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6-{3-[4-(2-methoxybenzoyl)piperazin-1-yl]-3-oxopropyl}-2,3-dihydropyridazin-3-one
2-(3-{2-[2-(2-oxopyrrolidin-1-yl)ethyl]piperidine-1-carbonyl}phenoxy)acetamide
4-{[(2-methoxyethyl)(1-methylpiperidin-4-yl)amino]methyl}-2,6-dimethylphenyl acetate
4,4,4-trifluoro-1-[(1S,5R)-3-(pyrazine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]butan-1-one
(3aR,6aR)-2-(cyclobutylmethyl)-5-(3,4-dimethylbenzoyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
(4aR,7aS)-1-cyclobutanecarbonyl-4-(4-methyl-1H-imidazole-5-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-[(3S,4R)-1-[(4-chlorophenyl)methyl]-4-(morpholin-4-yl)piperidin-3-yl]-N-(cyclopropylmethyl)-N-propylpropanamide
5-{1-[2-(4-methoxyphenyl)ethyl]-1H-pyrazol-3-yl}-4-methyl-N-[(5-methylfuran-2-yl)methyl]-1,3-thiazol-2-amine
1-methyl-4-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]-2,3,4,5-tetrahydro-1H-1,4-benzodiazepine-2,5-dione
1-(3-{[3-(2-hydroxyethyl)-4-[(2-methylphenyl)methyl]piperazin-1-yl]methyl}phenyl)ethan-1-one
N,1-dimethyl-N-[(3-phenyl-1H-pyrazol-5-yl)methyl]-6-propyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
8-(5-chloro-2-hydroxybenzoyl)-2-(cyclopropylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
4-[2-(2,3-difluorophenyl)acetyl]-1-(1H-indazol-5-yl)piperazin-2-one
2-({4-[(4-fluorophenyl)methyl]-3-(2-hydroxyethyl)piperazin-1-yl}methyl)-3-methoxyphenol
2-(2-fluorophenyl)-1-[(1R,5R)-6-propyl-3,6-diazabicyclo[3.2.2]nonan-3-yl]ethan-1-one
1-ethyl-N-(furan-2-ylmethyl)-N-methyl-5-(pyrrolidin-1-yl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
3-methyl-7-{[2-(thiophen-2-yl)pyrimidin-5-yl]methyl}-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
3-(3-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidine-1-carbonyl)phenol
N,N-dimethyl-6-(quinolin-3-yl)pyrazine-2-carboxamide
N-(2H-1,3-benzodioxol-5-yl)-1-(pyridin-3-ylmethyl)piperidin-3-amine
5-[methyl({[2-(methylamino)pyrimidin-5-yl]methyl})amino]-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxylic acid
4,6-dimethyl-N-{[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]methyl}-2-oxo-1,2,3,4-tetrahydropyrimidine-5-carboxamide
1'-(3-fluoro-4-methylbenzoyl)-5-propyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
7-(3-chlorophenyl)-9-[(1-methylpiperidin-3-yl)methoxy]-4-(pyridin-2-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
4-{4-[3-(3,5-dimethyl-1H-pyrazol-1-yl)azetidin-1-yl]piperidin-1-yl}-6-methyl-2-propylpyrimidine
2-(benzyloxy)-1-{5-hydroxy-1-oxa-9-azaspiro[5.5]undecan-9-yl}ethan-1-one
3-[2-(4-cyclopentylpiperazin-1-yl)-2-oxoethyl]-4-[(3-fluorophenyl)methyl]piperazin-2-one
1-(5-methyl-3-phenyl-1,2-oxazole-4-carbonyl)-3-{[4-(pyrrolidine-1-carbonyl)-1H-1,2,3-triazol-1-yl]methyl}piperidine
5-{3-[2-(hydroxymethyl)piperidin-1-yl]-3-oxopropyl}-5-[(3-methoxyphenyl)methyl]pyrrolidin-2-one
8-[(2-hydroxyphenyl)methyl]-1-(2-phenylethyl)-3-(pyridin-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-benzyl-4-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]-1,4-diazepan-6-ol
6-{[3-(4H-1,2,4-triazol-4-yl)propyl]amino}-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3(8),6,12,14-pentaen-4-one
5-{4-[4-(3-fluorophenyl)-1H-pyrazol-5-yl]piperidine-1-carbonyl}-1H-indole
3-{[(3-ethoxy-2-hydroxypropyl)amino]methyl}-N,8-dimethyl-N-(2-phenylethyl)imidazo[1,2-a]pyridine-2-carboxamide
1-{5-[3-(3-fluoro-4-phenylbenzoyl)piperidine-1-carbonyl]-1H-pyrazol-3-yl}ethan-1-one
N-{[1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl}-1-(pyridin-2-yl)-4,5,6,7-tetrahydro-1H-indazol-4-amine
(3R,5S)-N-butyl-5-[(pyridin-3-yloxy)methyl]piperidine-3-carboxamide
[1-(1H-indazole-3-carbonyl)piperidin-4-yl](1-methyl-1H-imidazol-2-yl)methanol
2-[2,6-dimethyl-4-(piperidin-1-ylmethyl)phenoxy]-3-methoxypyrazine
N-benzyl-4-[1-(4-fluorophenyl)-1H-pyrazol-4-yl]pyrimidin-2-amine
3-{1-methyl-1H-pyrrolo[2,3-b]pyridin-4-yl}-6-(pyrrolidin-1-yl)pyridazine
5-{2-methoxy-4-[(2-methyl-3-oxopiperazin-1-yl)methyl]phenoxymethyl}furan-2-carboxylic acid
N,N-dimethyl-2-[(1S,5R)-7-oxo-3-[3-(pyridin-4-yl)propanoyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]acetamide
N-{[2-(1H-imidazol-1-yl)pyridin-3-yl]methyl}-3-methyl-1-propyl-1H-pyrazole-4-carboxamide
5-{[2,5-dimethyl-1-(4H-1,2,4-triazol-4-yl)-1H-pyrrol-3-yl]methyl}-10-methoxy-3,4,5,6-tetrahydro-2H-1,5-benzoxazocine
4-hydroxy-N-[3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)phenyl]-4-(pyridin-3-yl)piperidine-1-carboxamide
N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)pyrrolidin-3-yl]methyl}-4-(1H-pyrazol-4-yl)butanamide
1-{4-[3-(2-chlorophenyl)pyrrolidin-1-yl]piperidin-1-yl}ethan-1-one
N-(2-hydroxyethyl)-3-[5-(3-methylbutanoyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]propanamide
2-({1-[4-(methylsulfanyl)phenyl]-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl}methyl)-1H-imidazole