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(2R,6S)-4-({3-[(2-chlorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-2,6-dimethylmorpholine
6-{1-[(3-chloropyridin-4-yl)methyl]piperidin-4-yl}-2-methylpyrimidin-4-ol
(1-{[2-(difluoromethoxy)phenyl]methyl}-4-[(4-methoxyphenyl)methyl]piperidin-4-yl)methanol
N,6-dimethyl-N-[(5-phenyl-1H-pyrazol-4-yl)methyl]pyrazolo[1,5-a]pyrimidine-3-carboxamide
6-(5-methoxypyridin-3-yl)quinazolin-4-amine
4-(5-{1-[(2-methoxy-4,6-dimethylpyridin-3-yl)methyl]-1H-1,2,3-triazol-4-yl}pyrimidin-2-yl)morpholine
1-{[1-butyl-2-(4-methylpentanesulfonyl)-1H-imidazol-5-yl]methyl}-3-(methoxymethyl)piperidine
(2R)-1-[(5,6,7-trimethoxy-2-oxo-1,2-dihydroquinolin-3-yl)methyl]pyrrolidine-2-carboxamide
1-[4-(6-hydroxy-1,4-oxazepane-4-carbonyl)piperidin-1-yl]-2-phenylethan-1-one
3-[3-(2-ethylphenoxy)azetidine-1-carbonyl]pyridine
3-{[(4-sulfamoylphenyl)methyl]amino}-N-(1,3-thiazol-2-yl)propanamide
methyl({[5-(oxan-2-yl)thiophen-2-yl]methyl})(4,5,6,7-tetrahydro-1H-indazol-3-ylmethyl)amine
methyl 3-{[2-(2-chloro-6-fluorophenyl)acetamido]methyl}-5-(furan-2-amido)benzoate
N,N-dimethyl-3-(3-methylpiperidin-1-yl)propanamide
1-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-3-(4-methoxy-3,5-dimethylbenzoyl)piperidine
1-(cyclohexylmethyl)-N-methyl-5-{[2-(methylsulfanyl)ethyl]amino}-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
3-(2H-1,3-benzodioxole-5-carbonyl)-1-[(2-fluoro-4-methoxyphenyl)methyl]piperidine
(1S,5R)-6-(2,6-difluorobenzoyl)-3-(2,3-dihydro-1H-inden-2-yl)-3,6-diazabicyclo[3.2.2]nonane
4-{1-[4-phenyl-5-(pyridin-4-yl)-1H-imidazol-1-yl]butan-2-yl}morpholine
(3S,4S)-3,4-bis(hydroxymethyl)-N-(5-methoxy-2-methylphenyl)pyrrolidine-1-carboxamide
1-[4-(4-{[(1-benzothiophen-2-ylmethyl)(methyl)amino]methyl}phenoxy)piperidin-1-yl]-2-(thiophen-3-yl)ethan-1-one
4-(4-cyclopropyl-1H-1,2,3-triazol-1-yl)-1-(5-methylhexan-2-yl)piperidine
3,5-difluoro-N-({1-[2-(4-methoxyphenyl)ethyl]piperidin-3-yl}methyl)-N-methylbenzamide
2-[(1-methyl-1H-indol-3-yl)sulfanyl]-1-[2-(propan-2-yl)-2,5-dihydro-1H-pyrrol-1-yl]ethan-1-one
(1S,5R)-6-(3-fluoropyridine-4-carbonyl)-3-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
4-[(4-butyl-1H-1,2,3-triazol-1-yl)methyl]-1-(dimethyl-1,3-thiazole-5-carbonyl)piperidine
7-(1-methylpiperidine-3-carbonyl)-2-(pyridin-2-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
(2S)-1-{2-[(2H-1,3-benzodioxol-5-yloxy)methyl]-1,3-oxazole-4-carbonyl}-N-ethylpyrrolidine-2-carboxamide
N-(2-ethoxyethyl)-4-(trimethyl-1H-pyrazol-4-yl)pyrimidin-2-amine
1-(2-{methyl[(2E)-3-phenylprop-2-en-1-yl]amino}pyrimidin-4-yl)pyrrolidin-3-ol
N-[2-(5-cyclopropyl-1,2,4-oxadiazol-3-yl)ethyl]-N,2-dimethyl-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
N-(1,1-dioxo-2,3-dihydro-1λ6-thiophen-3-yl)-2,5-dimethyl-1-phenyl-1H-pyrrole-3-carboxamide
1-(5-{[(3S,4S)-3-hydroxy-4-(naphthalen-2-yl)piperidin-1-yl]methyl}-1-methyl-1H-pyrrol-3-yl)ethan-1-one
N-methyl-N-(quinolin-2-ylmethyl)-5-[(4H-1,2,4-triazol-3-ylsulfanyl)methyl]furan-2-carboxamide
1-(2,2-dimethylbutanoyl)-4'-[2-(pyrrolidin-1-yl)ethyl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
2-[(5-amino-1,3,4-thiadiazol-2-yl)sulfanyl]-N-[4-(pyridin-2-yl)butyl]acetamide
N-(5-methyl-1,2-oxazol-3-yl)-N'-(3-phenylprop-2-yn-1-yl)-N'-propylethanediamide
N-[(5-fluoro-1H-indol-2-yl)methyl]-N-methyl-2-({6-[4-(pyridin-2-yl)piperazin-1-yl]pyridazin-3-yl}oxy)acetamide
N-[(3-methyl-1,2-oxazol-5-yl)methyl]-1-[1-(pyridin-3-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
1-[4-cyclohexyl-3-oxo-6-(pyridin-3-ylmethoxy)-1,4-diazepan-1-yl]-4-(4-fluorophenyl)butane-1,4-dione
1-methyl-4-[(3-phenoxyphenyl)methyl]-1,4,9-triazaspiro[5.6]dodecan-10-one
4-[4-(4-ethylpiperazine-1-carbonyl)piperidin-1-yl]-2-[2-(2-fluorophenyl)ethyl]-2,3-dihydro-1H-isoindole-1,3-dione
N-(3-cyclopentylpropyl)-6-oxo-1-(3-phenylpropyl)piperidine-3-carboxamide
6-methyl-2-{[3-(2-methylpiperidin-1-yl)azetidin-1-yl]methyl}quinolin-4-ol
5-[1-ethyl-3-(2-methylpropyl)-1H-pyrazol-5-yl]-3-(propan-2-yl)-1,2,4-oxadiazole
4-(1H-1,3-benzodiazol-1-yl)-1-(pyrimidin-2-yl)piperidine-4-carboxylic acid
2-{1-[(4-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-[(5-methylthiophen-2-yl)methyl]acetamide
N-[(6-chloro-1H-1,3-benzodiazol-2-yl)methyl]-2,5-dimethylpyrazolo[1,5-a]pyrimidin-7-amine
N-[2-(4-ethoxyphenyl)phenyl]cyclopropanecarboxamide
2-(dimethylamino)-4-methyl-N-{1-[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]ethyl}pyrimidine-5-carboxamide