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3-{2-[4-(morpholin-4-yl)piperidin-1-yl]-2-oxoethyl}-4-(2-phenylethyl)piperazin-2-one
N-methyl-N-[(1-methylpiperidin-2-yl)methyl]-2-[(prop-2-en-1-yl)amino]benzamide
1-(7-methanesulfonyl-4-methylquinazolin-2-yl)-N-(2-methylpropyl)piperidine-4-carboxamide
(1S,9R)-11-[3-amino-6-(2-methylphenyl)pyrazin-2-yl]-7,11-diazatricyclo[7.3.1.02,7]trideca-2,4-dien-6-one
{4-[(4-chlorophenyl)methyl]-1-{[4-(methylsulfanyl)phenyl]methyl}piperidin-4-yl}methanol
1-(morpholin-4-yl)-3-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propan-1-one
N-[2-(furan-2-yl)ethyl]-2,5-dimethylpyrazolo[1,5-a]pyrimidin-7-amine
5-[(3-methoxyphenyl)methyl]-3-(3-methylbut-2-en-1-yl)-5-(piperidin-4-yl)imidazolidine-2,4-dione
(2-{4-[(3-fluorophenyl)methyl]piperazin-1-yl}quinolin-3-yl)methanol
1-[(2-butyl-1H-imidazol-4-yl)methyl]-4-(5-chloropyridin-2-yl)piperazine
N-({2-[2-(3-fluorobenzenesulfonamido)phenyl]-5-methyl-1,3-oxazol-4-yl}methyl)-2-methylbutanamide
3-[(3S,7S,8aS)-3-methyl-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(3-chlorophenyl)urea
3-[2-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)ethyl]-1-[2-methyl-5-(5-methyl-1,3,4-oxadiazol-2-yl)phenyl]urea
N-[2-(1-methylpiperidin-2-yl)ethyl]-6-[(2-methylprop-2-en-1-yl)amino]pyridine-3-carboxamide
6-[3-(methoxymethyl)piperidin-1-yl]-N-(thiophen-2-ylmethyl)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-amine
N-({1-[4-(1H-imidazol-1-yl)butanoyl]piperidin-4-yl}methyl)acetamide
N-[4-({[1-(furan-2-yl)ethyl]carbamoyl}methyl)phenyl]butanamide
N-(3-chloro-4-methoxyphenyl)-6-{[2-(trifluoromethyl)phenyl]methyl}-6-azaspiro[2.5]octane-1-carboxamide
5-{[2-(2-cyclohexyl-1H-imidazol-1-yl)ethyl]sulfanyl}-1-methyl-1H-1,2,3,4-tetrazole
[2-(2-chlorophenyl)ethyl]({[6-(thiophen-3-yl)-2H-[1,3]dioxolo[4,5-g]quinolin-7-yl]methyl})amine
(1S,5R)-6-[(1-ethyl-1H-indol-6-yl)methyl]-3-(pyridin-3-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
1-cyclohexyl-3-(oxolan-3-yl)-5-(1H-pyrazol-4-yl)-1H-1,2,4-triazole
N-[1-phenyl-2-(1H-pyrazol-1-yl)ethyl]-4-sulfamoylbenzamide
5-{1-[(2-ethoxyphenyl)methyl]piperidin-4-yl}-3-(oxolan-2-ylmethyl)-5-(pyridin-2-yl)imidazolidine-2,4-dione
9-[(2S)-2-aminobutanoyl]-1,4,9-triazaspiro[5.5]undecan-5-one
ethyl 2-[(2-{[(1S,6R)-6-carbamoylcyclohex-3-en-1-yl]carbamoyl}phenyl)amino]acetate
2-methyl-N-[2-(3-{[methyl(quinolin-8-ylmethyl)amino]methyl}phenoxy)ethyl]-1,3-thiazole-4-carboxamide
3-cyano-5-fluoro-N-[1-methyl-4-(propan-2-yloxy)-1H-indazol-3-yl]benzamide
8-(5-fluoropyrimidin-2-yl)-2-propyl-2,8-diazaspiro[4.5]decane-3-carboxylic acid
N-{[5-(benzylsulfanyl)-4-(4-methoxyphenyl)-4H-1,2,4-triazol-3-yl]methyl}-5-(methoxymethyl)furan-2-carboxamide
2-[methyl(pyridin-4-ylmethyl)amino]-1-[4-(naphthalen-2-yl)piperazin-1-yl]ethan-1-one
2-{5-[3-(propan-2-yl)-1-(pyridin-2-yl)-1H-1,2,4-triazol-5-yl]-1H-pyrazol-3-yl}phenol
3-methyl-1-(1-{6-[methyl(propyl)amino]pyridine-3-carbonyl}piperidin-3-yl)butan-1-one
N-[(2,2-dimethyl-2,3-dihydro-1-benzofuran-5-yl)methyl]-5-(morpholin-4-ylmethyl)furan-3-carboxamide
6-ethyl-N-[3-(1H-imidazol-1-yl)propyl]-1,5-dimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
N-(2-{[(2-methylphenyl)methyl]sulfanyl}ethyl)-2-(trimethyl-1H-pyrazol-1-yl)acetamide
4-[(3-chloro-5-fluorophenyl)methyl]-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
N-[(5-methylpyrazin-2-yl)methyl]-5-(oxolan-2-yl)thiophene-2-carboxamide
(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-5-[1-(propan-2-yl)piperidin-4-yl]-1,5-diazatricyclo[5.2.2.02,6]undecane
1-{4-[(2-methoxyethyl)amino]-2-(pyridin-2-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl}ethan-1-one
4-(6-methoxypyridin-2-yl)-2-({methyl[(3-methyl-1,2-oxazol-5-yl)methyl]amino}methyl)phenol
(1S,5R)-6-[(dimethyl-1,2-oxazol-4-yl)methyl]-3-[(1s,4s)-4-hydroxycyclohexanecarbonyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
N-ethyl-3-(4-methyl-1,3-thiazol-5-yl)-N-(pyridin-4-ylmethyl)propanamide
N-[(3R,4S)-4-cyclopropyl-1-(pyridin-4-ylmethyl)pyrrolidin-3-yl]-3-(methylsulfanyl)propanamide
2,3,5,6-tetramethyl-N-{2-[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]ethyl}benzamide
3-[(3R,4S)-1-[(2,3-dichlorophenyl)methyl]-4-(dimethylamino)piperidin-3-yl]propan-1-ol
(1S,5R)-6-(3-methylthiophene-2-carbonyl)-3-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
(4aS,7aR)-1-(1-methyl-1H-imidazole-5-carbonyl)-4-propanoyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-{[(2S)-2-amino-2-cyclohexylacetamido]methyl}-N,N-dimethyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carboxamide
1-{7-[(2-fluorophenyl)methyl]-2,7-diazaspiro[4.5]decan-2-yl}-2-methoxyethan-1-one