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1-(cyclobutylmethyl)-3-hydroxy-3-(1,4-oxazepan-4-ylmethyl)piperidin-2-one
N-[4-(pyridin-3-yloxy)-1-(2,2,2-trifluoroethyl)-1H-indazol-3-yl]-1H-pyrazole-3-carboxamide
5-[3-(2,5-dimethoxyphenyl)pyrrolidine-1-carbonyl]-1H-imidazole-4-carboxylic acid
1-[(2E)-3-phenylprop-2-en-1-yl]-4-[4-(thiophen-3-yl)-1H-1,2,3-triazol-1-yl]piperidine
methyl 2-{1-[6-(2-fluorophenyl)imidazo[2,1-b][1,3]thiazole-3-carbonyl]-3-oxopiperazin-2-yl}acetate
N-[1-(4-propyl-4H-1,2,4-triazol-3-yl)ethyl]-1-[(1s,4s)-4-aminocyclohexyl]-1H-1,2,3-triazole-4-carboxamide
6-ethyl-1-methyl-N-[(1S)-1-(3-methylpyridin-2-yl)ethyl]-1H-pyrazolo[3,4-d]pyrimidin-4-amine
N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-5-oxo-1-phenyl-2,5-dihydro-1H-pyrazole-3-carboxamide
N-(2-hydroxy-2-phenylethyl)-N-(pyridin-4-ylmethyl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
5-[4-(1-ethyl-6-oxopiperidine-3-carbonyl)piperazin-1-yl]-2-methyl-2,3-dihydropyridazin-3-one
5-cyclopropanecarbonyl-1'-(3-methoxybenzoyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
5-[3-(2-methoxyethyl)-1-(4-methoxyphenyl)-1H-1,2,4-triazol-5-yl]-2-(4H-1,2,4-triazol-4-yl)pyridine
N-{[1-(3-chlorophenyl)pyrrolidin-3-yl]methyl}-1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carboxamide
3-(4-fluorophenyl)-1-{4-[(1-methyl-1H-imidazol-2-yl)methyl]piperazin-1-yl}propan-1-one
N-[(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)methyl]-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
ethyl 1-(7-oxo-1-propylazepan-4-yl)piperidine-4-carboxylate
{[3-(1-benzofuran-2-yl)-1H-pyrazol-4-yl]methyl}(methyl)(1,2-oxazol-3-ylmethyl)amine
2-{benzyl[5-(4-fluorophenyl)-1,2,4-triazin-3-yl]amino}ethan-1-ol
5-{1-[2-(2,2,3,3-tetrafluoropropoxy)acetyl]pyrrolidin-2-yl}thiophene-2-carboxamide
5-(dimethyl-1,2-oxazol-4-yl)-3-(oxolan-3-yl)-1,2,4-oxadiazole
N-{2-[3-(3,4-difluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-2-oxoethyl}methanesulfonamide
N-[(1-cyclopentylpiperidin-4-yl)methyl]-6-methyl-N-(pyridin-3-ylmethyl)pyridine-3-carboxamide
N-[2-(5-methyl-4-{[3-(1H-pyrazol-1-yl)propanamido]methyl}-1,3-oxazol-2-yl)phenyl]-3-phenoxypropanamide
(3R,4R)-1-[2-methyl-6-(1H-pyrazol-1-yl)pyrimidin-4-yl]-4-(morpholin-4-yl)piperidin-3-ol
3-(1-ethyl-2-methyl-1H-indol-5-yl)-1-(1-methanesulfonylpiperidin-4-yl)urea
[3-(2-phenylethyl)-1-[4-(1H-pyrazol-1-yl)benzoyl]piperidin-3-yl]methanol
2-{4-[(E)-2-cyclohexylethenyl]phenyl}-N,N-dimethylacetamide
N-[(4-chlorophenyl)methyl]-3-[2-(trifluoromethyl)morpholin-4-yl]propanamide
N-(2-fluorophenyl)-3-oxo-2-(pyridin-4-ylmethyl)-2,9-diazaspiro[5.5]undecane-9-carboxamide
3-(5-{1-[(1-ethylpiperidin-2-yl)methyl]-4-phenyl-1H-imidazol-5-yl}thiophen-2-yl)prop-2-yn-1-ol
3-[2-(5-methylfuran-2-yl)ethyl]-1-[4-(piperidine-1-carbonyl)phenyl]urea
(1R,5R)-6-methyl-3-[3-(piperidine-1-carbonyl)pyrazine-2-carbonyl]-3,6-diazabicyclo[3.2.2]nonane
1-[(1,3-dimethyl-1H-pyrazol-5-yl)methyl]-4-[(2-fluorophenyl)methyl]piperidine
3-(cyclopropylmethyl)-1-[3-(5-methyl-1H-1,2,4-triazol-3-yl)propanoyl]piperidine-3-carboxylic acid
1-{4-[(3-{1H,2H,3H,4H,5H-pyrido[4,3-b]indole-2-carbonyl}-1,2-oxazol-5-yl)methoxy]phenyl}-1H-1,2,4-triazole
2-{[5-(4-hydroxyphenyl)-4-(2-methoxy-5-methylphenyl)-4H-1,2,4-triazol-3-yl]sulfanyl}acetic acid
1-(1-cyclopropanecarbonylpiperidin-4-yl)-N-[2-(pyrazin-2-yl)ethyl]piperidine-3-carboxamide
3-methoxy-N-{[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-N,5-dimethylthiophene-2-carboxamide
(1R,7S)-3-[(4-fluorophenyl)methyl]-N-methyl-4-oxo-N-(pyrimidin-4-ylmethyl)-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
2,4-dimethoxy-N-{[7-methoxy-2-(morpholin-4-yl)quinolin-3-yl]methyl}-N-(oxolan-2-ylmethyl)benzamide
2-(4-{[4-(1,3-benzoxazol-2-yl)phenyl]carbamoyl}piperidin-1-yl)acetic acid
1-(4-benzylpiperidin-1-yl)-3-(5-cyclohexyl-1,3,4-oxadiazol-2-yl)propan-1-one
4-hydroxy-2-({[(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)methyl]amino}methyl)quinoline-6-carboxamide
1-cyclopentyl-N5-[(2,3-difluorophenyl)methyl]-N3-methyl-N3-(2-methylpropyl)-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
N-({6-cyclopentyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-2-(pyridin-3-yloxy)acetamide
1-{1-[4-(5-methyl-1,3,4-thiadiazol-2-yl)phenyl]ethyl}piperidine
1-methyl-5-{1-[(5-methylfuran-2-yl)methyl]-1H,4H-pyrazolo[3,4-d]imidazol-5-yl}-1H-imidazole
3-({[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]amino}methyl)-3-hydroxy-1-[(3-methylphenyl)methyl]piperidin-2-one
1-[5-(4-methoxyphenyl)-1,2,4-triazin-3-yl]-4-phenyl-1,4-diazepane
1-ethyl-N-(2-hydroxy-1-phenylethyl)-6-methyl-2-oxo-1,2-dihydropyridine-3-carboxamide