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4-[(1-{[5-(2-fluorophenyl)furan-2-yl]methyl}piperidin-2-yl)methyl]morpholine
5-(azepane-1-carbonyl)-N-(2-methylpropyl)-4-oxo-1-(propan-2-yl)-1,4-dihydropyridine-3-carboxamide
6-cyclopentyl-3-({[1-(1H-imidazol-1-yl)propan-2-yl]amino}methyl)-2-methoxy-5H,6H,7H-pyrrolo[3,4-b]pyridin-5-one
N-methyl-N-[(2E)-3-phenylprop-2-en-1-yl]-3-propyl-1H-pyrazole-5-carboxamide
2-methoxy-4-[(2-phenyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)methyl]phenol
3-[(1S,5R)-3-benzyl-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-N,N-dimethylaniline
2-(2,5-dimethylphenyl)-1-[3-(1-methyl-1H-pyrazol-4-yl)propyl]-1H-imidazole
1-[3-(4-chlorophenyl)propyl]-5-oxopyrrolidine-3-carboxylic acid
3-(8-methoxy-2-methylquinolin-5-yl)-1-methyl-6-(6-methylpyridine-2-carbonyl)-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
4-cyclopentyl-7-(3,4-dimethoxyphenyl)-9-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepine
1-(4-{[(3-methyl-1,2-oxazol-5-yl)methyl]amino}-2-(pyridin-2-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl)ethan-1-one
N-cyclohexyl-7-(oxan-4-yl)-6-oxo-2,7-diazaspiro[4.5]decane-2-carboxamide
8-[1-(4-fluorophenyl)cyclopropanecarbonyl]-3-methyl-1-oxa-3,8-diazaspiro[4.5]decan-2-one
2-[3-benzyl-1-(2-methoxyphenyl)-5-oxo-4,5-dihydro-1H-1,2,4-triazol-4-yl]-N-(1-cyclopropylethyl)acetamide
ethyl[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl](1,3-thiazol-2-ylmethyl)amine
2-cyclopropanecarbonyl-8-[(3-fluorophenyl)methyl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid
3,5-dimethyl-N-[1-phenyl-3-(1H-1,2,4-triazol-1-yl)propyl]-1-benzofuran-2-carboxamide
N-methyl-N-{[3-(pyridin-4-yl)-1,2-oxazol-5-yl]methyl}pyridin-4-amine
4,4-difluoro-1-(2-methyl-1-benzofuran-5-carbonyl)piperidine
3-methyl-3-[(4-methyl-1,3-thiazol-2-yl)methyl]-1-[2-methyl-5-(2-methyl-2H-1,2,3,4-tetrazol-5-yl)phenyl]urea
3-(azepane-1-sulfonyl)-7-methoxy-2,3,4,5-tetrahydro-1H-3-benzazepine
methyl 1-[(3S,5S)-1-[(3-chlorophenyl)methyl]-5-(cycloheptylcarbamoyl)pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate
(3S,4R)-1-[(4-methylpiperazin-1-yl)sulfonyl]-4-(pyridin-4-yl)pyrrolidine-3-carboxylic acid
8-{[3-(4-methylphenyl)-1,2-oxazol-5-yl]methyl}-1-oxa-8-azaspiro[4.6]undecan-9-one
1-[2-(1H-imidazol-2-yl)benzoyl]-3-(1H-pyrazol-5-yl)piperidine
ethyl 4-[(2R,3R,6R)-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]butanoate
ethyl 3-[(3-chlorophenyl)methyl]-1-[2-(1H-imidazol-2-yl)benzoyl]piperidine-3-carboxylate
4-{1-[1-(thiophen-3-ylmethyl)piperidin-4-yl]ethyl}morpholine
2-(2-hydroxyethyl)-9-(naphthalene-2-carbonyl)-2,9-diazaspiro[5.5]undecan-3-one
1-ethyl-N-[(4-methoxyphenyl)methyl]-5-[(2-oxo-1,2-dihydroquinolin-3-yl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
2,2-dimethylpropyl 3-oxo-2-[2-(pyridin-4-yl)ethyl]-2,9-diazaspiro[5.5]undecane-9-carboxylate
N-(2-methyl-2H-1,2,3-triazol-4-yl)-2-{1H-pyrazolo[3,4-b]pyridin-1-yl}acetamide
(1H-1,3-benzodiazol-2-ylmethyl)({[2-cyclopropylmethanesulfonyl-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl})methylamine
N-ethyl-1,5-dimethyl-N-({1-[2-(2-methylphenyl)ethyl]piperidin-4-yl}methyl)-1H-pyrazole-3-carboxamide
1-({3-[1-(4-methylphenyl)cyclopentyl]-1,2,4-oxadiazol-5-yl}methyl)-3-propoxypiperidine
methyl N-{1-oxo-1-[3-oxo-2-(2-phenylethyl)-2,9-diazaspiro[5.5]undecan-9-yl]propan-2-yl}carbamate
4-[3-(2-fluorophenyl)-1H-pyrazole-5-carbonyl]-1-methyl-1,4,9-triazaspiro[5.5]undecane
3-(4-aminopyridine-2-carbonyl)-7-methyl-3,7,11-triazaspiro[5.6]dodecan-12-one
4-{8-thiatricyclo[7.4.0.02,7]trideca-1(9),2(7),3,5,10,12-hexaen-6-yl}-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
N-(1H-imidazol-2-ylmethyl)-N-methyl-5-[(quinolin-8-yloxy)methyl]-1,2-oxazole-3-carboxamide
N-[(3R,4S)-1-acetyl-4-cyclopropylpyrrolidin-3-yl]-2-(1H-1,2,3,4-tetrazol-5-yl)benzamide
1-(4-{1-[2-(dimethylamino)ethyl]-1H-imidazol-2-yl}piperidin-1-yl)-2-(morpholin-2-yl)ethan-1-one
1-{4-[(2-fluorophenyl)methyl]-1,4-diazepan-1-yl}-2-{8-methylimidazo[1,2-a]pyridin-3-yl}ethan-1-one
N-[3-(1H-imidazol-2-yl)propyl]-6-(propan-2-yl)pyrimidin-4-amine
(1R,5R)-6-(5-chlorothiophene-2-carbonyl)-N,N-dimethyl-3,6-diazabicyclo[3.2.2]nonane-3-sulfonamide
1-{[1-(2-methoxyphenyl)-3-(2-methylpropyl)-1H-1,2,4-triazol-5-yl]methyl}-5-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
1-[3-(2-methoxyphenoxy)azetidin-1-yl]-2-(pyrrolidin-1-yl)ethan-1-one
8-(1,3-benzothiazol-2-ylmethyl)-1-(3-methoxypropyl)-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-(2H-1,3-benzodioxol-5-ylmethyl)-4-(4-{[3-(1H-pyrazol-1-yl)propyl]amino}piperidin-1-yl)benzamide
3-chloro-N-{[5-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-N-methylpyridine-4-carboxamide