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4-[(4-cyclopentyl-1H-1,2,3-triazol-1-yl)methyl]-1-(oxolane-2-carbonyl)piperidine
4-[(3-methoxyphenyl)methyl]-1-(4-methylbenzoyl)-1,4-diazepan-5-one
N-methyl-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}-2-(1H-1,2,4-triazol-3-yl)benzamide
2,4-difluoro-N-{[4-(2-methylpropoxy)phenyl]methyl}-N-(pyridin-4-ylmethyl)benzene-1-sulfonamide
N-[(5-chlorothiophen-2-yl)methyl]-2-(4-methoxyphenyl)acetamide
N,N,4-trimethyl-5-{3-[(methylsulfanyl)methyl]piperidine-1-carbonyl}pyrimidin-2-amine
N-[(4-ethyl-2-methyl-1,3-thiazol-5-yl)methyl]-3-[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl]propanamide
2-(oxolan-2-ylmethyl)-9-(quinolin-4-yl)-2,9-diazaspiro[5.5]undecan-3-one
N-(2-{[(4-methyl-1H-imidazol-5-yl)methyl]sulfanyl}ethyl)-2-(4-oxo-3,4-dihydroquinazolin-3-yl)acetamide
2-(4-chloro-2-{[1-(2-hydroxyethyl)-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-5-yl]methyl}phenoxy)acetic acid
(3S,4S)-N-(3,4-difluorophenyl)-3-hydroxy-4-(4-methylpiperazin-1-yl)pyrrolidine-1-carboxamide
[2-(6-aminopyridin-3-yl)phenyl]methanol
1-[3-(hydroxymethyl)-3-(3-phenylpropyl)piperidin-1-yl]-3-(1H-1,2,4-triazol-1-yl)propan-1-one
4-{[(3-chloro-2,6-difluorophenyl)methyl]amino}-N-(propan-2-yl)pyridine-2-carboxamide
4-ethyl-3-{1-[3-(2-methylpropyl)-1,2-oxazole-5-carbonyl]piperidin-3-yl}-4,5-dihydro-1H-1,2,4-triazol-5-one
N-{[3-(2-methoxyphenyl)-1,2-oxazol-5-yl]methyl}-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
1-{6-chloroimidazo[1,2-a]pyrimidine-2-carbonyl}-3-[(dimethylamino)methyl]pyrrolidin-3-ol
[(3R,4R)-4-[(4-methylpiperazin-1-yl)methyl]-1-[4-(propan-2-yl)-1,2,3-thiadiazole-5-carbonyl]pyrrolidin-3-yl]methanol
(2R)-N-[2-(4-methyl-1H-1,3-benzodiazol-2-yl)ethyl]oxolane-2-carboxamide
4-phenyl-1-{pyrazolo[1,5-a]pyrimidin-3-ylmethyl}-1,2,3,6-tetrahydropyridine
N-{[2-(3,4-difluorophenoxy)pyridin-3-yl]methyl}pyrimidin-2-amine
5-[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]-3-phenyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
N-[2-(1-methylpiperidin-2-yl)ethyl]-6-[(oxan-4-ylmethyl)amino]pyridine-3-carboxamide
[(5-chloro-3-ethyl-1-methyl-1H-pyrazol-4-yl)methyl](methyl)[1-(pyrazin-2-yl)propan-2-yl]amine
4-phenyl-2-{[3-(2-phenylethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]methyl}-1,3-thiazole
2-(5-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-1H-1,2,3,4-tetrazol-1-yl)-N-ethyl-N-(pyridin-4-ylmethyl)acetamide
(4aS,8aR)-1-(3-methoxypropyl)-6-[(4-methyl-1H-imidazol-5-yl)methyl]-decahydro-1,6-naphthyridin-2-one
8-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-1-[2-(4-methoxyphenyl)ethyl]-3-(2-methylpropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-(3-hydroxyadamantan-1-yl)-1-(7-methanesulfonyl-4-methylquinazolin-2-yl)piperidine-4-carboxamide
1-[(1-methyl-1H-imidazol-4-yl)sulfonyl]-2-[2-(pyrrolidin-1-yl)ethyl]piperidine
3-[5-(4,5,6,7-tetrahydro-1,2-benzoxazole-3-carbonyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]propanoic acid
3-[(6,7-dimethoxy-1,2,3,4-tetrahydroisoquinolin-2-yl)methyl]-7-methyl-1-(2-phenoxyethyl)-1,2-dihydroquinolin-2-one
1-[3-({[2-(diethylamino)ethyl](methyl)amino}methyl)phenoxy]-3-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-2-ol
1-(6-chloro-2H-chromene-3-carbonyl)-3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidine
2-[8-(1,1-dioxo-1λ6-thiolane-3-carbonyl)-2-oxo-1-oxa-3,8-diazaspiro[4.5]decan-3-yl]acetic acid
N-[(4-methylphenyl)(pyridin-4-yl)methyl]-4-(trimethyl-1H-pyrazol-4-yl)pyrimidin-2-amine
2-(1-{[2-(4-methoxy-2,3-dimethylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-1H-pyrazol-4-yl)ethan-1-ol
(1R,7S)-3-(4-fluoro-2-methylphenyl)-6-[4-(propan-2-yl)piperazine-1-carbonyl]-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-en-4-one
1-[2-(dimethylamino)ethyl]-N-methyl-6-oxo-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}piperidine-3-carboxamide
N-{[4-(2-fluoro-4-methoxyphenyl)phenyl]methyl}acetamide
2-(dimethylamino)-N-{2-[3-(hydroxymethyl)piperidin-1-yl]ethyl}-4-methylpyrimidine-5-carboxamide
N-cyclobutyl-4-({[1-(prop-2-en-1-yl)pyrrolidin-3-yl]methyl}sulfamoyl)benzamide
2-(1,3-dimethyl-2,5-dioxoimidazolidin-4-yl)-N-[3-(1,2,3,4-tetrahydroquinolin-1-yl)propyl]acetamide
1-[(1R,5R)-6-[(5-methylthiophen-2-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-3-yl]ethan-1-one
N-[1-(2,4-difluorophenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-1H-indazole-3-carboxamide
3-{N-benzyl-1-[1-(4-fluorophenyl)-2,2-dimethylcyclopropyl]formamido}propanamide
2-ethoxy-N-(1-hydroxybutan-2-yl)-N-(pyridin-2-ylmethyl)pyridine-3-carboxamide
5-{[(4-methoxynaphthalen-1-yl)oxy]methyl}-N-(pyridin-2-ylmethyl)-1,2-oxazole-3-carboxamide
4-(4-{pyrazolo[1,5-a]pyridine-3-carbonyl}piperazin-1-yl)quinazoline
1-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}-3-(2,5-dimethoxyphenyl)pyrrolidine