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3-{2-[4-(benzyloxy)piperidin-1-yl]-2-oxoethyl}-1-(2-methoxyethyl)-3-(3-methoxyphenyl)pyrrolidine-2,5-dione
8-[2-(3-phenyl-1H-1,2,4-triazol-5-yl)acetyl]-2,8-diazaspiro[4.5]decan-3-one
N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]-4,5,6,7-tetrahydro-2-benzothiophene-1-carboxamide
2-[(2R)-2-(methoxymethyl)pyrrolidin-1-yl]-4-[1-(2-methylphenyl)-1H-pyrazol-4-yl]pyrimidine
5-(1H-1,3-benzodiazol-1-ylmethyl)-N-[2-methyl-1-(pyridin-3-yl)propyl]-1H-pyrazole-3-carboxamide
1-(2-cyclohexylethyl)-3-({[(1-ethyl-1H-imidazol-2-yl)methyl](methyl)amino}methyl)-3-hydroxypiperidin-2-one
N-[(4-fluorophenyl)methyl]-2-methoxy-N-(1-phenylethyl)acetamide
5-benzamido-1-cyclopentyl-N-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-N-methyl-1H-1,3-benzodiazole-7-carboxamide
5-methyl-N-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)-1,3,4-thiadiazol-2-amine
N-[2-(piperidin-1-yl)ethyl]-3-[(thiophen-2-ylmethyl)amino]benzamide
8-{[2-(2-fluoro-5-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-1-oxa-3,8-diazaspiro[4.5]decan-2-one
2-({4-[4-cyclopropyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}methyl)pyrimidine
N-({1-[2-(4-fluorophenyl)ethyl]piperidin-3-yl}methyl)-N,3,5-trimethyl-1,2-oxazole-4-carboxamide
2-(1-propoxyethyl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
4-{5-[4-(pyridin-3-yloxy)piperidine-1-carbonyl]pyridin-2-yl}phenol
4-[2-(1-{[2-(dimethylamino)-1,3-thiazol-5-yl]methyl}piperidin-2-yl)ethyl]phenol
N-{[1-(morpholin-4-yl)cyclopentyl]methyl}-5-[3-(trifluoromethyl)phenyl]-1,2,4-triazin-3-amine
(3S)-1-ethyl-4-{[3-(6-methoxynaphthalen-2-yl)-1H-pyrazol-4-yl]methyl}-3-methylpiperazin-2-one
(2R,3R,6R)-5-methanesulfonyl-3-(4-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
2-methyl-N-[3-(methylsulfanyl)propyl]-7-(pyrimidin-2-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
2-cyclopropyl-9-(3-phenoxypropyl)-2,9-diazaspiro[5.5]undecan-3-one
3-[(4-methyl-1,2,3,6-tetrahydropyridin-1-yl)methyl]benzoic acid
1,3-dimethyl-N-{3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]propyl}-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
(3S,4R)-1-[3-(2-ethyl-1H-imidazol-1-yl)propanoyl]-4-(4-fluorophenyl)pyrrolidine-3-carboxylic acid
1-{1-[2-methyl-2-(morpholin-4-yl)propyl]piperidin-3-yl}-3-phenylpropan-1-one
(2,3-dihydro-1-benzofuran-2-ylmethyl)({[2-(furan-2-yl)-5-methyl-1,3-oxazol-4-yl]methyl})methylamine
4-(5-methylpyridin-2-yl)-1-(5-phenyl-1H-pyrrole-2-carbonyl)piperidin-4-ol
methyl 9-[2-(2-fluorophenyl)ethoxy]-3-(2-methylpropyl)-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
N-(2-chlorophenyl)-3-[1-(pyridin-4-ylmethyl)piperidin-4-yl]propanamide
(3aR,6aS)-5-(4-methanesulfonylbenzoyl)-1-oxo-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-benzyl-2-[8-(cyclopropylmethyl)-9-oxo-2,8-diazaspiro[5.5]undecan-2-yl]acetamide
2-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl}-1H-indole
ethyl 4-[(4-methoxyphenyl)methyl]-1-[3-(1H-pyrazol-1-yl)propanoyl]piperidine-4-carboxylate
3-[1-(1,3-benzothiazol-2-ylmethyl)piperidin-3-yl]-N-methyl-N-[2-(pyridin-2-yl)ethyl]propanamide
5-{[5-(6-chloropyridin-3-yl)-4-phenyl-1H-imidazol-1-yl]methyl}-N-methylfuran-2-carboxamide
2-{2-[(3,4-difluorophenyl)methyl]-3-oxo-2,8-diazaspiro[4.5]decan-8-yl}propanamide
N-methyl-N-[4-(morpholin-4-yl)butyl]-6-(piperidin-1-yl)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-amine
4-[2-(4H-1,2,4-triazol-4-yl)ethyl]benzene-1-sulfonamide
N-[(1-ethylpyrrolidin-2-yl)methyl]-4-methoxy-3-{[1-(propan-2-yl)piperidin-4-yl]oxy}benzamide
2-{[3-(2-hydroxyethyl)-4-methylpiperazin-1-yl]methyl}-4-methoxyphenol
(1R,5R)-6-[4-(benzyloxy)butanoyl]-N,N-dimethyl-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
2,5-dimethyl-N-{[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]methyl}-[1,3]oxazolo[5,4-d]pyrimidin-7-amine
N-[(5-{[2-(piperidin-1-yl)pyrimidin-5-yl]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl)methyl]acetamide
N-[(6-hydroxypyrimidin-4-yl)methyl]-2-[1-(propan-2-yl)piperidin-4-yl]acetamide
3-[1-(1-phenoxypropan-2-yl)piperidin-4-yl]-1-(4-phenylpiperazin-1-yl)propan-1-one
N-({6-cyclopentyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-5-hydroxypyridine-2-carboxamide
5-[6-methyl-1-(propan-2-yl)-1H-pyrazolo[3,4-b]pyridin-4-yl]-3-(2-phenylethyl)-1H-1,2,4-triazole
2-{[methyl({[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]methyl})amino]methyl}quinolin-8-ol
(3R)-3,4,4-trimethyl-1-(3-methylpyrazin-2-yl)pyrrolidin-3-ol
methyl 1-[(3R,5S)-1-{[4-(propan-2-yl)phenyl]methyl}-5-[(thiophen-2-ylmethyl)carbamoyl]pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate