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N-[(4-{[(2-fluorophenyl)methyl]amino}-8-methylquinazolin-2-yl)methyl]-6-methylpyridine-2-carboxamide
N-[4-(2-fluorophenoxy)phenyl]-3-(N-methylacetamido)pyrrolidine-1-carboxamide
3-(4-{4-ethyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidin-1-yl)propanoic acid
2-({2-[5-(4-methyl-1H-imidazol-5-yl)-4-phenyl-1H-imidazol-1-yl]ethyl}sulfanyl)pyridine
N-(2,1,3-benzothiadiazol-5-ylmethyl)-4-(pyridin-3-yl)pyrimidin-2-amine
9-methoxy-3-({6-methylimidazo[2,1-b][1,3]thiazol-5-yl}methyl)-10-(thiomorpholine-4-carbonyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepin-7-one
N-[2-(5-cyano-2-methyl-1H-indol-3-yl)ethyl]-2-[3-oxo-1-(propan-2-yl)piperazin-2-yl]acetamide
(3R,4S)-4-cyclopropyl-1-{[2-(2-methoxyethyl)pyrimidin-5-yl]methyl}pyrrolidin-3-amine
methyl 2-{[3-(3-methylthiophene-2-carbonyl)piperidine-1-carbonyl]amino}benzoate
5-(pyrrolidin-1-ylmethyl)-2-(3,4,5-trimethoxyphenyl)pyridine
(2S,4R)-N-methyl-4-[4-(2-methylpropyl)-1H-1,2,3-triazol-1-yl]pyrrolidine-2-carboxamide
N-{[7-(3,6-dimethylpyrazin-2-yl)-4-fluoro-2,3-dihydro-1-benzofuran-2-yl]methyl}-1H-1,3-benzodiazole-5-carboxamide
N3-(butan-2-yl)-N5-cyclohexyl-1-cyclopentyl-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
methyl 3-(2-chloro-4-fluorobenzoyl)-7-oxo-9-(pyridin-2-ylmethoxy)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
N-[2-(2-oxo-1,3-oxazinan-3-yl)ethyl]-2,3,4,5-tetrahydro-1-benzoxepine-4-carboxamide
6-{1-[(5-cyclopentylthiophen-2-yl)methyl]piperidin-4-yl}-2-methylpyrimidin-4-ol
N-(2,3-dihydro-1H-inden-2-yl)-2-[3-oxo-1-(pyridin-3-ylmethyl)piperazin-2-yl]acetamide
N5-(3-methoxypropyl)-N6-(1-phenylcyclopropyl)-[1,2,5]oxadiazolo[3,4-b]pyrazine-5,6-diamine
4-[(2-fluorophenyl)methyl]-1-[(4-phenyl-1,3-thiazol-2-yl)methyl]-1,4-diazepan-5-one
N-({1-[(3,7-dimethyl-1H-indol-2-yl)methyl]pyrrolidin-3-yl}methyl)methanesulfonamide
3-(1H-1,3-benzodiazol-1-yl)-N-methyl-N-{[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl}propanamide
(1S,5R)-6-(3-methylbut-2-en-1-yl)-3-[3-(pyridin-4-yl)propanoyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
N-[4-(1,3-thiazol-4-yl)phenyl]-1-[(trimethylpyrazin-2-yl)methyl]piperidine-3-carboxamide
3-{3-[(dimethylsulfamoyl)amino]phenyl}-1-(oxan-4-yl)urea
2-[(1S,5R)-6-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]-N,N-dimethylacetamide
(2S,3R)-2-amino-3-hydroxy-1-{4-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}butan-1-one
1-(5-chloropyridin-2-yl)-4-{5-[(methylsulfanyl)methyl]pyridin-2-yl}piperazine
N-[2-(4-ethylphenoxy)ethyl]-N,3-dimethyl-1H-pyrazole-4-carboxamide
2-methyl-8-[1-(pyridin-2-ylmethyl)piperidin-4-yl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid
3-{3-[methyl(2-methylpropyl)amino]propyl}-8-[(3-methyl-1,2-oxazol-5-yl)methyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
2-methoxy-6-({3-[4-(propan-2-yl)-1H-pyrazol-5-yl]piperidin-1-yl}methyl)phenol
N-[1-(1-{[4-(furan-2-yl)phenyl]methyl}piperidin-4-yl)-1H-pyrazol-5-yl]pyridine-3-carboxamide
N-methyl-N-(1,2,3,4-tetrahydronaphthalen-1-yl)-4-(4H-1,2,4-triazol-4-yl)benzamide
(1S,5R)-6-(5-propyl-1,2-oxazole-3-carbonyl)-3-(pyrazine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
8-[(4-hydroxyphenyl)methyl]-3-[(4-methoxyphenyl)methyl]-1-(3-methoxypropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
4-amino-2-[(3S,4S)-3-hydroxy-4-(naphthalen-2-yl)piperidin-1-yl]pyrimidine-5-carbonitrile
6-[(3S,4R)-3,4-dihydroxy-4-methylpiperidin-1-yl]pyridine-3-carboxamide
methyl 3-[2-(morpholin-4-yl)propanoyl]-7-oxo-9-[2-(thiophen-2-yl)ethoxy]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
2-[5-({2-[2-(thiophen-2-yl)ethyl]piperidin-1-yl}methyl)-1,2-oxazol-3-yl]pyridine
4-({1-[5-(phenoxymethyl)-1,2-oxazole-3-carbonyl]piperidin-3-yl}methyl)morpholine
N-{2-[2-(1,5-dimethyl-3-oxo-2-phenyl-2,3-dihydro-1H-pyrazol-4-yl)-1H-imidazol-1-yl]ethyl}acetamide
N-(3,4-difluorophenyl)-1-(4-methyl-1H-pyrrole-2-carbonyl)piperidin-3-amine
N-[1-(1-cyclopropanecarbonylpiperidin-4-yl)-1H-pyrazol-5-yl]-1-phenylmethanesulfonamide
[1-({[2-(pyridin-3-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl]amino}methyl)cyclobutyl]methanol
4-{1-[(2-chloro-4,5-dimethoxyphenyl)methyl]piperidin-3-yl}-5-(4-fluorophenyl)-2-methylpyrimidine
N-[4-methyl-2-(4H-1,2,4-triazol-4-yl)phenyl]benzamide
(3R,7S,8aS)-7-{[(2,4-difluorophenyl)methyl]amino}-3-methyl-octahydropyrrolo[1,2-a]piperazine-1,4-dione
2-(2,5-dimethylphenoxy)-N-[2-(1H-imidazol-1-yl)ethyl]propanamide
2-{2-chloro-4-[(7-methoxy-2,3,4,5-tetrahydro-1H-3-benzazepin-3-yl)methyl]phenoxy}acetamide
5-({8-methyl-octahydro-1H-pyrazino[1,2-a]piperazin-2-yl}methyl)-2-(propylsulfanyl)pyrimidine