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N-methyl-N,1-bis(2-methylpropyl)-3-(morpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
N-methyl-3-(4-methyl-1,2,3,6-tetrahydropyridine-1-carbonyl)-N-(1,2-oxazol-3-ylmethyl)benzene-1-sulfonamide
2-{2-[2-(2,1,3-benzoxadiazol-4-yl)-1H-imidazol-1-yl]phenyl}ethan-1-ol
3-{2-[(3R,4R)-3-cyclobutyl-3-hydroxy-4-methylpyrrolidin-1-yl]-2-oxoethyl}imidazolidine-2,4-dione
N-[2-(5-methyl-1,3,4-thiadiazol-2-yl)ethyl]-1-(propan-2-yl)piperidine-4-carboxamide
2-(dimethylamino)-N-[3-(2-oxopyrrolidin-1-yl)propyl]pyridine-3-carboxamide
3-hydroxy-3-(hydroxymethyl)-N-{3-[(2-methylprop-2-en-1-yl)oxy]phenyl}pyrrolidine-1-carboxamide
(3aR,6aS)-5-{[3-(ethoxymethyl)-4-methoxyphenyl]methyl}-2-methyl-octahydropyrrolo[3,4-c]pyrrole-1,3-dione
N-[(4-fluorophenyl)methyl]-N-(3-hydroxypropyl)-2,3-dihydro-1H-indene-1-carboxamide
N-[2-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-5-(propan-2-yl)-1,2-oxazole-3-carboxamide
2-{3-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-1,3-benzoxazole
1-[4-(3-methylphenoxy)piperidin-1-yl]-2-(methylsulfanyl)ethan-1-one
6-{4-[4-ethyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyrimidin-4-amine
1-{1-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]azetidin-3-yl}-2-methylpiperidine
N-[(4-methanesulfonylmorpholin-2-yl)methyl]-3-(trimethyl-1H-pyrazol-4-yl)propanamide
4-methanesulfonyl-N-[3-(1H-1,2,4-triazol-1-yl)phenyl]piperazine-1-carboxamide
ethyl 4-[1-(4-methyl-2-oxopentanoyl)piperidin-3-yl]piperazine-1-carboxylate
N-(hexahydro-1H-pyrrolizin-7a-ylmethyl)-2,6-dimethylquinoline-4-carboxamide
3-[(3R,7S,8aS)-3-[(4-hydroxyphenyl)methyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(4-fluorophenyl)urea
{[2-(azepane-1-carbonyl)-7-methylimidazo[1,2-a]pyridin-3-yl]methyl}[(1R)-1-(4-methoxyphenyl)ethyl]amine
1-(2H-1,3-benzodioxol-4-ylmethyl)-N-[3-(furan-2-yl)phenyl]piperidine-4-carboxamide
(1S,5R)-3-[(4-methoxyphenyl)methyl]-6-{[3-(propan-2-yl)-1,2-oxazol-5-yl]methyl}-3,6-diazabicyclo[3.2.2]nonane
N-[2-(2,3-dimethoxyphenyl)ethyl]-5-(3,4-dimethylphenoxymethyl)-1,2-oxazole-3-carboxamide
2-(5-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)-N-[2-(pyridin-3-yl)-5,6,7,8-tetrahydroquinazolin-5-yl]acetamide
2-methyl-1-(propan-2-yl)-4-[(1-propyl-1H-imidazol-2-yl)methyl]piperazine
2-(3-amino-1H-indazol-5-yl)-6-methoxy-N,N-bis(propan-2-yl)benzamide
2-methyl-9-[3-(5-methylfuran-2-yl)benzoyl]-2,9-diazaspiro[5.5]undecan-3-one
2-[(4-methoxypyridin-2-yl)methyl]-5-(morpholin-4-yl)-2,3-dihydropyridazin-3-one
6-methoxy-3-(1,2,3,4-tetrahydroisoquinolin-5-yl)quinoline
N-(1-methylpiperidin-4-yl)-2-[1-(propan-2-yl)-1H-pyrazol-4-yl]quinoline-4-carboxamide
methyl 3-[(2,3-dihydro-1-benzofuran-2-ylformamido)methyl]-5-(1,3-dimethyl-1H-pyrazole-5-amido)benzoate
1-{1-[(4-chlorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}-2-(2-phenylethyl)piperidine
2-amino-6-(7-methoxy-1-benzofuran-2-yl)-4-(pyridin-4-yl)pyridine-3-carbonitrile
(4aR,8aR)-2-[(6-chloro-2-fluoro-3-methylphenyl)methyl]-7-cyclobutanecarbonyl-decahydro-2,7-naphthyridin-4a-ol
3-[1-(2-chloro-6-methylbenzenesulfonyl)azetidin-3-yl]pyridine
(4aS,8aR)-1-(piperidin-4-ylmethyl)-6-(pyridin-2-ylmethyl)-decahydro-1,6-naphthyridin-2-one
4,6-dimethyl-5-{3-[3-(4-methylpiperazin-1-yl)-3-oxopropyl]piperidine-1-carbonyl}-1,2-dihydropyridin-2-one
(3aR,6aS)-2-[(5-cyclopentylthiophen-2-yl)methyl]-octahydropyrrolo[3,4-c]pyrrole
1'-[(5-tert-butyl-1H-pyrazol-3-yl)methyl]-1,2-dihydrospiro[indole-3,3'-piperidine]-2-one
3-(4-benzyl-6-hydroxy-1,4-diazepan-1-yl)-N,N-dimethylpropane-1-sulfonamide
N-{5,7-dimethylpyrido[2,3-d]pyrimidin-4-yl}-1-propylpiperidin-4-amine
2,2-dimethyl-3-{[3-(piperidine-1-carbonyl)-1-propyl-4,5,6,7-tetrahydro-1H-indazol-5-yl]amino}propan-1-ol
2-ethyl-9-[4-(4-fluorophenyl)-4-oxobutyl]-2,9-diazaspiro[5.5]undecan-3-one
N-(dimethyl-1H-1,2,4-triazol-3-yl)-3-[(4-fluorophenyl)methyl]piperidine-1-carboxamide
1-[4-({3-[(2S)-2-(hydroxymethyl)pyrrolidine-1-carbonyl]-1,2-oxazol-5-yl}methoxy)phenyl]ethan-1-one
5-{2-[(4aS,7aR)-4-(2-methylpropyl)-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]-2-oxoethyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
N-[2-(dimethylamino)ethyl]-1-{1-[(4-methoxy-2,3-dimethylphenyl)methyl]piperidin-4-yl}-1H-1,2,3-triazole-4-carboxamide
1-[4-(2-methoxyethyl)piperazin-1-yl]-2-(4-phenylpiperidin-1-yl)ethan-1-one
3-{3-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-5-(pyrrolidin-1-yl)pyridazine
1-[1-(1,3-benzoxazol-2-yl)piperidin-4-yl]-N-cyclohexylpiperidine-3-carboxamide