1-yl)-3-(4-chloro-2-{[ethyl(2-hydroxyethyl)amino]methyl}phenoxy)propan-2-ol
4-(4-cyclopentylpyrimidin-2-yl)-2-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}morpholine
N-[2-(morpholin-4-yl)ethyl]-5-[2-(propan-2-yloxy)phenyl]pyridin-2-amine
N-(2-phenylethyl)-1-[1-(pyridin-2-ylmethyl)piperidin-4-yl]piperidine-4-carboxamide
5-{[3-(pyridin-3-yl)azetidin-1-yl]methyl}isoquinoline
2-methyl-N-(1,2-oxazol-3-ylmethyl)-4-phenylpyrimidine-5-carboxamide
4-[3-(3-fluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]-2,6-dimethylpyrimidine
methyl 4-(3-acetamidophenyl)-1-ethyl-1H-pyrazole-5-carboxylate
N-(oxolan-2-ylmethyl)-N-(pyridin-4-ylmethyl)-1H-1,2,4-triazole-5-carboxamide
3-methoxy-1-{2-[(1R,2R,6S,7S)-10-oxa-4-azatricyclo[5.2.1.02,6]decan-4-yl]-2-oxoethyl}-1,2-dihydropyridin-2-one
(1R,2R,6S,7S)-N-(6-cyanopyridin-3-yl)-10-oxa-4-azatricyclo[5.2.1.02,6]decane-4-carboxamide
2-[5-(3-cyclohexyl-1H-pyrazole-4-carbonyl)-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-1-yl]ethan-1-ol
2-(1-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}pyrrolidin-2-yl)pyridine
N-[4-({[2-(4-hydroxyphenyl)-2-oxoethyl](methyl)amino}methyl)phenyl]acetamide
2-[5-(2-amino-4-ethyl-1,3-thiazol-5-yl)-1-(2,3-dihydro-1H-inden-5-yl)-1H-1,2,4-triazol-3-yl]acetamide
3-{[6-(2,5-dimethylfuran-3-yl)-7-(3-methylbut-2-en-1-yl)-8-oxo-7H,8H-imidazo[1,2-a]pyrazin-2-yl]formamido}propanamide
2-{[2-(4-fluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-6,7-dimethoxy-1,2,3,4-tetrahydroisoquinoline
1-(3-fluorophenyl)-3-{1-[1-(1H-indole-6-carbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}urea
1-{[2-(2-fluorophenoxy)pyridin-3-yl]methyl}-3-propylurea
4-{3-[(4S)-4-hydroxy-3,3,4-trimethylpiperidine-1-carbonyl]phenyl}-1λ6-thiomorpholine-1,1-dione
ethyl 1-(naphthalen-1-ylmethyl)-4-(oxan-2-ylmethyl)piperidine-4-carboxylate
1-[(3,4-dimethoxypyridin-2-yl)methyl]-3-(2-methylpropyl)-2-oxo-1H,2H,3H-imidazo[4,5-b]pyridine-6-carboxylic acid
5-[6-(trifluoromethyl)pyridin-2-yl]-1,2,3,4-tetrahydroisoquinoline
N,1-dimethyl-N-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
2-(4-methyl-1,2,5-oxadiazol-3-yl)-N-{1-[5-methyl-1-(pyridin-2-yl)-1H-pyrazol-4-yl]ethyl}acetamide
2-[3-(3-fluorophenoxymethyl)-5-(2-methyl-1,3-thiazol-4-yl)-1H-1,2,4-triazol-1-yl]ethan-1-ol
1-{2-[(3R,4R)-3-(hydroxymethyl)-4-(morpholin-4-ylmethyl)pyrrolidin-1-yl]-2-oxoethyl}-1,2-dihydropyridin-2-one
[5-({1-[3-(trifluoromethyl)phenyl]-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl}methyl)furan-2-yl]methanol