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1-{2-[1-(3-cyclohexylpropanoyl)piperidin-2-yl]ethyl}-N-cyclopropyl-1H-1,2,3-triazole-4-carboxamide
4-methoxy-N-{2-[7-(naphthalen-1-ylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]ethyl}benzamide
5-{1-[2-(2-methoxyphenyl)acetyl]piperidin-4-yl}-5-methyl-3-[2-(morpholin-4-yl)ethyl]imidazolidine-2,4-dione
1-(2H-1,3-benzodioxole-5-carbonyl)-3-(1-butyl-1H-imidazol-2-yl)piperidine
2-amino-4-(2-aminopyrimidin-5-yl)-6-(3-fluorophenyl)pyridine-3-carbonitrile
5-methyl-4-(1-methyl-1H-1,2,4-triazol-5-yl)-2-(3-phenylpiperidin-1-yl)pyrimidine
4-{1-[3-(cyclopentylcarbamoyl)propanoyl]piperidin-3-yl}benzoic acid
3,4-dimethyl-N-propyl-5-sulfamoyl-N-(thiophen-3-ylmethyl)benzamide
2-(4-chloro-2-{[4-(4-methyl-4H-1,2,4-triazol-3-yl)piperidin-1-yl]methyl}phenoxy)acetamide
4-{1-[1-(1-methyl-1H-pyrazole-3-carbonyl)piperidin-4-yl]piperidine-3-carbonyl}morpholine
4-{3-[(3-cyclohexylpyrrolidin-1-yl)methyl]-8-methylimidazo[1,2-a]pyridine-2-carbonyl}morpholine
1-methyl-4-({5-[2-(3-phenyl-1,2,4-oxadiazol-5-yl)ethyl]-1,2,4-oxadiazol-3-yl}methyl)piperidine
2-[(1-methanesulfonylpiperidin-4-yl)oxy]-N-(3-phenylpropyl)benzamide
1-{1-[(2-chlorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}-3-(piperidin-1-ylmethyl)piperidine
2-methyl-N-[(2-phenyl-1,3-thiazol-5-yl)methyl]-2,8-diazaspiro[4.5]decane-3-carboxamide
methyl[(3-{octahydro-1H-pyrido[1,2-a]piperazine-2-carbonyl}-1,2-oxazol-5-yl)methyl](2-phenylethyl)amine
1-{1-[3-(2-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-5-carbonyl]cyclopentyl}pyrrolidine
N-{[(3S,4S)-3-hydroxypiperidin-4-yl]methyl}-4-phenyl-1,3-thiazole-2-carboxamide
N-{2-[2-(2-fluorophenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]ethyl}furan-2-carboxamide
2-{2-[1-(2H-1,3-benzodioxol-5-yl)propan-2-yl]-1H-imidazol-1-yl}-N,N-dimethylethane-1-sulfonamide
N-cyclopentyl-N-({1-[2-(2-methylphenyl)ethyl]piperidin-4-yl}methyl)-1H-imidazole-2-carboxamide
5-ethyl-3-(2-methylprop-2-en-1-yl)-5-[1-(3-phenylpropyl)piperidin-4-yl]imidazolidine-2,4-dione
1-(7-fluoro-3-methyl-1-benzofuran-2-carbonyl)-4-(pyridin-2-yl)piperazine
N-[(3-methyl-1H-pyrazol-5-yl)methyl]-5-[1-(piperidin-1-yl)ethyl]furan-2-carboxamide
N-({3-[2-(4-fluorophenyl)ethoxy]phenyl}methyl)-N-(pyridin-4-ylmethyl)-2,3-dihydro-1-benzofuran-2-carboxamide
1-cyclohexyl-5-[1-(1H-imidazol-1-yl)ethyl]-3-(2-methoxyethyl)-1H-1,2,4-triazole
2-methoxy-3-[5-methyl-2-(4H-1,2,4-triazol-4-yl)pyridin-3-yl]quinoline
2-{[4-(5-{[(3-chlorophenyl)methyl]sulfanyl}-4-(prop-2-en-1-yl)-4H-1,2,4-triazol-3-yl)piperidin-1-yl]methyl}-6-methylpyridine
N-(3,4-dihydro-1H-2-benzopyran-1-ylmethyl)-4-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]butanamide
N-[1-(hydroxymethyl)cycloheptyl]-6-methoxy-2-oxo-1,2,3,4-tetrahydroquinoline-4-carboxamide
(1S,5R)-6-benzyl-3-({2-methylimidazo[1,2-a]pyridin-3-yl}methyl)-3,6-diazabicyclo[3.2.2]nonane
methyl 4-(4-{[2-(4-fluorophenyl)-3-oxopiperazin-1-yl]methyl}-5-methyl-1,3-oxazol-2-yl)benzoate
N-{[1-(ethoxymethyl)cyclobutyl]methyl}-5-oxo-1-(pyridin-2-ylmethyl)pyrrolidine-3-carboxamide
4-(4-chlorophenyl)-N-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]butanamide
3-(3-methoxyphenyl)-N-[2-(1H-pyrrol-1-yl)ethyl]-1H-pyrazole-5-carboxamide
3-[(2,3,5,6-tetrafluoro-4-methylphenyl)methyl]-1,3-oxazolidin-2-one
N-(diphenylmethyl)-1-ethyl-3-(pyrrolidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
2-{5-[6-amino-2-(diethylamino)pyrimidin-4-yl]-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-1-yl}ethan-1-ol
3,3,3-trifluoro-1-{5-methanesulfonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}propan-1-one
methyl (1R,5S,6R)-6-[(4-methanesulfonamidopiperidin-1-yl)methyl]-3-azabicyclo[3.1.0]hexane-3-carboxylate
2-chloro-N-(2-{[1-methyl-3-(propan-2-yl)-1H-pyrazol-5-yl]formamido}ethyl)benzamide
N-(2H-1,3-benzodioxol-5-ylmethyl)-1-(1,3-dioxo-2-{spiro[bicyclo[2.2.1]heptane-7,1'-cyclopropan]-2-en-5-ylmethyl}-2,3-dihydro-1H-isoindol-4-yl)piperidine-3-carboxamide
methyl 2-[methyl(2-methylpropyl)sulfamoyl]-6-[(3-methylphenyl)methyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
1-{5H,6H,7H,8H,9H-imidazo[1,5-a][1,4]diazepin-8-yl}-2-(2-methylphenyl)ethan-1-one
N-{1-[(3,5-difluorophenyl)methyl]piperidin-4-yl}-3-(trifluoromethyl)-1H-pyrazole-5-carboxamide
[(5-methoxy-3-methyl-1H-indol-2-yl)methyl]({[2-(morpholin-4-yl)pyridin-3-yl]methyl})amine
2-(3-methylphenyl)-5-{[4-(1H-pyrazol-1-ylmethyl)piperidin-1-yl]methyl}pyrimidine
(2H-1,3-benzodioxol-4-ylmethyl)[(3-methylthiophen-2-yl)methyl](pyridin-2-ylmethyl)amine
7-[(3,5-dichloropyridin-4-yl)methyl]-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
3-(4-methyl-1,3-thiazol-5-yl)-N-[2-(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)ethyl]propanamide