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2-[3-(3-methoxybenzoyl)piperidin-1-yl]-3-(pyrrolidine-1-carbonyl)pyridine
N-[2-(3-phenylprop-2-ynoyl)-1,2,3,4-tetrahydroisoquinolin-7-yl]oxolane-2-carboxamide
1-[2-(4-methyl-1H-1,3-benzodiazol-2-yl)pyrrolidin-1-yl]-2-(methylamino)ethan-1-one
(2S)-2-amino-2-cyclohexyl-1-{2-phenyl-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}ethan-1-one
N-[2-(5-chloro-1H-1,3-benzodiazol-2-yl)ethyl]-2-[2-(2-methoxyphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]acetamide
N3-(2H-1,3-benzodioxol-5-ylmethyl)-1-(2-methoxyethyl)-4-oxo-N5-[1-(thiophen-2-yl)propyl]-1,4-dihydropyridine-3,5-dicarboxamide
(1R,3S,5S)-8-{[5-(pyrimidin-2-ylsulfanyl)furan-2-yl]methyl}-8-azabicyclo[3.2.1]octan-3-ol
3-amino-N-[(2R,3R)-2-(pyridin-3-ylmethoxy)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]propanamide
1-(3-phenylphenyl)-N-(pyrimidin-4-ylmethyl)piperidin-4-amine
9-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-2-(3-methoxypropyl)-2,9-diazaspiro[5.5]undecan-3-one
N-{1-[5-methyl-1-(naphthalen-1-yl)-1H-pyrazol-4-yl]ethyl}-3-(1H-1,2,3,4-tetrazol-1-yl)propanamide
N-(2,1,3-benzoxadiazol-5-ylmethyl)-N-methyl-2-[6-oxo-4-(pyrrolidin-1-yl)-1,6-dihydropyridazin-1-yl]acetamide
N-(4-fluorophenyl)-1-(1-methyl-1H-indole-2-carbonyl)piperidin-3-amine
methyl 2-oxo-1-(prop-2-en-1-yloxy)-8-(pyridin-3-ylmethyl)-1,8-diazaspiro[4.5]decane-4-carboxylate
2-methyl-N-(2-{2-methylimidazo[2,1-b][1,3,4]thiadiazol-6-yl}ethyl)-2,8-diazaspiro[4.5]decane-3-carboxamide
1-(4-chlorophenyl)-N-[(5-{[(4-fluorophenyl)methyl]sulfanyl}-4-methyl-4H-1,2,4-triazol-3-yl)methyl]cyclobutane-1-carboxamide
1-[1-(5-cyclopropyl-1,2-oxazole-3-carbonyl)piperidin-3-yl]-4-(4-fluorophenyl)piperazine
{[1-(cyclohexylmethyl)-2-methanesulfonyl-1H-imidazol-5-yl]methyl}(isoquinolin-5-ylmethyl)methylamine
1-(2-ethoxyethyl)-2-(3-fluorophenyl)piperidine
3-[5-(2H-1,3-benzodioxol-5-yl)-1,3,4-oxadiazol-2-yl]-N-[2-(2-fluorophenyl)ethyl]propanamide
2-[(4-chlorophenyl)methyl]-8-[(2S,4R)-4-hydroxypyrrolidine-2-carbonyl]-2,8-diazaspiro[4.5]decan-3-one
{[3-(2,4-difluorophenyl)-1H-pyrazol-4-yl]methyl}({[4-(1H-1,2,4-triazol-1-yl)phenyl]methyl})amine
1-{2-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl}-N-(2-hydroxy-2-phenylethyl)-N-methylpiperidine-4-carboxamide
N-(2-chloro-5-sulfamoylphenyl)-4-methyl-1,2,3,6-tetrahydropyridine-1-carboxamide
methyl 6-[(2E)-3-(4-chlorophenyl)prop-2-enoyl]-2-(cyclopropylsulfamoyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
2-(dimethylamino)-2-(3-methylphenyl)-N-{2-[(4-methylpyridin-2-yl)amino]ethyl}acetamide
N-[(5-methylfuran-2-yl)methyl]-3-(4,5,6,7-tetrahydro-1H-indazol-3-yl)propanamide
3-(4-ethyl-1,3-dimethyl-1H-pyrazol-5-yl)-1-[(1-methyl-1H-imidazol-2-yl)methyl]-1-propylurea
methyl[(3-methyl-1,2-oxazol-5-yl)methyl]{[1-methyl-3-(4-phenoxyphenyl)-1H-pyrazol-4-yl]methyl}amine
(3S,7S,8aS)-3-(4-aminobutyl)-7-[(thiophen-2-ylmethyl)amino]-octahydropyrrolo[1,2-a]piperazine-1,4-dione
1-{[(2-fluoro-4-methylphenyl)carbamoyl]methyl}-5-oxopyrrolidine-3-carboxylic acid
7-(2-hydroxyethyl)-2-[2-(2-oxoazepan-1-yl)acetyl]-2,7-diazaspiro[4.5]decan-6-one
N-(4-methoxy-2-methylphenyl)-3-{1-[2-(2-oxopiperidin-1-yl)acetyl]piperidin-3-yl}propanamide
4-{[(4-methylpyrimidin-2-yl)amino]methyl}azepan-4-ol
1-(3-{[4-(hydroxymethyl)phenyl]methyl}pyrrolidin-1-yl)-2-{5H,6H,7H-[1,3]thiazolo[3,2-a]pyrimidin-3-yl}ethan-1-one
1-{[4-(3-hydroxy-3-methylbutyl)phenyl]methyl}piperidine-3-carbonitrile
N-[3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)phenyl]-4-(pyrimidin-2-yl)-1,4-diazepane-1-carboxamide
(1R,3S)-3-{[3-(4-chlorophenyl)propyl]carbamoyl}cyclopentane-1-carboxylic acid
7-{[4-(propan-2-yl)phenyl]methyl}-2-[3-(trifluoromethyl)-1H-pyrazole-5-carbonyl]-2,7-diazaspiro[4.5]decane
(3S,4S)-1-[6-(2-fluorophenyl)imidazo[2,1-b][1,3]thiazole-3-carbonyl]-4-(pyrrolidin-1-yl)pyrrolidin-3-ol
1-(thiomorpholin-4-yl)-2-(2,4,7-trimethyl-1H-indol-3-yl)ethan-1-one
2-methyl-2-(thiophen-2-ylformamido)-N-(1H-1,2,4-triazol-5-ylmethyl)propanamide
N-[(3S,7S,8aS)-3-(2-methylpropyl)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-4-(trifluoromethyl)benzamide
1-(3-methyl-1-propyl-1H-pyrazole-4-carbonyl)-4-[3-(propan-2-yl)-1H-pyrazol-5-yl]piperidine
5-[1-(cyclohex-3-en-1-ylmethyl)piperidin-4-yl]-5-(pyridin-2-yl)-3-[2-(thiophen-2-yl)ethyl]imidazolidine-2,4-dione
(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-5-(3-methyl-1H-pyrazole-5-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
N-(4-{5-methyl-4-[(4,5,6,7-tetrahydro-2-benzothiophen-1-ylformamido)methyl]-1,3-oxazol-2-yl}phenyl)pyridine-3-carboxamide
3-methoxy-6-(3-{1-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-1H-pyrazol-3-yl}phenyl)pyridazine
1-benzyl-3-{2-[2-(hydroxymethyl)piperidin-1-yl]-2-oxoethyl}-3-(2-methylphenyl)pyrrolidine-2,5-dione
N-[1-(5-methyl-1,3,4-oxadiazol-2-yl)ethyl]-3-(morpholine-4-carbonyl)benzene-1-sulfonamide