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6-(morpholin-4-yl)-N4-[1-(oxolan-2-ylmethyl)piperidin-4-yl]pyrimidine-2,4-diamine
2-(1-{1-[1-(3,5-dimethyl-1H-pyrazol-4-yl)propan-2-yl]piperidin-4-yl}-1H-1,2,3-triazol-4-yl)pyridine
2-(2-{[4-(pyridin-3-ylmethyl)piperazin-1-yl]methyl}phenoxy)propanoic acid
ethyl 4-({2-phenyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl}amino)piperidine-1-carboxylate
3-({[5-(2-fluorophenyl)pyrazolo[1,5-a]pyrimidin-7-yl]amino}methyl)-1λ6-thiolane-1,1-dione
4-ethyl-3-({1-[(1-ethylpiperidin-3-yl)methyl]piperidin-4-yl}methyl)-1-methyl-4,5-dihydro-1H-1,2,4-triazol-5-one
N-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]-1-(2-methoxyphenyl)-1H-pyrazole-4-carboxamide
2-methyl-N-{[7-(3-phenylpropyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]methyl}butanamide
N-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-2-(1-methyl-1H-indol-3-yl)acetamide
1-(1H-imidazol-4-ylmethyl)-4-[3-(propan-2-yl)-1H-pyrazol-5-yl]piperidine
2-[3-(3-fluorophenyl)-1H-pyrazol-1-yl]-N-[3-methyl-1-(pyridin-2-yl)-1H-pyrazol-5-yl]acetamide
2-{[2-(azepan-1-yl)propanamido]methyl}-N,N-dimethyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carboxamide
1-cyclohexyl-3-{1-[2-(4-methoxyphenyl)ethyl]-5-oxopyrrolidin-3-yl}urea
4-(2,4-dioxoimidazolidin-1-yl)-N-{[2-(1H-pyrazol-1-yl)phenyl]methyl}benzamide
(1R,7S)-N-methyl-N-[(2-methyl-1,3-thiazol-4-yl)methyl]-4-oxo-3-(pyridin-3-ylmethyl)-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
N-cyclopentyl-4-fluoro-N-{[4-methoxy-3-(thiophen-2-ylmethoxy)phenyl]methyl}benzamide
(3S,4S)-1-(3-phenylpropyl)-4-[4-(pyridin-2-yl)piperazin-1-yl]pyrrolidin-3-ol
(2E)-3-(3-fluorophenyl)-1-{4-[2-(methoxymethyl)-5-(trifluoromethyl)-1H-1,3-benzodiazol-1-yl]piperidin-1-yl}prop-2-en-1-one
N-cyclopropyl-3-{4-[2-(5-methylfuran-2-yl)-1H-imidazol-1-yl]phenyl}propanamide
6-{4-[4-(pyridin-3-yl)-1H-1,2,3-triazol-1-yl]piperidin-1-yl}-9H-purin-2-amine
methyl 5-[3-(4-methoxybenzenesulfonamidomethyl)piperidin-1-yl]-5-oxopentanoate
3-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1-[4-(pyridin-4-yl)-1,4-diazepan-1-yl]propan-1-one
6-methyl-5-[2-methyl-4-(2-methylphenyl)piperazine-1-carbonyl]-2-oxo-1,2-dihydropyridine-3-carbonitrile
1-cyclopropyl-N-[2-(1-methyl-1H-1,3-benzodiazol-2-yl)ethyl]-5-oxopyrrolidine-3-carboxamide
1-methyl-N-[(2S)-oxolan-2-ylmethyl]-6-propyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
2-[4-({[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}amino)piperidin-1-yl]pyridine-3-carbonitrile
(2R,3S,6R)-5-(1-ethyl-1H-pyrazole-4-carbonyl)-3-(3-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
N-{1-[1-(9H-fluoren-2-ylmethyl)piperidin-4-yl]-1H-pyrazol-5-yl}-3-methylbutanamide
1-benzyl-N3-ethyl-N5-[(4-methoxyphenyl)methyl]-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
2-[1-(cyclohexylmethyl)-4-[(2-ethyl-4-methyl-1H-imidazol-5-yl)methyl]piperazin-2-yl]ethan-1-ol
3-{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}-3-methyl-1-(2-oxo-2,3-dihydro-1H-indol-5-yl)urea
N-(1-carbamoylcyclopentyl)-4-(1H-pyrazol-3-yl)benzamide
2-{1-[(3,5-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-(2-hydroxyethyl)acetamide
2-{1-cyclopentyl-4-[(6-fluoro-1H-1,3-benzodiazol-2-yl)methyl]piperazin-2-yl}ethan-1-ol
N-[4-(methylsulfanyl)phenyl]-6-[(2-phenyl-1,3-thiazol-5-yl)methyl]-6-azaspiro[2.5]octane-1-carboxamide
2-(1-cyclopentyl-4-{[3-(furan-2-yl)phenyl]methyl}piperazin-2-yl)ethan-1-ol
N-[1-(4-chlorophenyl)-5-oxopyrrolidin-3-yl]-2-[5-(pyrrolidin-1-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]acetamide
N-{[2-(dimethylamino)-5,6,7-trimethoxyquinolin-3-yl]methyl}-N-[2-(4-fluorophenyl)ethyl]imidazo[1,2-a]pyridine-2-carboxamide
1-[(4-fluorophenyl)methyl]-2-(propan-2-yl)-4-[2-(1H-pyrazol-4-yl)ethyl]-1,4-diazepane
1-{4-[4-chloro-2-(1,2-oxazolidine-2-carbonyl)phenoxy]piperidin-1-yl}ethan-1-one
(3S,4R)-1-(3-fluoropyridin-2-yl)-4-(4-methoxyphenyl)-N,N-dimethylpyrrolidin-3-amine
1-methyl-4-[4-(2-methylpyridin-4-yl)-1,4-diazepane-1-carbonyl]imidazolidin-2-one
(3aR,6aR)-2-(morpholine-4-sulfonyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-(3-methoxyphenyl)-3-[2-(methylamino)acetamido]benzamide
N-{[1-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)piperidin-3-yl]methyl}furan-2-carboxamide
5-{4-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidine-1-carbonyl}-2,4-dimethylpyridine
1-(carbamoylmethyl)-N-[(4-methoxyphenyl)methyl]-N-(oxolan-2-ylmethyl)piperidine-4-carboxamide
2-cyclopropyl-6-{4-[1-(morpholin-4-yl)ethyl]phenyl}quinoline-4-carboxylic acid
2-(1-{1-[(2-fluorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}piperidin-3-yl)-1H-1,3-benzodiazole
N-[(3-methoxyphenyl)methyl]-4-{[1-(pyridin-2-ylmethyl)piperidin-4-yl]oxy}benzamide