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N-(dimethyl-1H-1,2,4-triazol-3-yl)-4-(4-methoxyphenyl)-3,3-dimethylpiperazine-1-carboxamide
2-(5-{4-[2-(methylsulfanyl)ethyl]piperazine-1-carbonyl}-1H-1,3-benzodiazol-1-yl)ethan-1-ol
N-(1,3-benzothiazol-2-yl)-3-[2-(pyridin-2-yl)pyrrolidin-1-yl]propanamide
3,6-dimethyl-4-[(E)-2-phenylethenyl]-[1,2]oxazolo[5,4-d]pyrimidine
N-{[1-(pyridin-2-ylmethyl)piperidin-3-yl]methyl}-3-(trifluoromethyl)benzamide
1-cyclopentyl-N-[2-(5-methyl-1,3,4-thiadiazol-2-yl)ethyl]-5-oxopyrrolidine-3-carboxamide
3-(3-chlorobenzoyl)-N-propylpiperidine-1-carboxamide
3-[1-(dimethylsulfamoyl)piperidin-4-yl]-N-(3-methoxyphenyl)propanamide
N-(1-{1-[(2,4,5-trimethylphenyl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)cyclopentanecarboxamide
2-(3-fluorophenyl)-N-({7-[(2-hydroxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)acetamide
4-(2,6-dimethylpyridin-3-yl)-N-methyl-N-[(3-methylpyridin-4-yl)methyl]pyrimidin-2-amine
1-[(3-methoxyphenyl)methyl]-N-{[1-(1,3-thiazol-2-yl)-1H-pyrrol-2-yl]methyl}piperidin-3-amine
2-{7-methylthieno[3,2-d]pyrimidin-4-yl}-1,2,3,4-tetrahydroisoquinolin-4-ol
8-[(2-methyl-1,3-oxazol-4-yl)methyl]-3-{2-[4-(propan-2-yl)piperazin-1-yl]ethyl}-1-oxa-3,8-diazaspiro[4.5]decan-2-one
4-[4-(cyclopropylmethyl)-3-(propan-2-yl)-1,4-diazepane-1-carbonyl]-N-methyl-1,3-thiazol-2-amine
3-fluoro-N-(1-hydroxybutan-2-yl)-2-methoxy-N-(thiophen-3-ylmethyl)benzamide
1-{3-[4-(4-fluorophenyl)piperazin-1-yl]piperidin-1-yl}-5-phenylpentan-1-one
2,3-dimethoxy-N-{[1-(1,2,4-oxadiazol-3-ylmethyl)piperidin-3-yl]methyl}benzamide
1-(3-fluorophenyl)-3-(1-{1-[(3-hydroxyphenyl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)urea
N-[4-(furan-2-yl)phenyl]-4-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]piperidine-1-carboxamide
N-[(2-fluorophenyl)methyl]-3-[1-(2-oxo-1,2,5,6,7,8-hexahydroquinoline-3-carbonyl)piperidin-3-yl]propanamide
5-[4-(dimethylamino)-5-fluoropyrimidin-2-yl]-N-methyl-4H,5H,6H,7H-thieno[3,2-c]pyridine-2-carboxamide
2-methyl-6-(1-{5-[(methylsulfanyl)methyl]furan-2-carbonyl}piperidin-3-yl)pyrimidin-4-ol
(4aR,8aS)-1-[(4-fluorophenyl)methyl]-6-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]-decahydro-1,6-naphthyridin-2-one
2-{8-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]-2,4-dioxo-1-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decan-3-yl}acetamide
2-{1-[(2-chloro-4-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-[(1-ethyl-1H-imidazol-2-yl)methyl]acetamide
(2S,4R)-1-[(3-chlorophenyl)methyl]-4-{[(2,6-difluorophenyl)methyl]amino}-N-(2-methoxyethyl)pyrrolidine-2-carboxamide
3-(4-methoxyphenyl)-3-phenyl-N-(pyridin-3-ylmethyl)propanamide
[(8-methoxyquinolin-5-yl)methyl](methyl){[2-(propan-2-yl)-1,3-oxazol-4-yl]methyl}amine
N-methyl-3-(4-methyl-1,3-thiazol-5-yl)-N-(1,2,3,4-tetrahydronaphthalen-1-yl)propanamide
4-({5-[2-(ethylsulfanyl)pyrimidin-5-yl]-4-phenyl-1H-imidazol-1-yl}methyl)-1,3-thiazol-2-amine
8-[(3-ethyl-1,2-oxazol-5-yl)methyl]-1-oxa-8-azaspiro[4.6]undecan-9-one
N-{[3-methyl-7-(2-phenoxyacetyl)-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}propane-1-sulfonamide
N-ethyl-3-methyl-N-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}-4-oxo-3,4-dihydroquinazoline-7-carboxamide
3-{1-[(5-chlorofuran-2-yl)methyl]piperidin-3-yl}-1-(4-methylpiperazin-1-yl)propan-1-one
2-methoxy-N-({3-methoxy-4-[2-(4-methyl-1,3-thiazol-5-yl)ethoxy]phenyl}methyl)-N-[(3S)-2-oxoazepan-3-yl]benzamide
{5-[(3-{methyl[2-(pyridin-2-yl)ethyl]amino}piperidin-1-yl)methyl]furan-2-yl}methanol
2-(1-cyclopentyl-3-oxopiperazin-2-yl)-N-methyl-N-(2-phenylethyl)acetamide
1-[3-(3-methyl-1H-pyrazol-1-yl)propanoyl]-4-{[3-(trifluoromethyl)phenyl]methyl}-1,4-diazepan-5-one
N-benzyl-N-[2-(dimethylamino)ethyl]-1-{2-[2-(2-fluorophenyl)ethyl]-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl}piperidine-4-carboxamide
[4-(5-chloro-7-methoxy-1-benzofuran-2-carbonyl)-1,4-oxazepan-6-yl]methanol
4-[6-(4-fluorophenyl)imidazo[2,1-b][1,3]thiazole-3-carbonyl]-1,2-dimethylpiperazine
N-[(3,4-dimethoxyphenyl)methyl]-2-[3-(3-fluorophenyl)-1-methyl-2,5-dioxopyrrolidin-3-yl]-N-methylacetamide
2-benzyl-8-[3-(dimethylamino)benzoyl]-2,8-diazaspiro[4.5]decan-3-one
N-[(2,4-dimethoxyphenyl)methyl]-3-{1-[(3-methylthiophen-2-yl)methyl]piperidin-3-yl}propanamide
dimethyl[({1-[(2Z)-5-methyl-2-phenylhex-2-en-1-yl]piperidin-3-yl}methyl)sulfamoyl]amine
N-(1-{imidazo[2,1-b][1,3,4]thiadiazol-6-yl}ethyl)-2,6,8-trimethylquinoline-4-carboxamide
N-({3-[(2-chloroprop-2-en-1-yl)oxy]-4-methoxyphenyl}methyl)-N-[(3S)-2-oxoazepan-3-yl]furan-2-carboxamide
3-{2-[4-(4-ethylpiperazin-1-yl)piperidin-1-yl]-2-oxoethyl}-4-[(2-fluorophenyl)methyl]piperazin-2-one
methyl 4-{[(1R,2S,6R,7S)-4-azatricyclo[5.2.2.02,6]undecane-4-carbonyl]amino}benzoate