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2-[(3-methoxyphenyl)amino]-N-[2-(piperidin-1-yl)ethyl]butanamide
(2,1,3-benzothiadiazol-5-ylmethyl)({1-[2-(4-fluorophenyl)ethyl]piperidin-4-yl}methyl)methylamine
14-(2-cyclohexylpyrimidin-5-yl)-5-methyl-2,8,11-triazatricyclo[7.5.0.02,7]tetradeca-1(9),3,5,7-tetraen-12-one
N-{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}-6-oxo-1,6-dihydropyridine-3-carboxamide
1-[1-(2-methylpyrimidin-4-yl)piperidin-4-yl]-N-(pyridin-2-ylmethyl)piperidine-3-carboxamide
3-(2H-1,3-benzodioxol-5-ylmethyl)-9-methoxy-N-methyl-7-oxo-N-(1,3-thiazol-2-ylmethyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
(3R,4R)-3-methyl-4-(oxan-4-yl)-1-[4-(trifluoromethyl)pyridin-2-yl]piperidin-4-ol
4-[5-(4-phenylbutanamido)-1H-pyrazol-1-yl]-N-(prop-2-en-1-yl)piperidine-1-carboxamide
N-(2-fluorophenyl)-3-(1-{[2-(methylsulfanyl)pyrimidin-5-yl]methyl}piperidin-3-yl)propanamide
3-[3-(2,3-dimethoxyphenyl)pyrrolidine-1-carbonyl]-4,6-dimethyl-1,2-dihydropyridin-2-one
2-(dimethylamino)-8-(2-hydroxy-8-methylquinolin-3-yl)-4H,5H,6H,7H,8H-[1,3]thiazolo[4,5-c]azepin-6-one
2-[methyl(pyrazin-2-ylmethyl)amino]-2-[6-(piperidin-1-yl)pyridin-3-yl]acetic acid
3-(2-oxopyrrolidin-1-yl)-N-[1-(pyridin-2-yl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]benzamide
N-({1-[2-(4-methoxyphenyl)ethyl]piperidin-4-yl}methyl)-N-methylthiophene-3-carboxamide
2-[4-({3-[2-(2,6-difluorophenyl)ethyl]piperidin-1-yl}methyl)phenoxy]acetamide
ethyl 3-[(2-methylphenyl)methyl]-1-(1H-pyrazol-3-ylmethyl)piperidine-3-carboxylate
1-(3-cyano-4-ethoxyphenyl)-3-[2-(1-methyl-1H-pyrazol-5-yl)ethyl]urea
1-{4-[2-(2H-1,3-benzodioxol-5-yl)-5-fluoro-1H-1,3-benzodiazol-1-yl]piperidin-1-yl}-2-(3-methylphenyl)ethan-1-one
3-chloro-4-[(1-{[5-(hydroxymethyl)furan-2-yl]methyl}piperidin-4-yl)oxy]-N-(2-methoxyethyl)benzamide
(1R,3S)-N1,N1,2,2,3-pentamethyl-N3-{1-[(3-methylphenyl)methyl]cyclopropyl}cyclopentane-1,3-dicarboxamide
6-(3,5-dimethyl-1H-pyrrole-2-carbonyl)-3-(3-fluorophenyl)-1-[2-(piperidin-1-yl)ethyl]-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
2-{1-[(4-methylphenyl)methyl]-4-{[4-(pyrimidin-2-yloxy)phenyl]methyl}piperazin-2-yl}ethan-1-ol
1-[4-(2-methoxyphenyl)pyrimidin-2-yl]-5-methyl-N-[3-(morpholin-4-yl)propyl]-1H-pyrazole-4-carboxamide
N-[2-(3-methyl-1,2-oxazole-5-carbonyl)-1,2,3,4-tetrahydroisoquinolin-7-yl]-3-(4-methylphenyl)propanamide
1-(3-{[2-(2-hydroxyphenyl)-6-methylpyrimidin-4-yl]amino}propyl)pyrrolidin-2-one
N-{2-[(3,5-dimethyl-1H-pyrazol-4-yl)sulfanyl]phenyl}-1H-1,2,4-triazole-5-carboxamide
5-[1-(1-benzofuran-2-ylmethyl)piperidin-4-yl]-5-benzyl-3-(pyridin-3-ylmethyl)imidazolidine-2,4-dione
3-{[5-(methoxymethyl)pyrazolo[1,5-a]pyrimidin-7-yl](methyl)amino}propane-1,2-diol
N-(pentan-3-yl)-5-[4-(pyridin-3-yloxy)piperidine-1-carbonyl]pyridin-2-amine
{[2-fluoro-4-(trifluoromethyl)phenyl]methyl}(methyl)[2-(2-methyl-1H-imidazol-1-yl)ethyl]amine
methyl({[2-(trifluoromethyl)phenyl]methyl}){[3-(3,4,5-trimethoxyphenyl)-1H-pyrazol-4-yl]methyl}amine
2-chloro-N-({1-[2-(2-methoxyphenyl)ethyl]piperidin-4-yl}methyl)-N-methylpyridine-4-carboxamide
3-ethoxy-1-{2-phenyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}propan-1-one
(3R,4R)-1-(3-methoxybenzenesulfonyl)-3,4-dimethylpyrrolidin-3-ol
2-({4-[3-(3-chlorophenoxy)azetidine-1-carbonyl]phenyl}(methyl)amino)ethan-1-ol
5-cyclopropanecarbonyl-1'-(4-methylpyrimidine-5-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
5-chloro-3-[4-(4-phenyl-1H-pyrazol-5-yl)piperidine-1-carbonyl]-1,2-dihydropyridin-2-one
1-[(5-propylfuran-2-yl)methyl]-4-(pyrrolidine-1-sulfonyl)-1,4-diazepane
3-methyl-5-{[4-(4H-1,2,4-triazol-4-yl)phenyl]methyl}-4H-1,2,4-triazole
N-benzyl-6-[3-(pyridin-3-ylmethoxy)piperidin-1-yl]-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-amine
(2,1,3-benzothiadiazol-5-ylmethyl)(methyl)[(3-{[3-(trifluoromethyl)phenyl]methyl}-1,2,4-oxadiazol-5-yl)methyl]amine
2-{2-[1-(3-methylpyridin-4-yl)-3-(propan-2-yl)-1H-1,2,4-triazol-5-yl]pyrazolo[1,5-a]pyrimidin-6-yl}ethan-1-ol
1-[3-chloro-2-(propan-2-yloxy)phenyl]-3-[1-(4-methyl-1H-imidazol-2-yl)propyl]urea
N-cyclohexyl-2-{[1-(pyridine-3-carbonyl)piperidin-4-yl]oxy}benzamide
4-amino-N-{[2-(2-fluorophenoxy)pyridin-3-yl]methyl}butanamide
4-[2-(2-ethoxyphenoxy)ethyl]-1,3λ6,4-oxathiazinane-3,3-dione
N-(1H-1,3-benzodiazol-2-yl)-2-[(oxolan-2-ylmethyl)(pyridin-2-ylmethyl)amino]acetamide
3-benzyl-8-{[4-(dimethylamino)phenyl]methyl}-1-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-[2-(dimethylamino)ethyl]-2-(furan-2-yl)-N-({1-[(2-methoxyphenyl)methyl]piperidin-3-yl}methyl)-2-oxoacetamide
6-(2-cyanophenyl)-N,N-dimethylpyridine-3-carboxamide