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N-{4-[({[1-(2-hydroxyethyl)piperidin-3-yl]methyl}carbamoyl)methyl]phenyl}butanamide
N-(1H-1,3-benzodiazol-2-ylmethyl)-3-[(4-fluorophenyl)formamido]-N-methylpropanamide
4-fluoro-3-methoxy-N-methyl-N-[(1-methylpiperidin-2-yl)methyl]benzamide
1,3-dimethyl-N-{1-[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]ethyl}-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
(1R,5S,6S)-6-({4-[(3-fluorophenyl)methyl]piperazin-1-yl}methyl)-3-azabicyclo[3.1.0]hexane
1-[(3-chlorophenyl)methyl]-N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
N-{[7-(4-phenylbenzoyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]methyl}-3-(pyridin-3-yl)propanamide
(2R)-2-{[5-(3-methoxyphenoxymethyl)-1H-pyrazol-3-yl]formamido}propanamide
4-benzyl-1-({5-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidin-7-yl}methyl)pyrrolidin-2-one
N-[(3-fluoro-4-methoxyphenyl)methyl]-2-(1H-imidazol-2-yl)benzamide
9-(2-fluoro-5-methylbenzenesulfonyl)-2-methyl-2,9-diazaspiro[5.5]undecan-3-one
2-(4-{[3-(3-chlorobenzoyl)piperidin-1-yl]methyl}phenoxy)ethan-1-ol
N-(2-{7-[(4-methoxy-2,3-dimethylphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-2-phenoxyacetamide
4-[4-(3-hydroxy-3-methylbutyl)benzoyl]-N,N-dimethylpiperazine-1-sulfonamide
N-[2-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)ethyl]-8-methoxy-3,4-dihydro-2H-1-benzopyran-3-carboxamide
5-{[benzyl(methyl)amino]methyl}-N-(2-hydroxy-2-phenylethyl)-1,2-oxazole-3-carboxamide
6-chloro-N,N-dimethyl-3-{[3-(pyridin-3-ylmethoxy)piperidin-1-yl]methyl}imidazo[1,2-a]pyridine-2-carboxamide
2-(3-methoxypropyl)-9-[4-methyl-2-(methylamino)-1,3-thiazole-5-carbonyl]-2,9-diazaspiro[5.5]undecan-3-one
N-[3-(1H-1,2,3-benzotriazol-1-yl)propyl]-2-(2-methyl-1,3-thiazol-4-yl)acetamide
1-[(2R,3R,6R)-3-(3,5-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-3-(methylsulfanyl)propan-1-one
N-(butan-2-yl)-N-[(2-chlorophenyl)methyl]-4-oxo-4H-pyrido[1,2-a]pyrimidine-3-carboxamide
(4aR,7aS)-1-(pyridin-2-ylmethyl)-4-(pyrrolidine-1-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-{[4-(but-2-yn-1-yloxy)phenyl]methyl}-2-(3-oxo-2,3-dihydro-1H-isoindol-1-yl)-N-(pyridin-3-ylmethyl)acetamide
7-[2-(4-phenyl-1,3-thiazol-2-yl)ethyl]-2-oxa-7-azaspiro[4.5]decan-8-one
N-(2-{4-methyl-5H,6H,7H-cyclopenta[d]pyrimidin-2-yl}ethyl)-3-(piperidin-3-yl)benzamide
2-(5-methylpyrazine-2-carbonyl)-7-(2-phenylethyl)-2,7-diazaspiro[4.5]decane
2-{3-cyclopropyl-5-[3-(2-oxopyrrolidin-1-yl)propyl]-1H-1,2,4-triazol-1-yl}acetic acid
N-[3-(4-{[2-(3,5-dimethyl-1H-pyrazol-1-yl)propanamido]methyl}-5-methyl-1,3-oxazol-2-yl)phenyl]-2,5-dimethylfuran-3-carboxamide
3-(2-cyclohexyl-1H-imidazol-1-yl)benzamide
({3-methanesulfonylpyrazolo[1,5-a]pyrimidin-6-yl}methyl)(methyl)[(5-propyl-1H-pyrazol-3-yl)methyl]amine
N-[2-methyl-2-(1,2,3,4-tetrahydroisoquinolin-2-yl)propyl]pyrimidin-2-amine
N-(2-{1-[(2,2-difluoro-2H-1,3-benzodioxol-5-yl)methyl]piperidin-2-yl}ethyl)acetamide
2-[(2E)-but-2-en-1-yl]-5-{2-phenyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl}-1,3,4-oxadiazole
N-{2-[2-(trifluoromethyl)phenyl]ethyl}-[1,2,3,4]tetrazolo[1,5-a]pyridine-6-carboxamide
4-({methyl[(5-{[(2-methylphenyl)methyl]sulfanyl}-4-(oxolan-2-ylmethyl)-4H-1,2,4-triazol-3-yl)methyl]amino}methyl)phenol
1-[(2-fluorophenyl)methyl]-N-[2-(4-methoxyphenyl)ethyl]-1H-1,2,3-triazole-4-carboxamide
1-{[1-(2-methoxyethyl)pyrrolidin-3-yl]methyl}-5-(3-methyl-1H-pyrazol-5-yl)-4-phenyl-1H-imidazole
benzyl(methyl){[1-(3-methylbutyl)-2-(propane-2-sulfonyl)-1H-imidazol-5-yl]methyl}amine
2-({2-[(5-chloropyridin-2-yl)oxy]hex-5-en-1-yl}(methyl)amino)-N,N-dimethylacetamide
4-(5-cyclopropyl-1,2,4-oxadiazol-3-yl)-N-[(1-methylpyrrolidin-3-yl)methyl]benzamide
N-[(5-cyclobutyl-1,2,4-oxadiazol-3-yl)methyl]-N,2-dimethylthieno[3,2-d]pyrimidin-4-amine
N-methyl-1-{[4-(methylsulfanyl)phenyl]methyl}-N-[2-(pyridin-2-yl)ethyl]piperidin-3-amine
1-[(4-fluorophenyl)methyl]-4-(oxolane-3-carbonyl)-1,4-diazepane
1-[3-(pyridin-2-yl)azetidin-1-yl]-2-[4-(1H-1,2,3,4-tetrazol-1-yl)phenyl]ethan-1-one
1-[4-(2,5-dimethoxyphenyl)pyrimidin-2-yl]-N-[3-(dimethylamino)-2,2-dimethylpropyl]-5-methyl-1H-pyrazole-4-carboxamide
(4aR,7aS)-N,N-dimethyl-4-(4-methyl-1,3-thiazole-5-carbonyl)-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide
1-[1-(methoxymethyl)cyclobutanecarbonyl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
3-(2-{2-[5-(propan-2-yl)-1,2-oxazol-3-yl]pyrrolidin-1-yl}ethyl)-2,3-dihydro-1,3-benzoxazol-2-one
5-methyl-N-[(2-{methyl[2-(pyridin-2-yl)ethyl]amino}pyridin-3-yl)methyl]pyrazine-2-carboxamide
2-[(3-ethyl-1H-1,2,4-triazol-5-yl)sulfanyl]-N-(2-methanesulfonamidoethyl)acetamide