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2-(furan-3-carbonyl)-7-[(3-methylphenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one
N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-2-methoxypyridine-3-carboxamide
1-{[3-(2,5-dimethylphenyl)-1H-pyrazol-4-yl]methyl}-4-(5-methylpyridin-2-yl)piperidin-4-ol
4-{5-[(2S)-1-[(1-methyl-1H-imidazol-5-yl)methyl]pyrrolidin-2-yl]-1,2,4-oxadiazol-3-yl}pyridine
2-[4-(4H-1,2,4-triazol-4-yl)benzoyl]-1,2,3,4-tetrahydroisoquinoline
2-{2-[2-(1-ethylpiperidin-4-yl)acetamido]ethyl}-4-methyl-1,3-thiazole-5-carboxylic acid
1'-[2-(benzenesulfonyl)ethyl]-1-methyl-1,2-dihydrospiro[indole-3,4'-piperidine]-2-one
3-{1-[3-(1-methyl-1H-pyrazol-4-yl)propanoyl]piperidin-3-yl}benzoic acid
5-ethyl-N-(pyridin-4-ylmethyl)pyrazolo[1,5-a]pyrimidin-7-amine
N'-(3-chloro-2-methylphenyl)-N-[3-(4-methyl-1,3-thiazol-5-yl)propyl]propanediamide
5-acetyl-N-[furan-2-yl(phenyl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
1-[(3aR,7aS)-5-methyl-2,3,3a,4,7,7a-hexahydro-1H-isoindol-2-yl]-2-(4-methanesulfonylphenyl)ethan-1-one
(4aR,8aR)-2-cyclobutanecarbonyl-7-{[2-(dimethylamino)pyrimidin-5-yl]methyl}-decahydro-2,7-naphthyridin-4a-ol
(2S,4S)-N,N-diethyl-4-(4-{[methyl(pyrrolidine-1-carbonyl)amino]methyl}-1H-1,2,3-triazol-1-yl)pyrrolidine-2-carboxamide
4-{1-[(5-ethylpyridin-2-yl)methyl]-1H-imidazol-2-yl}-N-methylbenzene-1-sulfonamide
[(3R,4S)-1-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-4-[(4-methyl-1,4-diazepan-1-yl)methyl]pyrrolidin-3-yl]methanol
3-(4-chlorophenyl)-N-(1,2-oxazol-3-ylmethyl)-3-phenylpropanamide
2-[(4aS,7aR)-6,6-dioxo-4-(pyrimidin-2-yl)-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]-N-(furan-2-ylmethyl)acetamide
5-methyl-N-{4-[4-(1H-1,2,4-triazol-1-yl)butanamido]phenyl}furan-2-carboxamide
{[1-butyl-2-(4-methylpentanesulfonyl)-1H-imidazol-5-yl]methyl}(methyl)[(trimethyl-1H-pyrazol-4-yl)methyl]amine
ethyl 1-[3-(6-oxo-1,4,5,6-tetrahydropyridazin-3-yl)propanoyl]-4-(2-phenylethyl)piperidine-4-carboxylate
(3aR,7aS)-5-methyl-2-[4-methyl-2-(propan-2-yl)pyrimidine-5-carbonyl]-2,3,3a,4,7,7a-hexahydro-1H-isoindole
(2,1,3-benzoxadiazol-5-ylmethyl)[(2-ethyl-3-methyl-1H-indol-5-yl)methyl]amine
N-[2-(dimethyl-1,3-thiazol-2-yl)ethyl]-2-{[4-(2-fluorophenyl)piperazin-1-yl]methyl}-1,3-oxazole-4-carboxamide
N-(1-cyclopropylethyl)-6-(4-fluorophenyl)-7-(3-methylbut-2-en-1-yl)-8-oxo-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
4'-[2-(1H-indol-3-yl)ethyl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
3-[1-(naphthalen-2-ylmethyl)piperidin-3-yl]-1-[4-(pyridin-2-yl)piperazin-1-yl]propan-1-one
4-[2-({5-methyl-4-[1-(1-methylpiperidine-2-carbonyl)piperidin-3-yl]pyrimidin-2-yl}sulfanyl)ethyl]morpholine
5-[4-(2-methoxybenzoyl)piperazine-1-carbonyl]-4-methylpyrimidine
3-methyl-7-(5-phenoxyfuran-2-carbonyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine
1-(2-{2-methylimidazo[2,1-b][1,3,4]thiadiazol-6-yl}ethyl)-2-(3-methylthiophen-2-yl)-1H-imidazole
3-{1-[(2E)-3-(4-fluorophenyl)prop-2-en-1-yl]piperidin-2-yl}propanoic acid
(1R,2S,3R,4S)-3-amino-N-[2-(4-methoxyphenyl)ethyl]-N-[(1-methylpiperidin-4-yl)methyl]-7-oxabicyclo[2.2.1]hept-5-ene-2-carboxamide
N-(2,3-dihydro-1H-inden-2-yl)-2-(5-phenyl-2H-1,2,3,4-tetrazol-2-yl)acetamide
1-(oxolan-3-ylmethyl)-4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazine
2-[(1S,5R)-3-[3-(4-fluorophenyl)propanoyl]-7-oxo-3,6-diazabicyclo[3.2.2]nonan-6-yl]-N,N-dimethylacetamide
N-{[7-fluoro-2-(4-hydroxypiperidin-1-yl)quinolin-3-yl]methyl}-2-methyl-N-(oxolan-2-ylmethyl)propanamide
1-[2-amino-4-(pyridin-3-yl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl]-3-methylbut-2-en-1-one
N-[1-(4-fluorophenyl)propyl]-2-(hydroxymethyl)-1H-1,3-benzodiazole-5-carboxamide
(2S,4R)-4-amino-N-ethyl-1-[(2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl)sulfonyl]pyrrolidine-2-carboxamide
2-ethyl-8-{[4-(pyrrolidin-1-ylmethyl)thiophen-2-yl]methyl}-2,8-diazaspiro[5.5]undecan-3-one
1-[(4aR,8aR)-4a-hydroxy-7-methanesulfonyl-decahydro-2,7-naphthyridin-2-yl]-2-(5-amino-3-methyl-1H-pyrazol-1-yl)ethan-1-one
N-({1-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]cyclopropyl}methyl)-5-oxo-1-(pyridin-4-ylmethyl)pyrrolidine-3-carboxamide
2-butyl-5-[4-(thiophene-2-carbonyl)piperazine-1-carbonyl]-1,3-benzoxazole
N-[(3,4-dimethoxyphenyl)methyl]-1-methyl-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
N-[2-(benzylsulfanyl)ethyl]-2-cyclopropyl-4-methylpyrimidine-5-carboxamide
5-(2-chlorophenyl)-N-[1-(pyridin-2-yl)propan-2-yl]furan-2-carboxamide
2-{[(2,5-dimethylfuran-3-yl)formamido]methyl}-N,N-dimethyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carboxamide
N-{[1-(2-fluorophenyl)cyclopentyl]methyl}-3-(2-methylpropyl)-1,2-oxazole-5-carboxamide
1-[(1-ethylpiperidin-3-yl)methyl]-4-(1H-pyrrole-2-carbonyl)piperazine