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1-{5,7-dimethylpyrido[2,3-d]pyrimidin-4-yl}-3-(3-methylthiophene-2-carbonyl)piperidine
N-[3-(dimethylamino)-2,2-dimethylpropyl]-5-(methoxymethyl)-1-[4-(thiophen-2-yl)pyrimidin-2-yl]-1H-pyrazole-4-carboxamide
2-[4-(adamantan-2-yl)-1-[(2-methylphenyl)methyl]piperazin-2-yl]ethan-1-ol
1-{[3-(1-benzofuran-2-yl)-1-benzyl-1H-pyrazol-4-yl]methyl}piperidine-3-carbonitrile
2-[(2H-1,3-benzodioxol-5-yloxy)methyl]-N-[(2,5-difluorophenyl)methyl]-1,3-oxazole-4-carboxamide
5-(4-chlorophenyl)-N-methyl-N-(quinolin-2-ylmethyl)-1,2,4-triazin-3-amine
4-{3-[1-(3-fluoropropyl)-1H-pyrazol-3-yl]phenyl}-N,N,5,6-tetramethylpyrimidin-2-amine
1-[(5-{1-[1-(1,3-thiazol-2-yl)ethyl]-1H-1,2,3-triazol-4-yl}thiophen-3-yl)methyl]piperidine
4-benzyl-3-{1-[2-(1H-1,2,3,4-tetrazol-5-yl)acetyl]piperidin-4-yl}-4,5-dihydro-1H-1,2,4-triazol-5-one
1-methyl-N-({2-[(methylsulfanyl)methyl]-1,3-thiazol-4-yl}methyl)azepane-2-carboxamide
N-ethyl-N-({1-[2-(2-methylphenyl)ethyl]piperidin-4-yl}methyl)-2-(pyridin-2-yl)acetamide
4-[(2-methylpyridin-3-yl)oxy]-1-{[2-(propan-2-yl)-1,3-oxazol-4-yl]methyl}piperidine-4-carboxylic acid
3-(2-hydroxy-4,6-dimethylpyrimidin-5-yl)-1-[3-(hydroxymethyl)-3-(prop-2-en-1-yl)piperidin-1-yl]propan-1-one
N-(3-methoxypropyl)-1-[1-(pyridin-4-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
2-methoxy-5-{2-[5-(oxolan-2-yl)thiophen-2-yl]-1H-imidazol-1-yl}pyridine
(1S,6R)-3-methyl-9-[3-(propan-2-yl)-1H-pyrazole-5-carbonyl]-3,9-diazabicyclo[4.2.1]nonan-4-one
N-[1-(cyclohexylmethyl)piperidin-3-yl]-3-(1,2-oxazolidin-2-yl)propanamide
2-[(4-chlorophenyl)methyl]-8-(piperidin-3-yl)-2,8-diazaspiro[4.5]decan-3-one
2-amino-6-(2H-1,3-benzodioxol-5-yl)-4-(3-hydroxyphenyl)pyridine-3-carbonitrile
1,1-dioxo-N-propyl-N-(pyridin-3-ylmethyl)-1λ6-thiane-4-carboxamide
methyl 4-[(3-{3-oxo-3-[4-(pyridin-2-yl)piperazin-1-yl]propyl}piperidin-1-yl)methyl]benzoate
7-(cyclopropylmethyl)-2-[(3-ethenylphenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one
1-({3-[2-(morpholin-4-yl)ethoxy]phenyl}methyl)pyrrolidin-3-amine
N-[2-(4-hydroxypiperidin-1-yl)-7,7-dimethyl-5,6,7,8-tetrahydroquinazolin-5-yl]but-3-enamide
3-{[1-(2-hydroxyacetyl)piperidin-4-yl]oxy}-N-(2-phenylethyl)benzamide
(2R,3R,6R)-3-(2-methoxyphenyl)-5-(4-methyl-1H-imidazole-5-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
3-(3-{5-[(dimethylamino)methyl]-4-methyl-4H-1,2,4-triazol-3-yl}piperidine-1-carbonyl)pyridin-2-ol
1-({3-[(2-chlorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-2-ethylpiperidine
5-{1-[(2E)-3-(2,4-difluorophenyl)prop-2-enoyl]piperidin-4-yl}-5-methyl-3-[2-(morpholin-4-yl)ethyl]imidazolidine-2,4-dione
1-[(2-chlorophenyl)methyl]-N-[2-(2-methoxyphenyl)ethyl]-1H-1,2,3-triazole-4-carboxamide
N-(3-ethyl-4-methyl-1-phenyl-1H-pyrazol-5-yl)-2-(1,2,3,6-tetrahydropyridin-4-yl)acetamide
1-[4-(2,3-dihydro-1H-inden-2-yl)-1,4-diazepan-1-yl]-4-(1H-pyrazol-4-yl)butan-1-one
1-(3,5-dimethyl-4-{4-[3-(propan-2-yl)-1H-pyrazol-5-yl]piperidine-1-carbonyl}-1H-pyrrol-2-yl)ethan-1-one
1-[2-(4-methoxyphenyl)ethyl]-N,N-dimethyl-5-(quinoxalin-5-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
N-[5-({ethyl[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl]carbamoyl}amino)-2-methoxyphenyl]acetamide
N-{2-[7-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]ethyl}-4-fluorobenzamide
N-[(3-chlorophenyl)methyl]-4-{[1-(3-methoxypropanoyl)piperidin-4-yl]oxy}benzamide
N-[(1-methylpiperidin-4-yl)methyl]-N-(2-phenylethyl)-4-(4H-1,2,4-triazol-4-yl)benzamide
[(2S,4R,5R)-5-(2-fluorophenyl)-1-methyl-4-{[(quinolin-8-ylmethyl)amino]methyl}pyrrolidin-2-yl]methanol
dimethyl[(5-{[2-(2-methylphenyl)pyrimidin-5-yl]methyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl)methyl]amine
3-[(4-{1-[(1,2-dimethyl-1H-imidazol-5-yl)methyl]pyrrolidin-3-yl}piperidin-1-yl)methyl]pyridine
N-[2-(7-{[4-(pyrrolidin-1-yl)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)ethyl]oxolane-2-carboxamide
2-[4-(2,1,3-benzoxadiazol-5-ylmethyl)-1-[(3-methoxyphenyl)methyl]piperazin-2-yl]ethan-1-ol
2-{3-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyrimidine
3-(1-cyclopentyl-1H-pyrazol-5-yl)-1-[(3,4-difluorophenyl)methyl]urea
3-({1-[(4-fluorophenyl)methyl]pyrrolidin-2-yl}methyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-{[2-fluoro-5-(trifluoromethyl)phenyl]methyl}-3-(4-methylpiperazine-1-carbonyl)-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
{4-[(1-{3-fluoro-5-methylimidazo[1,2-a]pyridine-2-carbonyl}pyrrolidin-3-yl)methyl]phenyl}methanol
2-({3-[5-(hydroxymethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidin-1-yl}methyl)benzonitrile
N-{1,9-dioxaspiro[5.5]undecan-4-yl}-6-phenylpyridine-2-carboxamide